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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	quipazine
Molecular formula	C13H15N3
IUPAC name	2-piperazin-1-ylquinoline
Molecular weight	213.284
Hydrogen bond acceptor	3
Hydrogen bond donor	1
XlogP	1.5
Synonyms	Quipazine [INN] AC1Q1I54 SPBio_001223 AS-38262 TC-071714 BRD-K77925998-332-03-8 CHEMBL18772 GTPL173 KBioGR_001818 MCULE-2654170894 2-(1-piperazinyl)-quinoline NCGC00024694-02 2-Piperazin-1-ylquinoline Prestwick2_000617 AB00053761 RP26765 AK-26012 Spectrum3_001824 Biomol-NT_000103 UNII-4WCY05C0SJ BSPBio_003467 DB-021505 KBio1_000911 L000958 1-(2-Quinolyl)piperazine NCGC00015872-02 2-(piperazin-1-yl)-quinoline Oprea1_342540 4WCY05C0SJ Quinoline, 2-(1-piperazinyl)- AB00053761_12 AC-22858 SBI-0050992.P003 AMOT0412 ST50232723 BRD-K77925998-001-01-3 XRXDAJYKGWNHTQ-UHFFFAOYSA-N CHEBI:93368 F3306-0004 KBio2_007349 LS-142110 NCGC00015872-06 2-Piperazin-1-yl-quinoline (Quipazine) Prestwick0_000617 5786-68-5 (maleate (1:1)) Quipazina [INN-Spanish] Quipazinum AC1Q4WAV SPBio_002773 BAS 00505227 Tocris-0629 BRN 0196945 CTK4J0220 IDI1_000911 KBioSS_002213 MolPort-000-006-267 2-(1-Piperazinyl)chinolin NCGC00024694-03 2-quinolylpiperazine Prestwick3_000617 AB00053761-06 AB0076939 S14-1965 AKOS000124312 Spectrum4_001259 BPBio1_000610 VQ10136 CAS-4774-24-7 DivK1c_000911 KBio2_002213 Lopac-Q-1004 1-(quinolin-2-yl)piperazine NCGC00015872-03 2-(piperazin-1-yl)quinoline P67440 5-23-03-00069 (Beilstein Handbook Reference) Quinoline,2-(1-piperazinyl)- AC1L1JEX SCHEMBL322181 ANW-66727 STL308727 BRD-K77925998-050-02-8 ZINC2020 FT-0635438 KBio3_002971 MA-1291 2-(1-PIPERAZINO)QUINOLINE NCGC00024694-01 2-Piperazin-1-yl-quinoline(Quipazine) Prestwick1_000617 774P247 Quipazinum [INN-Latin] AJ-73031 Spectrum2_001182 BDBM50014407 TPC-A004 BSPBio_000554 D08BCF KB-25984 L-2584 1-(2-Quinolinyl)piperazine NCGC00015872-01 2-(1-Piperazinyl)quinoline NINDS_000911 4774-24-7 Q-103520 AB00053761_11 AB05466 SBB011283 AM20061242 Spectrum_001733 BPBio1_001393 VU0005330-3 CCG-205099 DTXSID3046952 KBio2_004781 Lopac0_001019 130895-61-3 NCGC00015872-04 2-Piperazin-1-yl-quinoline piperazin-1-yl-quinoline Quipazina [ Show all ]
Inchi Key	XRXDAJYKGWNHTQ-UHFFFAOYSA-N
Inchi ID	InChI=1S/C13H15N3/c1-2-4-12-11(3-1)5-6-13(15-12)16-9-7-14-8-10-16/h1-6,14H,7-10H2
PubChem CID	5011
ChEMBL	CHEMBL18772
IUPHAR	173
BindingDB	50014407
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
399353	5-hydroxytryptamine receptor 1A	P19327	Htr1a	Rattus norvegicus (Rat)	422
399365	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
399355	5-hydroxytryptamine receptor 1B	P28564	Htr1b	Rattus norvegicus (Rat)	386
399374	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
399364	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
399371	5-hydroxytryptamine receptor 1D	P79400	HTR1D	Sus scrofa (Pig)	291
399362	5-hydroxytryptamine receptor 2A	P28223	HTR2A	Homo sapiens (Human)	471
399366	5-hydroxytryptamine receptor 2A	P14842	Htr2a	Rattus norvegicus (Rat)	471
399372	5-hydroxytryptamine receptor 2A	Q75Z89	HTR2A	Bos taurus (Bovine)	470
399354	5-hydroxytryptamine receptor 2B	P30994	Htr2b	Rattus norvegicus (Rat)	479
399361	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
557147	5-hydroxytryptamine receptor 2B	Q02152	Htr2b	Mus musculus (Mouse)	479
399356	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
399357	5-hydroxytryptamine receptor 2C	P08909	Htr2c	Rattus norvegicus (Rat)	460
399363	5-hydroxytryptamine receptor 4	O70528	HTR4	Cavia porcellus (Guinea pig)	388
399367	5-hydroxytryptamine receptor 4	Q62758	Htr4	Rattus norvegicus (Rat)	406
399375	5-hydroxytryptamine receptor 5A	P30966	Htr5a	Mus musculus (Mouse)	357
399369	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
399376	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
557145	5-hydroxytryptamine receptor 7	P32305	Htr7	Rattus norvegicus (Rat)	448

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