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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	Rauwolscine
Molecular formula	C21H26N2O3
IUPAC name	methyl (1S,15S,18S,19S,20S)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carboxylate
Molecular weight	354.45
Hydrogen bond acceptor	4
Hydrogen bond donor	2
XlogP	2.9
Synonyms	CHEMBL10347 DTXSID2045608 KBio2_004506 Methyl (16beta,17alpha,20alpha)-17-hydroxyyohimban-16-carboxylate Prestwick0_000577 SPBio_000919 SR-01000075289-6 yohimban-16-carboxylic acid, 17-hydroxy-, methyl ester, (16beta,17alpha,20alpha)- AB00514662 BRD-K77474816-003-05-9 BSPBio_003221 D0Z7EA GTPL223 KBioGR_000938 methyl hydroxy[?]carboxylate Prestwick3_000577 Spectrum3_001761 T4LJ7LU45W 20-alpha-Yohimban-16-beta-carboxylic acid, 17-alpha-hydroxy-, methyl ester Yohimban-16-carboxylicacid, 17-hydroxy-, methyl ester, (16b,17a,20a)- AKOS032948426 CHEBI:48562 DSSTox_GSID_45608 KBio1_000414 meso-Yohimbine NCGC00017260-06 SCHEMBL244514 Spectrum_001458 .alpha.-Yohimbine W1076 4CN-1422 BPBio1_000434 Corynanthidine EINECS 205-006-9 KBio2_007074 methyl (1S,15S,18S,19S,20S)-18-hydroxy-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carboxylate Prestwick1_000577 SPBio_002613 SR-01000075289-7 17-alpha-Hydroxy-20-alpha-yohimban-16-beta-carboxylic acid methyl ester Yohimban-16-carboxylic acid, 17-hydroxy-, methyl ester, (16beta,17alpha,20alpha)- (9CI) AC1LD7LA BRD-K77474816-003-09-1 CAS-131-03-3 DivK1c_000414 IDI1_000414 KBioSS_001938 MolPort-002-513-616 Spectrum4_000319 Tox21_110811 20alpha-Yohimban-16beta-carboxylic acid, 17alpha-hydroxy-, methyl ester (8CI) ZINC3977785 alpha-Yohimbine DSSTox_RID_81001 KBio2_001938 Mesoyohimbine NINDS_000414 SDCCGMLS-0066742.P001 SR-01000075289 131-03-3 Yohimban-16-carboxylic acid, 17-hydroxy-, methyl ester, (16-beta,17-alpha,20-alpha)- (9CI) BRD-K77474816-003-04-2 D02MFI GTPL136 KBio3_002721 methyl 17alpha-hydroxy-20alpha-yohimban-16beta-carboxylate Prestwick2_000577 Spectrum2_000870 SR-01000075289-8 17alpha-hydroxy-20alpha-yohimban-16beta-carboxylic acid methyl ester Yohimban-16-carboxylic acid, 17-hydroxy-, methyl ester, (17alpha,20alpha)- AJ-47559 BSPBio_000394 CCG-205170 DSSTox_CID_25608 Isoyohimbine Lopac0_001093 NCGC00017260-05 Rauwolscine (6CI,7CI) Spectrum5_001121 UNII-T4LJ7LU45W [3H]rauwolscine BDBM50026636 [ Show all ]
Inchi Key	BLGXFZZNTVWLAY-DIRVCLHFSA-N
Inchi ID	InChI=1S/C21H26N2O3/c1-26-21(25)19-15-10-17-20-14(13-4-2-3-5-16(13)22-20)8-9-23(17)11-12(15)6-7-18(19)24/h2-5,12,15,17-19,22,24H,6-11H2,1H3/t12-,15+,17+,18+,19+/m1/s1
PubChem CID	643606
ChEMBL	CHEMBL10347
IUPHAR	136, 223
BindingDB	50026636
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
26560	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
553395	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
553393	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
553394	5-hydroxytryptamine receptor 1E	P28566	HTR1E	Homo sapiens (Human)	365
553391	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
553392	5-hydroxytryptamine receptor 2B	P30994	Htr2b	Rattus norvegicus (Rat)	479
26551	Adenosine receptor A2b	P29276	Adora2b	Rattus norvegicus (Rat)	332
26545	Alpha-1A adrenergic receptor	O02824	ADRA1A	Oryctolagus cuniculus (Rabbit)	466
26553	Alpha-1A adrenergic receptor	P43140	Adra1a	Rattus norvegicus (Rat)	466
26559	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
26561	Alpha-1A adrenergic receptor	P18130	ADRA1A	Bos taurus (Bovine)	466
26557	Alpha-1B adrenergic receptor	P35368	ADRA1B	Homo sapiens (Human)	520
26548	Alpha-1D adrenergic receptor	P23944	Adra1d	Rattus norvegicus (Rat)	561
26555	Alpha-1D adrenergic receptor	P25100	ADRA1D	Homo sapiens (Human)	572
26549	Alpha-2A adrenergic receptor	Q28838	ADRA2A	Bos taurus (Bovine)	452
26552	Alpha-2A adrenergic receptor	Q60474	ADRA2A	Cavia porcellus (Guinea pig)	450
26558	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450
26546	Alpha-2B adrenergic receptor	P18089	ADRA2B	Homo sapiens (Human)	450
26543	Alpha-2C adrenergic receptor	P18825	ADRA2C	Homo sapiens (Human)	462
26556	Alpha-2C adrenergic receptor	P22086	Adra2c	Rattus norvegicus (Rat)	458

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