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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
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GPCR

Name	Beta-1 adrenergic receptor
Species	Homo sapiens (Human)
Gene	ADRB1
Synonym	Adrenergic receptor beta 1 Adrb-1 ADRB1R adrenergic receptor beta 1-AR beta1-adrenoceptor beta-1 adrenoreceptor Beta-1 adrenoceptor B1AR beta-1 adrenergic receptor [ Show all ]
Disease	Heart failure; Cardiogenic shock Heart failure Glaucoma Diabetes Coronary artery disease Circulatory disorders Chronic open-angle glaucoma; Ocular hypertension Chronic open-angle glaucoma High blood pressure High blood pressure; Angina Hypertension Septic shock; Neurogenic shock Open-angle glaucoma; Ocular hypertension Migraine Maintenance of normal sinus rhythm Hypertension; Ventricular premature beats Hypertension; Heart arrhythmia Hypertension; Angina pectoris Hypertension; Angina Ventricular fibrillation Central and peripheral nervous diseases Acute supraventricular tachycardia Open-angle glaucoma Allergy; Sepsis Angina pectoris Angina pectoris; Hypertension Bronchodilator Cardiac arrhythmias [ Show all ]
Length	477
Amino acid sequence	MGAGVLVLGASEPGNLSSAAPLPDGAATAARLLVPASPPASLLPPASESPEPLSQQWTAGMGLLMALIVLLIVAGNVLVIVAIAKTPRLQTLTNLFIMSLASADLVMGLLVVPFGATIVVWGRWEYGSFFCELWTSVDVLCVTASIETLCVIALDRYLAITSPFRYQSLLTRARARGLVCTVWAISALVSFLPILMHWWRAESDEARRCYNDPKCCDFVTNRAYAIASSVVSFYVPLCIMAFVYLRVFREAQKQVKKIDSCERRFLGGPARPPSPSPSPVPAPAPPPGPPRPAAAAATAPLANGRAGKRRPSRLVALREQKALKTLGIIMGVFTLCWLPFFLANVVKAFHRELVPDRLFVFFNWLGYANSAFNPIIYCRSPDFRKAFQRLLCCARRAARRRHATHGDRPRASGCLARPGPPPSPGAASDDDDDDVVGATPPARLLEPWAGCNGGAAADSDSSLDEPCRPGFASESKV
UniProt	P08588
Protein Data Bank	N/A
GPCR-HGmod model	P08588
3D structure model	This predicted structure model is from GPCR-EXP P08588.
BioLiP	N/A
Therapeutic Target Database	T44068
ChEMBL	CHEMBL213
IUPHAR	28
DrugBank	BE0000172

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
974	CHEMBL3298692	C32H38N4O6	574.678	8 / 6	3.9	No
1012	CHEMBL2205816	C18H20N2O	280.371	3 / 1	1.8	Yes
1072	CHEMBL516056	C28H44N2O8S	568.726	10 / 6	N/A	No
1245	CHEMBL556022	C20H30Cl2N4O3S	477.445	7 / 5	N/A	N/A
1339	CHEMBL2261203	C29H36N4O5S2	584.75	8 / 4	3.9	No
2153	BDBM50097799	C29H32N4O6S2	596.717	10 / 6	3.3	No
2277	1-(cyclohexylmethyl)pyrrolidine	C11H21N	167.296	1 / 0	3.1	Yes
2925	CHEMBL418308	C35H32N4O3S2	620.786	8 / 3	6.0	No
3100	Prenalterol	C12H19NO3	225.288	4 / 3	1.4	Yes
