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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	pergolide
Molecular formula	C19H26N2S
IUPAC name	(6aR,9R,10aR)-9-(methylsulfanylmethyl)-7-propyl-6,6a,8,9,10,10a-hexahydro-4H-indolo[4,3-fg]quinoline
Molecular weight	314.491
Hydrogen bond acceptor	2
Hydrogen bond donor	1
XlogP	4.2
Synonyms	NCGC00017366-04 (6aR,9R,10aR)-9-(Methylthiomethyl)-7-propyl-4,6,6a,7,8,9,10,10a-octahydroindolo[4,3-fg]quinoline P2200 5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid (10b-hydroxy-5-isobutyl-2-isopropyl-3,6-dioxo-octahydro-oxazolo[3,2-a]pyrrolo[2,1-c]pyrazin-2-yl)-amide Pergolidum [INN-Latin] 9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinoline, mesylate (Pergolide) SCHEMBL26921 AN-599 SR-01000721840 BRD-K60770992-001-01-8 CCG-205064 D08339 IDI1_000442 KBioSS_002127 NCGC00017366-10 (8beta)-8-[(methylsulfanyl)methyl]-6-propylergoline 66104-22-1 Prestwick0_000295 AB00053740_14 Spectrum2_001970 BDBM50028421 TNP00315 BSPBio_000230 DivK1c_000442 KBio2_002127 LY 141B (2R,4R,7R)-4-[(methylsulfanyl)methyl]-6-propyl-6,11-diazatetracyclo[7.6.1.0;{2,7}.0;{12,16}]hexadeca-1(16),9,12,14-tetraene NCGC00142538-03 24MJ822NZ9 Pergolide [INN:BAN] 9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinoline Prestwick3_000295 AC1Q7DT2 Spectrum5_001649 BPBio1_000254 ZINC3786466 C07425 D-8beta-[(Methylthio)methyl]-6-propylergoline GTPL48 KBio3_002656 NCGC00017366-02 NCGC00017366-05 (6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinolin-7-ium Pergolida Permax 9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinoline; compound with methanesulfonic acid SPBio_002099 BCP18331 SR-01000721840-8 BRD-K60770992-066-05-2 CHEBI:63617 InChI=1/C19H26N2S/c1-3-7-21-11-13(12-22-2)8-16-15-5-4-6-17-19(15)14(10-20-17)9-18(16)21/h4-6,10,13,16,18,20H,3,7-9,11-12H2,1-2H3/t13-,16-,18-/m1/s Lopac0_000984 NCGC00142538-01 (8beta)-8-[(methylthio)methyl]-6-propylergoline Pergolide (INN) 66104-23-2 (mesylate) Prestwick1_000295 AB00053740_15 Spectrum3_001588 BIDD:GT0177 UNII-24MJ822NZ9 BSPBio_003156 CHEMBL531 DTXSID2023438 KBio2_004695 LY-127,809 (2R,4R,7R)-4-[(methylsulfanyl)methyl]-6-propyl-6,11-diazatetracyclo[7.6.1.0^{2,7}.0^{12,16}]hexadeca-1(16),9,12,14-tetraene NINDS_000442 Pergolidum 9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinoline(pergolide) SBI-0050957.P003 AJ-45611 Spectrum_001647 BPBio1_001211 [2-(1H-Indol-4-yl)-ethyl]-methyl-amine CC-33590 D04JCN HMS2089C18 KBioGR_001409 NCGC00017366-03 NCGC00017366-06 (6aR,9R,10aR)-9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinoline Pergolida [INN-Spanish] Permax (TN) AB00053740-13 SPBio_002449 BDBM50017543 ST057534 BRD-K60770992-066-15-1 CHEMBL1275 DB01186 KBio1_000442 LS-64479 NCGC00142538-02 104P221 Pergolide Methanesulfonate 9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10a-octahydro-indolo[4,3-fg]quinolin-7-ium(Pergolide) Prestwick2_000295 AC1L2IT3 Spectrum4_000835 Biomol-NT_000025 YEHCICAEULNIGD-MZMPZRCHSA-N C-19410 cid_47811 Ergoline, 8-((methylthio)methyl)-6-propyl-, (8beta)- KBio2_007263 LY-127809 [ Show all ]
Inchi Key	YEHCICAEULNIGD-MZMPZRCHSA-N
Inchi ID	InChI=1S/C19H26N2S/c1-3-7-21-11-13(12-22-2)8-16-15-5-4-6-17-19(15)14(10-20-17)9-18(16)21/h4-6,10,13,16,18,20H,3,7-9,11-12H2,1-2H3/t13-,16-,18-/m1/s1
PubChem CID	47811
ChEMBL	CHEMBL531
IUPHAR	48
BindingDB	50017543, 50028421
DrugBank	DB01186
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
408055	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
408077	5-hydroxytryptamine receptor 1A	P19327	Htr1a	Rattus norvegicus (Rat)	422
408053	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
408061	5-hydroxytryptamine receptor 1B	P28564	Htr1b	Rattus norvegicus (Rat)	386
408078	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
408054	5-hydroxytryptamine receptor 2A	P35363	Htr2a	Mus musculus (Mouse)	471
408062	5-hydroxytryptamine receptor 2A	P28223	HTR2A	Homo sapiens (Human)	471
408064	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
408071	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
408070	5-hydroxytryptamine receptor 6	P31388	Htr6	Rattus norvegicus (Rat)	436
408079	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
555319	5-hydroxytryptamine receptor 7	P32305	Htr7	Rattus norvegicus (Rat)	448
557182	5-hydroxytryptamine receptor 7	P50407	HTR7	Cavia porcellus (Guinea pig)	446
408058	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
457903	Alpha-1A adrenergic receptor	P43140	Adra1a	Rattus norvegicus (Rat)	466
408069	Alpha-1B adrenergic receptor	P15823	Adra1b	Rattus norvegicus (Rat)	515
408083	Alpha-1B adrenergic receptor	P35368	ADRA1B	Homo sapiens (Human)	520
408067	Alpha-1D adrenergic receptor	P25100	ADRA1D	Homo sapiens (Human)	572
408074	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450
408060	Alpha-2B adrenergic receptor	P18089	ADRA2B	Homo sapiens (Human)	450

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