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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	B1 bradykinin receptor
Species	Homo sapiens (Human)
Gene	BDKRB1
Synonym	kinin B1 receptor bradykinin receptor BKR1 BK-1 receptor B1R B1BKR B1 receptor [ Show all ]
Disease	Diabetic macular edema Rheumatoid arthritis Pain Osteoarthritis
Length	353
Amino acid sequence	MASSWPPLELQSSNQSQLFPQNATACDNAPEAWDLLHRVLPTFIISICFFGLLGNLFVLLVFLLPRRQLNVAEIYLANLAASDLVFVLGLPFWAENIWNQFNWPFGALLCRVINGVIKANLFISIFLVVAISQDRYRVLVHPMASRRQQRRRQARVTCVLIWVVGGLLSIPTFLLRSIQAVPDLNITACILLLPHEAWHFARIVELNILGFLLPLAAIVFFNYHILASLRTREEVSRTRCGGRKDSKTTALILTLVVAFLVCWAPYHFFAFLEFLFQVQAVRGCFWEDFIDLGLQLANFFAFTNSSLNPVIYVFVGRLFRTKVWELYKQCTPKSLAPISSSHRKEIFQLFWRN
UniProt	P46663
Protein Data Bank	N/A
GPCR-HGmod model	P46663
3D structure model	This predicted structure model is from GPCR-EXP P46663.
BioLiP	N/A
Therapeutic Target Database	T58589
ChEMBL	CHEMBL4308
IUPHAR	41
DrugBank	BE0005831

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
348	CHEMBL603907	C20H20ClF2N7O2	463.874	8 / 2	3.1	Yes
669	CHEMBL210427	C27H25Cl2N3O4S	558.474	6 / 2	5.8	No
951	CHEMBL206982	C26H26F2N4O5S	544.574	10 / 1	2.9	No
2207	CHEMBL243432	C21H17BrN6O3	481.31	5 / 4	2.3	Yes
2986	CHEMBL208247	C26H26F2N4O3	480.516	8 / 1	3.6	Yes
4145	CHEMBL375288	C24H20Cl2N4O3	483.349	6 / 2	5.4	No
4254	CHEMBL387331	C21H20F2N2O4	402.398	6 / 2	2.4	Yes
4770	CHEMBL589819	C24H21ClF2N6O5	546.916	10 / 2	4.4	No
4950	CHEMBL452238	C33H42ClN3O5S	628.225	7 / 1	6.0	No
5021	CHEMBL380260	C27H32Cl2N4O4S	579.537	7 / 3	4.5	No
5195	CHEMBL2311187	C47H75N13O11	1002.21	14 / 11	-4.1	No
5196	CHEMBL2369827	C47H75N13O11	998.197	14 / 11	-4.1	No
5198	CHEMBL413382	C47H75N13O11	998.197	14 / 11	-4.1	No
6222	CHEMBL299164	C34H41N7O2	579.749	6 / 2	5.4	No
6312	CHEMBL591110	C20H23N5O3	381.436	5 / 3	0.7	Yes
6327	des-Arg10-Kallidin	C50H73N13O11	1032.21	14 / 11	-3.8	No
6599	CHEMBL232750	C21H17Cl2F4N3O4	522.278	9 / 2	4.0	No
7456	CHEMBL1939763	C22H23N3O4S	425.503	5 / 2	1.8	Yes
7610	CHEMBL208210	C31H28F2N4O3	542.587	8 / 1	5.4	No
8356	CHEMBL221998	C24H20Cl2N4O3	483.349	6 / 2	5.4	No
9244	Safotibant	C25H34N4O5S	502.63	7 / 1	1.6	No
10067	CHEMBL453338	C31H38N2O4S	534.715	5 / 1	5.0	No