3277	CHEMBL475389	C25H38N2O6S	494.647	8 / 5	2.5	Yes
3508	CHEMBL2348219	C25H35N3O6	473.57	7 / 5	2.3	Yes
4601	CHEMBL208352	C24H25ClN2O3	424.925	5 / 3	4.4	Yes
4638	CHEMBL351183	C18H24N4O2S	360.476	6 / 3	2.1	Yes
5075	CHEMBL104481	C29H42N4O4	510.679	6 / 5	4.1	No
5144	CHEMBL466923	C30H30N4O3	494.595	5 / 4	4.5	Yes
5189	CHEMBL498519	C25H24ClNO4	437.92	5 / 3	2.5	Yes
5274	CHEMBL279931	C19H21ClN2O	328.84	2 / 3	3.8	Yes
5275	CHEMBL25823	C19H21ClN2O	328.84	2 / 3	3.8	Yes
5277	CHEMBL282039	C19H21ClN2O	328.84	2 / 3	3.8	Yes
5283	CHEMBL26393	C19H21ClN2O	328.84	2 / 3	3.8	Yes
5527	CHEMBL3128185	C30H29FN4O2S	528.646	7 / 3	4.2	No
6386	CHEMBL7776	C20H26N2O5S	406.497	7 / 3	2.7	Yes
6464	CHEMBL443435	C29H41N3O10S	623.718	12 / 7	N/A	No
6668	CHEMBL1203989	C24H27ClN4O4S	503.014	6 / 5	N/A	No
463738	CHEMBL3633757	C26H24BrNO4	494.385	5 / 0	5.4	No
536144	CHEMBL3899832	C22H19N5O4	417.425	8 / 2	3.6	Yes
7284	CHEMBL1807874	C23H31N3O4S	445.578	7 / 4	2.2	Yes
7841	CHEMBL1078695	C30H31N3O2	465.597	4 / 3	4.6	Yes
8215	BW-723C86	C16H18N2OS	286.393	3 / 2	3.0	Yes
8577	CHEMBL585751	C27H38N4O8S	578.681	10 / 7	-2.2	No
8581	CHEMBL479530	C26H35Cl3N4O4S	606.0	7 / 7	N/A	No
8599	CHEMBL34406	C31H31N5O6S	601.678	11 / 3	3.4	No
9122	CHEMBL183611	C26H31N3O5	465.55	6 / 5	2.7	Yes
9406	CHEMBL100351	C30H34N4O8S2	642.742	11 / 5	-0.2	No
9622	CHEMBL1083053	C30H35N3O4	501.627	6 / 1	4.2	No
9856	AC-42	C20H31NO	301.474	2 / 0	5.2	No
10105	CHEMBL604333	C21H23F3N2O4	424.42	8 / 4	2.7	Yes
10436	SB 204070 hydrochloride	C19H27ClN2O4	382.885	6 / 1	3.5	Yes
10464	BDBM50097795	C25H27N5O5S	509.581	8 / 4	2.0	No
10591	CHEMBL39269	C30H28N4O4S	540.638	8 / 3	3.8	No
10656	CHEMBL350581	C18H23N3O3S	361.46	6 / 2	2.1	Yes
10719	CHEMBL3287723	C25H32O7	444.524	7 / 2	5.7	No
10894	CHEMBL1085837	C30H41NO7	527.658	8 / 5	N/A	No
11694	Propranolol, L-	C16H21NO2	259.349	3 / 2	3.0	Yes
11705	DEXPROPRANOLOL	C16H21NO2	259.349	3 / 2	3.0	Yes
11719	propranolol	C16H21NO2	259.349	3 / 2	3.0	Yes
11772	CHEMBL550445	C25H29N3O3S	451.585	5 / 4	3.9	Yes
11805	CHEMBL321957	C28H36N4O5S	540.679	8 / 4	4.0	No
11817	CHEMBL466713	C23H26N4O3	406.486	6 / 3	1.5	Yes
11892	CHEMBL551350	C26H30N2O5	450.535	6 / 4	3.2	Yes
11931	ESMOLOL	C16H25NO4	295.379	5 / 2	1.9	Yes
12228	CHEMBL516804	C26H28FNO4	437.511	6 / 3	2.3	Yes
12975	CHEMBL1204006	C25H30ClN3O2S	472.044	4 / 5	N/A	N/A
12998	CHEMBL67998	C33H38N4O5S	602.75	7 / 6	5.7	No
13132	CHEMBL506518	C32H50N2O8S	622.818	10 / 5	N/A	No
