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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	venlafaxine
Molecular formula	C17H27NO2
IUPAC name	1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol
Molecular weight	277.408
Hydrogen bond acceptor	3
Hydrogen bond donor	1
XlogP	2.9
Synonyms	D0P1UX Wy 45030 EC 618-944-2 HMS2093A12 KBio2_007287 N,N,O-Didesmethylvenlafaxine 1-[2-dimethylamino-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol NCGC00095109-06 AB00053751-11 SC-25322 AN-14846 Spectrum4_001115 BSPBio_002657 Tox21_111425 CHEMBL637 Venlafaxine (INN) Venlafaxine [INN:BAN] DL-Venlafaxine Elafax HY-B0196 KBioSS_002151 NCGC00095109-01 NSC758676 AB1004809 SPBio_000583 AX8023170 SR-01000762930 CAS_93413-69-5 Venlafaxin Cyclohexanol, 1-(2-(dimethylamino)-1-(4-methoxyphenyl)ethyl)-, (+-)- Venlafaxinum [INN-Latin] DSSTox_RID_77175 HMS1922F05 KBio2_002151 MLS006011859 1-[2-(Dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexanol NCGC00095109-04 AB00053751-08 PNVNVHUZROJLTJ-UHFFFAOYSA-N AK116310 Spectrum2_000542 BRD-A51714012-001-02-3 ST24037045 CHEBI:9943 D,L-Venlafaxine DB00285 WY-45655 Efectin HMS3714K11 KBio3_001877 N,N-dimethyl-2-(1-hydroxycyclohexyl)-2-(4-methoxyphenyl)ethylamine 1-{2-(dimethylamino)-1-[4-(methyloxy)phenyl]ethyl}cyclohexanol NCGC00095109-08 AB00053751_12 SCHEMBL35154 API0004581 Spectrum5_001516 C07187 Tox21_111425_1 CS-2129 Venlafaxine ER VenlafaxineXR DSSTox_CID_3737 FT-0642242 K700 LS-57095 1-(2-(dimethylamino)-1-(4-methoxyphenyl)ethyl)cyclohexanol NCGC00095109-02 93413-69-5 NSC_62923 AC-1547 SpecPlus_000842 BC209117 SR-01000762930-3 CAS_99300-78-4 Venlafaxina Cyclohexanol, 1-(2-(dimethylamino)-1-(4-methoxyphenyl)ethyl)-, hydrochloride D08670 Venlafexine DTXSID6023737 HMS2090F04 KBio2_004719 MolPort-003-666-534 1-[2-dimethylamino-1-(4-methoxylphenyl)ethyl]cyclohexanol NCGC00095109-05 AB00053751-10 SBI-0052740.P002 AKOS005555049 Spectrum3_000989 BRD-A51714012-003-01-1 STK621394 venlafaxine (Effexor) DivK1c_006938 Efectin (TN) HSDB 6699 KBioGR_001590 (RS)-1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexanol N,N-dimethyl-2-(1-hydroxycyclohexyl)-2-(4-methoxyphenyl)ethylamine; 1-[2-dimethylamino-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol; 1-[(1R)-2-(Dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexanol 413V695 NSC-758676 AB00053751_13 SMR002204138 AT-6375 Spectrum_001671 CAS-93413-69-5 Venflaxine EP CTK8F8921 Venlafaxine [BAN:INN] Venlafaxinum DSSTox_GSID_23737 GTPL7321 KBio1_001882 MCULE-6632261838 1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol NCGC00095109-03 99300-78-4 (hydrochloride) Pharmakon1600-01504171 AC1L1KU8 SPECTRUM1504171 BDBM82071 SR-01000762930-4 CCG-39577 Venlafaxina [INN-Spanish] Cyclohexanol, 1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]- [ Show all ]
Inchi Key	PNVNVHUZROJLTJ-UHFFFAOYSA-N
Inchi ID	InChI=1S/C17H27NO2/c1-18(2)13-16(17(19)11-5-4-6-12-17)14-7-9-15(20-3)10-8-14/h7-10,16,19H,4-6,11-13H2,1-3H3
PubChem CID	5656
ChEMBL	CHEMBL637
IUPHAR	N/A
BindingDB	82071
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
264413	5-hydroxytryptamine receptor 1A	P19327	Htr1a	Rattus norvegicus (Rat)	422
264426	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
264412	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
264423	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
264402	5-hydroxytryptamine receptor 1E	P28566	HTR1E	Homo sapiens (Human)	365
264401	5-hydroxytryptamine receptor 1F	P30939	HTR1F	Homo sapiens (Human)	366
264395	5-hydroxytryptamine receptor 2A	P14842	Htr2a	Rattus norvegicus (Rat)	471
264408	5-hydroxytryptamine receptor 2A	P28223	HTR2A	Homo sapiens (Human)	471
264409	5-hydroxytryptamine receptor 2B	P41595	HTR2B	Homo sapiens (Human)	481
264391	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
264396	5-hydroxytryptamine receptor 2C	P08909	Htr2c	Rattus norvegicus (Rat)	460
264393	5-hydroxytryptamine receptor 4	O70528	HTR4	Cavia porcellus (Guinea pig)	388
264405	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
264416	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
264406	Adenosine receptor A1	P25099	Adora1	Rattus norvegicus (Rat)	326
264418	Adenosine receptor A2b	Q1LZD0	ADORA2B	Bos taurus (Bovine)	332
264389	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
264411	Alpha-1A adrenergic receptor	P43140	Adra1a	Rattus norvegicus (Rat)	466
264429	Alpha-1B adrenergic receptor	P15823	Adra1b	Rattus norvegicus (Rat)	515
264410	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450

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