557578	SCHEMBL10147804	C24H19ClF2N6O5	544.9	11 / 2	2.4	No
548001	CHEMBL3980627	C24H19ClF2N6O5	544.9	11 / 2	2.4	No
10810	CHEMBL447392	C33H43ClN4O5S	643.24	8 / 1	5.0	No
10940	CHEMBL227828	C29H29N3O4S	515.628	6 / 3	3.4	No
12010	CHEMBL1939920	C23H25N3O5S	455.529	6 / 3	1.0	Yes
12024	CHEMBL516783	C21H17FN2O4S	412.435	6 / 2	3.6	Yes
12075	CHEMBL426681	C32H30F2N4O3	556.614	8 / 1	5.1	No
12216	CHEMBL390916	C23H24Cl2N6O2	487.385	5 / 3	4.1	Yes
12902	913064-47-8	C29H29ClN4O2	501.027	4 / 0	4.4	No
12967	CHEMBL241935	C24H26BrClN6O2	545.866	5 / 2	4.2	No
13275	CHEMBL206246	C26H39N5O3S	501.69	6 / 2	2.3	No
14884	CHEMBL381372	C28H36F3N3O4S	567.668	9 / 2	3.6	No
15060	CHEMBL507168	C26H32Cl2N2O5S	555.511	6 / 3	4.0	No
15124	CHEMBL1210753	C32H36F3N3O3S	599.713	8 / 3	6.0	No
15171	CHEMBL386794	C36H48Cl2N5O5S+	733.77	7 / 1	5.2	No
15226	CHEMBL470693	C21H17ClN2O4S	428.887	5 / 2	4.1	Yes
15850	CHEMBL272491	C21H23F2NO4	391.415	6 / 2	3.8	Yes
15976	CHEMBL2372168	C50H72N18O11	1101.24	16 / 12	-3.8	No
15982	CHEMBL444431	C30H32Cl2N4O5S	631.569	7 / 3	4.5	No
16465	CHEMBL244284	C27H33BrClN7O2	602.962	6 / 2	4.2	No
17135	CHEMBL2440659	C15H11FN4O2S	330.337	7 / 1	2.4	Yes
17172	CHEMBL2372142	C50H79N15O11	1066.28	14 / 12	-3.6	No
17629	CHEMBL1777968	C28H36N4O5S	540.679	7 / 2	2.1	No
17793	CHEMBL379259	C25H30Cl2N4O4S	553.499	7 / 3	4.0	No
18255	CHEMBL412762	C33H35N3O5S	585.719	7 / 2	4.0	No
18264	CHEMBL1939770	C22H22N4O5S	454.501	6 / 3	0.3	Yes
19229	CHEMBL1835757	C32H32N2O3	492.619	4 / 1	5.4	No
19231	CHEMBL1934259	C32H32N2O3	492.619	4 / 1	5.4	No
19573	CHEMBL216618	C49H69N15O12S	1092.24	16 / 13	-5.6	No
20926	CHEMBL1956869	C34H46Cl2N5O5S+	707.732	8 / 1	4.6	No
20967	CHEMBL2016601	C33H38Cl2N4O3S	641.652	6 / 1	6.7	No
21799	CHEMBL390272	C26H19BrN6O3	543.381	5 / 4	4.0	No
22647	CHEMBL3038098	C59H91N19O13S	1306.56	18 / 15	-5.9	No
22698	CHEMBL381366	C29H38F3N3O3S	565.696	8 / 2	4.7	No
22794	8-Leu-9-des-arg-BK	C41H63N11O10	870.022	12 / 9	-3.6	No
23320	CHEMBL1788318	C35H48N6O2	584.809	5 / 2	6.3	No
23321	CHEMBL1744082	C35H48N6O2	584.809	5 / 2	6.3	No
24310	CHEMBL207000	C28H26F2N4O3	504.538	8 / 1	3.7	No
24698	CHEMBL1956722	C36H48Cl2N5O6S+	749.769	8 / 1	4.3	No