13272	CHEMBL526472	C23H22ClNO3S	427.943	5 / 3	2.6	Yes
13748	CHEMBL310679	C12H12N2O2	216.24	2 / 2	1.4	Yes
548035	spermidine	C7H19N3	145.25	3 / 3	-1.0	Yes
14076	CHEMBL3128199	C25H27FN4O2S	466.575	7 / 4	3.3	Yes
14149	CHEMBL184407	C24H27N3O6S3	549.675	9 / 4	3.2	No
14151	CHEMBL107382	C30H36F2N4O4	554.639	8 / 5	4.0	No
14243	180083-23-2	C32H32N4O3	520.633	6 / 0	5.6	No
14611	CHEMBL469884	C26H30N2O4	434.536	6 / 4	1.6	Yes
14730	CHEMBL109288	C19H26ClN3O3S	411.945	6 / 2	2.3	Yes
15120	CHEMBL289390	C19H23ClN4O7S3	551.044	11 / 5	0.2	No
15365	CHEMBL1089734	C28H27N3O2	437.543	4 / 3	4.0	Yes
15463	CHEMBL2205829	C19H19NO3	309.365	4 / 1	2.2	Yes
16055	CHEMBL63825	C31H29F3N6O5S	654.665	13 / 3	4.7	No
521955	AM-0902	C17H15ClN6O2	370.797	6 / 0	2.3	Yes
16428	CHEMBL29141	C10H12N2O3S	240.277	5 / 4	0.0	Yes
16495	FORMOTEROL FUMARATE HYDRATE	C23H30N2O9	478.498	10 / 7	N/A	No
16500	YM-08316	C23H30N2O9	478.498	10 / 7	N/A	No
16580	CHEMBL1257914	C26H28N4O3S	476.595	8 / 3	4.5	Yes
16677	CHEMBL101132	C27H33N5O6S	555.65	9 / 5	1.9	No
16785	Pipamperone	C21H30FN3O2	375.488	5 / 1	2.0	Yes
17139	CHEMBL2440659	C15H11FN4O2S	330.337	7 / 1	2.4	Yes
17166	CHEMBL490222	C30H27ClN2O5	531.005	6 / 4	3.4	No
17347	CHEMBL101606	C25H31N5O8S2	593.67	12 / 5	-1.9	No
17495	CHEMBL559486	C31H38N2O6S	566.713	7 / 4	4.2	No
17515	CHEMBL2348210	C25H35N3O6	473.57	7 / 5	2.3	Yes
17603	CHEMBL33155	C32H31FN6O6S	646.694	12 / 4	3.3	No
18020	CHEMBL264819	C25H28N4O5S2	528.642	8 / 5	2.4	No
18714	CHEMBL67416	C23H28N4O5S	472.56	9 / 4	1.9	Yes
18732	CHEMBL270964	C26H30N2O3	418.537	5 / 4	2.8	Yes
18885	CHEMBL497281	C26H26ClNO4	451.947	5 / 3	2.6	Yes
19305	CHEMBL453048	C27H31NO4	433.548	5 / 3	2.8	Yes
19569	CHEMBL3298325	C33H34N4O4	550.659	7 / 6	3.7	No
20353	CHEMBL3128187	C23H27N5O2	405.502	5 / 3	1.9	Yes
20601	CHEMBL104180	C21H23N3O3S	397.493	6 / 3	2.1	Yes
20830	CHEMBL1084656	C26H40N2O9S	556.671	11 / 6	N/A	No
21352	CHEMBL1684585	C23H26N4O2S	422.547	6 / 4	2.7	Yes
22062	CHEMBL2348205	C25H34BrN3O5	536.467	6 / 4	3.3	No
522147	CHEMBL3775436	C15H26ClNO3	303.827	4 / 3	N/A	N/A
522165	CHEMBL3775769	C15H26ClNO3	303.827	4 / 3	N/A	N/A
22157	CHEMBL250352	C21H25N3O3	367.449	6 / 2	2.5	Yes
22427	CHEMBL293818	C29H39N5O4S	553.722	7 / 4	3.6	No
22442	CHEMBL284612	C23H30N4O7S	506.574	10 / 6	-1.2	No
22947	CHEMBL383511	C24H25ClN2O3	424.925	5 / 4	2.3	Yes
23024	CHEMBL250579	C41H42N4O5	670.81	7 / 4	5.7	No
23116	CHEMBL1945292	C21H27N3O4S	417.524	7 / 5	1.2	Yes

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