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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	Cipargamin
Molecular formula	C19H14Cl2FN3O
IUPAC name	(3R,3'S)-5,7'-dichloro-6'-fluoro-3'-methylspiro[1H-indole-3,1'-2,3,4,9-tetrahydropyrido[3,4-b]indole]-2-one
Molecular weight	390.239
Hydrogen bond acceptor	3
Hydrogen bond donor	3
XlogP	3.9
Synonyms	(1R,3S)-5,7-Dichloro-6-fluoro-3-methyl-2,3,4,9-tetrahydrospiro[indoline-3,1-pyrido[3,4-b]indol]-2-one BDBM50318666 DTXSID70152424 NITD-609 1252008-89-1 KAE609 SCHEMBL1306342 (1R,3S)-5'',7-Dichloro-6-fluoro-3-methyl-2,3,4,9-tetrahydrospiro-[beta-carboline-1,3''-indol]-2''(1''H)-one AKOS027253851 D0LI1C NCGC00263785-01 Z7Q4FWA04P (3R,3'S)-5,7'-dichloro-6'-fluoro-3'-methylspiro[1H-indole-3,1'-2,3,4,9-tetrahydropyrido[3,4-b]indole]-2-one GTPL9721 NITD609 (1'R,3'S)-5,7'-dichloro-6'-fluoro-2',3',4',9'-tetrahydro-3'-methylspiro[3H-indole-3,1'-[1H]pyrido[3,4-b]indol]-2(1H)-one Cipargamin [INN] KS-00000630 Spiro[3H-indole-3,1'-[1H]pyrido[3,4-b]indol]-2(1H)-one, 5,7'-dichloro-6'-fluoro-2',3',4',9'-tetrahydro-3'-methyl-, (1'R,3'S)- (1R,3S)-5',7-dichloro-6-fluoro-3-methyl-spiro[2,3,4,9-tetrahydropyrido[3,4-b]indole-1,3'-indoline]-2'-one AS-51977 DB12306 NITD 609 ZINC49037032 1193314-23-6 CHEMBL1082723 HY-14430 SB16518 (1'R,3'S)-5,7'-Dichloro-6'-fluoro-3'-methyl-2',3',4',9'-tetrahydrospiro[indoline-3,1'-pyrido[3,4-b]indol]-2-one AK203988 CS-7486 MolPort-039-337-269 UNII-Z7Q4FWA04P [ Show all ]
Inchi Key	CKLPLPZSUQEDRT-WPCRTTGESA-N
Inchi ID	InChI=1S/C19H14Cl2FN3O/c1-8-4-11-10-6-14(22)13(21)7-16(10)23-17(11)19(25-8)12-5-9(20)2-3-15(12)24-18(19)26/h2-3,5-8,23,25H,4H2,1H3,(H,24,26)/t8-,19+/m0/s1
PubChem CID	44469321
ChEMBL	CHEMBL1082723
IUPHAR	N/A
BindingDB	50318666
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
44187	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
44224	5-hydroxytryptamine receptor 2A	P28223	HTR2A	Homo sapiens (Human)	471
44205	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
44211	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
44208	Adenosine receptor A2a	P29274	ADORA2A	Homo sapiens (Human)	412
443414	Adenosine receptor A3	P0DMS8	ADORA3	Homo sapiens (Human)	318
44198	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
44227	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450
44229	Alpha-2B adrenergic receptor	P18089	ADRA2B	Homo sapiens (Human)	450
44210	Alpha-2C adrenergic receptor	P18825	ADRA2C	Homo sapiens (Human)	462
44231	B1 bradykinin receptor	P46663	BDKRB1	Homo sapiens (Human)	353
44214	B2 bradykinin receptor	P30411	BDKRB2	Homo sapiens (Human)	391
44196	Beta-1 adrenergic receptor	P08588	ADRB1	Homo sapiens (Human)	477
44185	Beta-2 adrenergic receptor	P07550	ADRB2	Homo sapiens (Human)	413
44194	Beta-3 adrenergic receptor	P13945	ADRB3	Homo sapiens (Human)	408
44188	Cannabinoid receptor 1	P21554	CNR1	Homo sapiens (Human)	472
44207	Cholecystokinin receptor type A	P32238	CCKAR	Homo sapiens (Human)	428
44225	Corticotropin-releasing factor receptor 1	P34998	CRHR1	Homo sapiens (Human)	444
44192	Corticotropin-releasing factor receptor 2	Q13324	CRHR2	Homo sapiens (Human)	411
44199	D(1A) dopamine receptor	P21728	DRD1	Homo sapiens (Human)	446

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