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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Beta-2 adrenergic receptor
Species	Rattus norvegicus (Rat)
Gene	Adrb2
Synonym	beta2-adrenoceptor Beta-2 adrenoreceptor Beta-2 adrenoceptor beta-2 adrenergic receptor beta 2-AR B2AR adrenoceptor beta 2, surface adrenergic receptor ADRBR ADRB2R Adrb-2 Gpcr7 [ Show all ]
Disease	N/A for non-human GPCRs
Length	418
Amino acid sequence	MEPHGNDSDFLLAPNGSRAPGHDITQERDEAWVVGMAILMSVIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGASHILMKMWNFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYVAITSPFKYQSLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRATHKQAIDCYAKETCCDFFTNQAYAIASSIVSFYVPLVVMVFVYSRVFQVAKRQLQKIDKSEGRFHAQNLSQVEQDGRSGHGLRSSSKFCLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIRANLIPKEVYILLNWLGYVNSAFNPLIYCRSPDFRIAFQELLCLRRSSSKTYGNGYSSNSNGRTDYTGEQSAYQLGQEKENELLCEEAPGMEGFVNCQGTVPSLSIDSQGRNCNTNDSPL
UniProt	P10608
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3754
IUPHAR	29
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
459236	Eticlopride	C17H25ClN2O3	340.848	4 / 2	3.1	Yes
459251	AC1N0YGA	C3H7NO4S	153.152	5 / 2	-4.7	Yes
459275	paroxetine	C19H20FNO3	329.371	5 / 1	3.5	Yes
11728	propranolol	C16H21NO2	259.349	3 / 2	3.0	Yes
13067	CHEMBL3230442	C27H38N2O9	534.606	10 / 5	N/A	No
14326	CHEMBL243266	C21H24N4O7	444.444	9 / 5	1.6	Yes
459389	CHEMBL287651	C17H23NO2	273.376	3 / 2	3.5	Yes
21609	CHEMBL543964	C16H16ClN3O	301.774	1 / 3	N/A	N/A
459414	CHEMBL43345	C17H17NO2	267.328	3 / 3	2.5	Yes
459416	sulpiride	C15H23N3O4S	341.426	6 / 2	0.6	Yes
459423	Arotinolol	C15H21N3O2S3	371.532	7 / 3	2.3	Yes
459571	oxprenolol	C15H23NO3	265.353	4 / 2	2.1	Yes
459604	fluvoxamine	C15H21F3N2O2	318.34	7 / 1	2.6	Yes
459616	CHEMBL276031	C19H26N2O	298.43	2 / 1	3.9	Yes
459621	CHEMBL62429	C19H30N2O3	334.46	4 / 2	3.9	Yes
45799	CHEMBL129190	C8H10FNO3	187.17	5 / 4	-0.5	Yes
46538	CHEMBL32470	C26H30N2O4	434.536	6 / 4	1.6	Yes
61596	CHEMBL3230447	C23H27NO8	445.468	9 / 5	N/A	N/A
68706	CHEMBL164145	C30H46N4O6	558.72	8 / 6	2.0	No
69363	practolol	C14H22N2O3	266.341	4 / 3	0.8	Yes
73178	CHEMBL1258452	C18H28N2O3	320.433	5 / 1	3.1	Yes
76052	CHEMBL3230436	C14H21NO6	299.323	7 / 4	N/A	N/A
459923	methionine zwitterion	C5H11NO2S	149.208	3 / 1	-1.2	Yes
459924	DL-Homocysteine	C4H9NO2S	135.181	4 / 3	-3.4	Yes
83600	CHEMBL287587	C8H10FNO3	187.17	5 / 4	-0.5	Yes
83966	CHEMBL349175	C32H52N6O6	616.804	10 / 8	1.3	No
87866	CL-316243	C20H18ClNNa2O7	465.794	8 / 2	N/A	N/A
98502	BRN 2116323	C13H20N2O3	252.314	4 / 3	0.6	Yes
460107	LY 344864 racemate	C21H22FN3O	351.425	3 / 2	3.8	Yes
99467	CHEMBL3247308	C16H25NO3	279.38	4 / 2	2.7	Yes
99469	CHEMBL3247309	C16H25NO3	279.38	4 / 2	2.7	Yes
99699	CHEMBL32670	C19H23ClN2O4	378.853	6 / 5	0.6	Yes
460121	acebutolol	C18H28N2O4	336.432	5 / 3	1.7	Yes
460136	CHEMBL516641	C35H52O4	536.797	4 / 0	10.0	No
460165	Remoxipride	C16H23BrN2O3	371.275	4 / 1	2.1	Yes
460223	desipramine	C18H22N2	266.388	2 / 1	4.9	Yes
113531	CHEMBL164146	C32H50N4O6	586.774	8 / 6	3.1	No
125779	CHEMBL363325	C10H10N2O5S	270.259	6 / 0	1.8	Yes
126284	CHEMBL3230445	C25H33ClN2O8	524.995	9 / 6	N/A	No
460382	139290-69-0	C22H28FNO3	373.468	5 / 1	3.9	Yes
127311	CHEMBL35459	C21H28N2O4	372.465	6 / 5	0.6	Yes