25113	CHEMBL2087036	C23H26Cl2N4O3S	509.446	5 / 1	2.9	No
25540	CHEMBL2087415	C23H29ClN4O4S	493.019	6 / 1	1.9	Yes
26205	RS 39604	C26H36ClN3O6S	554.099	9 / 2	3.1	No
27059	CHEMBL1834749	C31H33N5O2	507.638	5 / 1	4.3	No
28179	CHEMBL234296	C22H22F4N4O	434.439	8 / 2	4.2	Yes
28776	CHEMBL1956857	C36H45Cl2F3N6O8S	849.745	15 / 4	N/A	No
29429	CHEMBL2372164	C50H72N17O11+	1087.23	15 / 12	-4.1	No
29656	CHEMBL389054	C30H34F3N3O4S	589.674	9 / 3	4.5	No
30313	CHEMBL222156	C35H45Cl2N7O5S	746.749	8 / 3	4.0	No
558220	SCHEMBL10182621	C26H23ClF2N8O4	584.969	11 / 2	2.8	No
548222	CHEMBL3892284	C26H23ClF2N8O4	584.969	11 / 2	2.8	No
31306	CHEMBL256793	C21H23F2NO4	391.415	6 / 2	3.7	Yes
31314	CHEMBL487444	C23H24N4O4S	452.529	6 / 4	2.9	Yes
31967	CHEMBL1939949	C23H31ClN4O4S	495.035	6 / 1	2.1	Yes
31997	CHEMBL609157	C23H21ClF2N8O4	546.92	10 / 2	4.0	No
33118	CHEMBL1835766	C31H32N4O2	492.623	4 / 1	4.7	Yes
33284	CHEMBL498393	C23H31N5O3S	457.593	5 / 3	1.4	Yes
33447	CHEMBL388031	C22H21F5N4O	452.429	9 / 2	4.3	Yes
33987	CHEMBL160547	C31H28ClN5O4S	602.106	6 / 3	3.7	No
34186	CHEMBL1777880	C23H34N4O4S	462.609	6 / 2	0.9	Yes
35950	CHEMBL205093	C34H46Cl2N6O5S	721.739	9 / 2	3.8	No
36614	CHEMBL598868	C15H12ClF2N7O2	395.755	8 / 3	1.7	Yes
37354	CHEMBL2372151	C44H61N11O11	920.038	13 / 10	-3.7	No
558415	SCHEMBL10147835	C26H22ClF2N7O5	585.953	12 / 2	2.2	No
548322	CHEMBL3987084	C26H22ClF2N7O5	585.953	12 / 2	2.2	No
38018	CHEMBL404280	C25H23Cl2F3N4O5	587.377	10 / 2	5.0	No
38057	CHEMBL204562	C29H30F2N4O3	520.581	8 / 1	4.5	No
38376	CHEMBL196494	C24H23F3N4O2	456.469	7 / 3	4.2	Yes
38588	CHEMBL208386	C28H39N3O3S	497.698	5 / 2	3.9	Yes
41168	CHEMBL218605	C23H19F5N4O3	494.422	10 / 2	4.4	Yes
42232	CHEMBL525092	C30H34N4O5S	562.685	7 / 3	2.9	No
558605	SCHEMBL10147810	C25H21ClF2N6O5	558.927	11 / 2	2.8	No
548383	CHEMBL3910554	C25H21ClF2N6O5	558.927	11 / 2	2.8	No
43927	CHEMBL604999	C24H18ClF2N7O4	541.9	11 / 3	4.7	No
44231	Cipargamin	C19H14Cl2FN3O	390.239	3 / 3	3.9	Yes
44700	CHEMBL1939764	C24H27N3O5S	469.556	6 / 2	2.1	Yes
44732	CHEMBL496341	C26H37N3O5S	503.658	7 / 2	2.7	No
45091	CHEMBL298158	C35H42N6O2	578.761	5 / 2	6.5	No
45817	CHEMBL360500	C22H21N5O3	403.442	6 / 2	3.2	Yes

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