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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	methylphenidate
Molecular formula	C14H19NO2
IUPAC name	methyl 2-phenyl-2-piperidin-2-ylacetate
Molecular weight	233.311
Hydrogen bond acceptor	3
Hydrogen bond donor	1
XlogP	0.2
Synonyms	Cotempla XR-ODT Rubifen (TN) DEA No. 1724 HY-B1091 Metadate ER (TN) Methyl alpha-phenyl-alpha-(2-piperidyl)acetate Methylfenidan AC1L1HJM Methylphenidylacetate hydrochloride Biphentin (TN) Phenidylate Centedrin (Salt/Mix) Ritalin LA Ritalin-SR D02PPN Tsentedrin EINECS 204-028-6 LS-565 Methyl .alpha.-phenyl-.alpha.-2-piperidinylacetate Methyl phenidate Methylin (TN) 2-Piperidineacetic acid, .alpha.-phenyl-, methyl ester Methylphenidate HCl alpha-Phenyl-alpha-(2-piperidyl)acetic acid methyl ester Metilfenidato [INN-Spanish] C07196 PMS-Methylphenidate CHEBI:84276 Ritcher works Daytrana (TN) GTPL7236 Metadate CD Methyl 2-phenyl-2-(piperidin-2-yl)acetate Methyl phenyl(2-piperidinyl)acetate # Methylphen 4311/B Ciba Methylphenidatum BCP18286 NCGC00248587-01 Centedein (Salt/Mix) Ritalin (Salt/Mix) Concerta (TN) CS-4657 SBI-0206868.P001 DTXSID5023299 Jornay PM (a.k.a. HLD200) Methyl (2-phenyl-2-(2-piperidyl)acetate) Methyl alpha-phenyl-alpha-2-piperidinylacetate Methylin .alpha.-Phenyl-2-piperidineacetic acid methyl ester METHYLPHENIDATE (SEE ALSO: METHYLPHENIDATE HYDROCHLORIDE, CAS 298-59-9, NTPNO 10266-R) AKOS022506757 MethyPatch BRD-A19585813-003-01-7 phenyl-piperidin-2-yl-acetic acid methyl ester Centedrine (Salt/Mix) Ritalin LA (TN) Ritaline D04999 Equasym (TN) Meridil Methyl .alpha.-phenyl-2-piperidine-acetate Methyl phenidyl acetate Methylin ER 2-Piperidineacetic acid, alpha-phenyl-, methyl ester Methylphenidate [INN:BAN] API0008866 Metilfenidato [Italian] Calocain Riphenidate CHEMBL796 Concerta, Methylin, Ritalin Rubifen DB00422 HSDB 3126 Metadate ER methyl 2-phenyl-2-piperidin-2-ylacetate methyl phenyl(piperidin-2-yl)acetate Methylphenidan AB01563134_01 Methylphenidatum [INN-Latin] BDBM50062912 NCI-C56280 Centedrin Ritalin (TN) d-methylphenidate HCl SCHEMBL37178 DUGOZIWVEXMGBE-UHFFFAOYSA-N L001307 Methyl .alpha.-phenyl-.alpha.-(2-piperidyl)acetate methyl alpha-piperid-2-ylphenylacetate Methylin (Salt/Mix) 113-45-1 Methylphenidate (USAN/INN) alpha-Phenyl-2-piperidineacetic acid methyl ester Metilfenidato C 4311 Plimasine Centredin Ritalin SR Ritaline (Salt/Mix) Daytrana FT-0700534 Metadate Methyl .alpha.-phenyl-2-piperidineacetate Methyl phenidylacetate Methylofenidan 298-59-9 (hydrochloride) Methylphenidate [USAN:INN:BAN] Attenta (TN) Motiron (TN) Centedein Ritalin Concerta [ Show all ]
Inchi Key	DUGOZIWVEXMGBE-UHFFFAOYSA-N
Inchi ID	InChI=1S/C14H19NO2/c1-17-14(16)13(11-7-3-2-4-8-11)12-9-5-6-10-15-12/h2-4,7-8,12-13,15H,5-6,9-10H2,1H3
PubChem CID	4158
ChEMBL	N/A
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
69035	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
69045	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
69031	5-hydroxytryptamine receptor 1E	P28566	HTR1E	Homo sapiens (Human)	365
69040	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
69032	5-hydroxytryptamine receptor 5A	P47898	HTR5A	Homo sapiens (Human)	357
69028	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
69037	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
69030	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
69029	Alpha-1B adrenergic receptor	P35368	ADRA1B	Homo sapiens (Human)	520
69043	Alpha-1D adrenergic receptor	P25100	ADRA1D	Homo sapiens (Human)	572
69034	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450
69036	Alpha-2B adrenergic receptor	P18089	ADRA2B	Homo sapiens (Human)	450
69039	Alpha-2C adrenergic receptor	P18825	ADRA2C	Homo sapiens (Human)	462
69046	D(1A) dopamine receptor	P21728	DRD1	Homo sapiens (Human)	446
69033	D(2) dopamine receptor	P14416	DRD2	Homo sapiens (Human)	443
69044	Muscarinic acetylcholine receptor M1	P11229	CHRM1	Homo sapiens (Human)	460
69038	Muscarinic acetylcholine receptor M2	P08172	CHRM2	Homo sapiens (Human)	466
69047	Muscarinic acetylcholine receptor M3	P20309	CHRM3	Homo sapiens (Human)	590
69041	Muscarinic acetylcholine receptor M4	P08173	CHRM4	Homo sapiens (Human)	479
69042	Muscarinic acetylcholine receptor M5	P08912	CHRM5	Homo sapiens (Human)	532

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