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Check the ligand table for details.
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Ligand

Name	pindolol
Molecular formula	C14H20N2O2
IUPAC name	1-(1H-indol-4-yloxy)-3-(propan-2-ylamino)propan-2-ol
Molecular weight	248.326
Hydrogen bond acceptor	3
Hydrogen bond donor	3
XlogP	1.8
Synonyms	SMR000059120 Spectrum_001109 Tox21_110221 NINDS_000837 PDSP2_000759 Pindolol (JP15/USP/INN) Pindololum Prindolol (TN) EINECS 236-867-9 1-(1H-indol-4-yloxy)-3-[(propan-2-yl)amino]propan-2-ol HMS1568A22 2-Propanol, 1-(4-indolyloxy)-3-(isopropylamino)- HMS3369E14 523P869 KBio2_001589 AKOS015969756 LB-46 Blocklin L MLS002548891 BSPBio_000020 NCGC00015786-11 CCG-39223 D00513 (rs)-pindolol DL-LB 46 1-(1H-indol-4-yloxy)-3-(isopropylamino)propan-2-ol SPECTRUM1500488 SR-01000000027-4 Visken NCGC00024925-04 Oprea1_770884 Pectobloc (TN) Pindolol [USAN:USP:INN:BAN:JAN] Prestwick1_000090 Pynastin (TN) 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol FT-0630406 1-[1H-INDOL-4-YLOXY]-3-[ISOPROPYLAMINO]-2-PROPANOL HMS2091P20 3-indol-4-yloxy-1-[(methylethyl)amino]propan-2-ol HSDB 6539 AB00052072-11 KBio3_001693 Betapindol LP00955 Blocklin-L (TN) NCGC00015786-06 Calvisken NCGC00015786-16 (+-)-Pindolol DB00960 1-((1H-indol-4-yl)oxy)-3-(isopropylamino)propan-2-ol DSSTox_GSID_23476 SC-25688 Spectrum4_000479 ST50319990 [2-hydroxy-3-(1H-indol-4-yloxy)propyl](propan-2-yl)amine NCGC00024925-07 PDSP1_000771 Pinbetol (TN) Pindolol, United States Pharmacopeia (USP) Reference Standard Prestwick_397 Durapindol 1-(1H-Indol-4-yloxy)-3-[(1-methylethyl)amino]-2-propanol Glauco-Viskin 2-Propanol, 1-(1H-indol-4-yloxy)-3-(1-methylethyl)amino- HMS3262P12 5-21-03-00017 (Beilstein Handbook Reference) JZQKKSLKJUAGIC-UHFFFAOYSA-N AC1L1J1N L000006 Blockin L (TN) MFCD00010530 BRD-A97701745-001-09-5 NCGC00015786-09 Carvisken (TN) CS-4473 (1)-1-(1H-Indol-4-yloxy)-3-(isopropylamino)propan-2-ol DivK1c_000837 1-(1H-Indol-4-yloxy)-3-(isopropylamino)-2-propanol SPBio_001289 SR-01000000027 Tox21_110221_1 NCGC00015786-20 NSC-757276 PDSP2_000760 Pindolol (JP17/USP/INN) Pindololum [INN-Latin] Prinodolol EINECS 244-623-8 1-(4-Indolyloxy)-3-(isopropylamino)-2-propanol HMS1920H16 2-Propanol, 1-(indol-4-yloxy)-3-(isopropylamino)-, (+-)- HMS3712A22 KBio2_004157 AN-18448 LB46 Blocklin L (TN) MolPort-001-792-503 BSPBio_002193 NCGC00015786-13 CCRIS 9215 (+-)-4-(2-hydroxy-3-(isopropylamino)propoxy)indole D0F2PO DL-Pindolol 1-(1H-indol-4-yloxy)-3-(propan-2-ylamino)-propan-2-ol Spectrum2_001285 SR-01000000027-5 Visken (TN) NCGC00024925-05 P 0778 Pharmakon1600-01500488 Pindolol, >=98% (TLC), powder Prestwick2_000090 SAM002264631 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol((-)-Pindolol) Glauco-visken 13523-86-9 HMS2095A22 4-(2-Hydroxy-3-isopropylaminopropoxy)-indole HY-B0982 AB00052072_12 KBioGR_000958 Betapindol (TN) LS-122385 BPBio1_000022 NCGC00015786-07 Calvisken (TN) CHEMBL500 (+/-)-Pindolol-d7(iso-propyl-d7) Decreten 1-(1h-indol-4-yloxy)-3-((1-methylethyl)amino)-2-propano DSSTox_RID_77043 SCHEMBL5219 Spectrum5_001266 SW196641-3 NCGC00261640-01 PDSP1_000772 PINDOLOL,(-) Prindolol Durapindol (TN) 1-(1H-indol-4-yloxy)-3-[(1-methylethyl)amino]propan-2-ol