460404	RS-102221	C27H31F3N4O7S	612.621	12 / 3	2.7	No
460447	QUIPAZINE,8-Me	C14H17N3	227.311	3 / 1	2.4	Yes
135455	CHEMBL32115	C20H25ClN2O4	392.88	6 / 4	0.7	Yes
138245	ritodrine	C17H21NO3	287.359	4 / 4	2.3	Yes
138593	CHEMBL206100	C4H5N3O4	159.101	5 / 2	-0.9	Yes
460506	(S)-Metoprolol	C15H25NO3	267.369	4 / 2	1.9	Yes
460507	(R)-Metoprolol	C15H25NO3	267.369	4 / 2	1.9	Yes
460508	metoprolol	C15H25NO3	267.369	4 / 2	1.9	Yes
143989	Bunolol	C17H25NO3	291.391	4 / 2	2.4	Yes
460556	RS 67333	C19H29ClN2O2	352.903	4 / 1	3.8	Yes
148729	CHEMBL32590	C20H18ClNO7-2	419.814	8 / 2	1.7	Yes
149882	CHEMBL163154	C34H56N6O6	644.858	10 / 8	2.0	No
460619	CHEMBL303334	C15H20Br2N2O3	436.144	4 / 2	3.0	Yes
162146	isoproterenol	C11H17NO3	211.261	4 / 4	-0.6	Yes
163955	pindolol	C14H20N2O2	248.326	3 / 3	1.8	Yes
164655	CHEMBL33360	C20H26N2O4	358.438	6 / 4	0.1	Yes
165114	CHEMBL32586	C21H27ClN2O4	406.907	6 / 5	1.2	Yes
165494	CHEMBL3247310	C17H27NO4	309.406	5 / 2	1.9	Yes
166019	CHEMBL126347	C9H11F2NO3	219.188	6 / 4	0.1	Yes
166471	CHEMBL32391	C19H22Cl2N2O4	413.295	6 / 5	1.2	Yes
168050	CHEMBL1800936	C18H23NO4	317.385	5 / 5	2.5	Yes
169064	CHEMBL3230437	C21H27NO8	421.446	9 / 4	N/A	N/A
460736	D-HOMOCYSTEINE THIOLACTONE	C4H7NOS	117.166	3 / 1	-0.1	Yes
460742	Homocysteine thiolactone	C4H7NOS	117.166	3 / 1	-0.1	Yes
171812	thioridazine	C21H26N2S2	370.573	4 / 0	5.9	No
175142	CHEMBL166033	C34H54N4O6	614.828	8 / 6	4.2	No
460791	amitriptyline	C20H23N	277.411	1 / 0	5.0	Yes
460873	DL-CYSTINE	C6H12N2O4S2	240.292	8 / 4	-6.3	Yes
187100	CHEMBL1800961	C21H23NO3	337.419	4 / 4	3.9	Yes
189284	PD 109394	C18H23FN4O2	346.406	5 / 1	2.9	Yes
191587	haloperidol	C21H23ClFNO2	375.868	4 / 1	3.2	Yes
193170	CHEMBL348897	C32H50N6O6	614.788	10 / 6	1.3	No
195122	CHEMBL3230444	C27H37ClN2O9	569.048	10 / 5	N/A	No
195318	UNII-5Z64M7W0JM	C17H21NO4	303.358	5 / 5	2.0	Yes
195321	(R,S)-(-)-fenoterol	C17H21NO4	303.358	5 / 5	2.0	Yes
460963	Amosulalol	C18H24N2O5S	380.459	7 / 3	1.2	Yes
201097	CHEMBL2114952	C20H25NO7	391.42	8 / 4	N/A	N/A
201099	CHEMBL2115407	C20H25NO7	391.42	8 / 4	N/A	N/A
201625	CHEMBL33399	C19H22Br2N2O4	502.203	6 / 5	1.4	No
461009	atenolol	C14H22N2O3	266.341	4 / 3	0.2	Yes
208567	CHEMBL1800963	C22H25NO4	367.445	5 / 4	3.5	Yes
461070	Robalzotan BNAD 299 HCL	C18H23FN2O2	318.392	4 / 1	2.8	Yes
216831	CHEMBL3230438	C19H23NO7	377.393	8 / 5	N/A	N/A
219190	CHEMBL3247304	C15H22N2O4	294.351	5 / 3	0.7	Yes
223493	CHEMBL3247303	C16H24N2O3	292.379	4 / 3	1.3	Yes
461225	amisulpride	C17H27N3O4S	369.48	6 / 2	1.5	Yes
233354	CHEMBL285888	C19H22Cl2N2O4	413.295	6 / 5	1.2	Yes
461239	Levobetaxolol	C18H29NO3	307.434	4 / 2	2.8	Yes
461264	Salvinorin A	C23H28O8	432.469	8 / 0	2.5	Yes
492646	Higenamine glucoside	C22H27NO8	433.457	9 / 7	0.4	No
242683	CHEMBL417137	C20H24Cl2N2O4	427.322	6 / 4	1.4	Yes
461311	143797-63-1	C15H14N4O	266.304	2 / 2	1.5	Yes
243882	CHEMBL3230448	C21H26N2O8	434.445	9 / 6	N/A	No
244658	CHEMBL284520	C19H22Cl2N2O4	413.295	6 / 5	1.2	Yes
245231	CHEMBL143467	C14H23NO2	237.343	3 / 2	2.6	Yes
248901	CHEMBL32933	C19H23ClN2O4	378.853	6 / 5	0.6	Yes
251905	CHEMBL544427	C21H26ClNO5	407.891	6 / 3	3.6	Yes
255367	alprenolol	C15H23NO2	249.354	3 / 2	3.1	Yes
256413	CHEMBL32939	C19H23BrN2O4	423.307	6 / 5	0.7	Yes

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