GTPL91 2-Propanol, 1-(1H-indol-4-yloxy)-3-[(1-methylethyl)amino]- HMS3267K17 KBio1_000837 AC1Q1QC1 LB 46 Blocklin MLS000069496 BRN 1536506 NCGC00015786-10 CAS-13523-86-9 CTK8G2432 (R,S)-PINDOLOL DL-4-[2-Hydroxy-3-(isopropylamino)propoxy]indole 1-(1H-Indol-4-yloxy)-3-(isopropylamino)-2-propanol # SPBio_001959 SR-01000000027-2 Tox21_500955 NCGC00024925-03 NSC757276 Pectobloc Pindolol [USAN:INN:BAN:JAN] Prestwick0_000090 Pynastin EU-0100955 1-(Indol-4-yloxy)-3-(isopropylamino)-2-propanol HMS2089I21 21870-06-4 HMS502J19 AB00052072 KBio2_006725 BDBM50019443 Lopac0_000955 Blocklin-L NC00467 C07445 NCGC00015786-14 CHEBI:8214 (+-)-lb46 1-((1-Methylethyl)amino)-3-(4-indolyloxy)-2-propanol DSSTox_CID_3476 1-(1H-indol-4-yloxy)-3-(propan-2-ylamino)propan-2-ol SBI-0050929.P004 Spectrum3_000547 SR-01000000027-7 Z3376 NCGC00024925-06 P-6820 Pinbetol Pindolol, European Pharmacopoeia (EP) Reference Standard Prestwick3_000090 1-(1H-Indol-4-yloxy)-3-isopropylamino-propan-2-ol(pindolol) Glauco-Visken (TN) 2-Propanol, 1-(1H-indol-4-yloxy)-3-((1-methylethyl)amino)- HMS3259I07 4-(3-(Isopropylamino)-2-hydroxypropoxy)indole IDI1_000837 AB00052072_13 KBioSS_001589 Blockin L MCULE-7764948919 BRD-A97701745-001-05-3 NCGC00015786-08 Carvisken CPD000059120 (.+/-.)-Pindolol Decreten (TN) 1-(1H-Indol-4-yloxy)-3-((1-methylethyl)amino)-2-propanol DTXSID8023476 [ Show all ]
Inchi Key	JZQKKSLKJUAGIC-UHFFFAOYSA-N
Inchi ID	InChI=1S/C14H20N2O2/c1-10(2)16-8-11(17)9-18-14-5-3-4-13-12(14)6-7-15-13/h3-7,10-11,15-17H,8-9H2,1-2H3
PubChem CID	4828
ChEMBL	CHEMBL500
IUPHAR	91
BindingDB	50019443
DrugBank	DB00960
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
163940	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
163947	5-hydroxytryptamine receptor 1A	P19327	Htr1a	Rattus norvegicus (Rat)	422
163942	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
163944	5-hydroxytryptamine receptor 1B	P28334	Htr1b	Mus musculus (Mouse)	386
163949	5-hydroxytryptamine receptor 1B	P28564	Htr1b	Rattus norvegicus (Rat)	386
163957	5-hydroxytryptamine receptor 1B	O08892	HTR1B	Cavia porcellus (Guinea pig)	389
163945	5-hydroxytryptamine receptor 1D	P79400	HTR1D	Sus scrofa (Pig)	291
163950	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
163953	5-hydroxytryptamine receptor 1E	P28566	HTR1E	Homo sapiens (Human)	365
163962	5-hydroxytryptamine receptor 1F	P30939	HTR1F	Homo sapiens (Human)	366
163958	5-hydroxytryptamine receptor 2A	P28223	HTR2A	Homo sapiens (Human)	471
163951	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
163948	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
163959	5-hydroxytryptamine receptor 5A	P30966	Htr5a	Mus musculus (Mouse)	357
163954	5-hydroxytryptamine receptor 5B	P35365	Htr5b	Rattus norvegicus (Rat)	370
163956	5-hydroxytryptamine receptor 6	Q9R1C8	Htr6	Mus musculus (Mouse)	440
163946	5-hydroxytryptamine receptor 7	P50407	HTR7	Cavia porcellus (Guinea pig)	446
163961	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
556122	5-hydroxytryptamine receptor 7	P32305	Htr7	Rattus norvegicus (Rat)	448
163938	Beta-1 adrenergic receptor	P08588	ADRB1	Homo sapiens (Human)	477

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