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| Name | Cholecystokinin receptor type A |
|---|---|
| Species | Rattus norvegicus (Rat) |
| Gene | Cckar |
| Synonym | CCK-A receptor CCK-AR CCK1 receptor CCK1-R cholecystokinin receptor type A [ Show all ] |
| Disease | N/A for non-human GPCRs |
| Length | 444 |
| Amino acid sequence | MSHSPARQHLVESSRMDVVDSLLMNGSNITPPCELGLENETLFCLDQPQPSKEWQSALQILLYSIIFLLSVLGNTLVITVLIRNKRMRTVTNIFLLSLAVSDLMLCLFCMPFNLIPNLLKDFIFGSAVCKTTTYFMGTSVSVSTFNLVAISLERYGAICRPLQSRVWQTKSHALKVIAATWCLSFTIMTPYPIYSNLVPFTKNNNQTANMCRFLLPSDAMQQSWQTFLLLILFLLPGIVMVVAYGLISLELYQGIKFDASQKKSAKEKKPSTGSSTRYEDSDGCYLQKSRPPRKLELQQLSSGSGGSRLNRIRSSSSAANLIAKKRVIRMLIVIVVLFFLCWMPIFSANAWRAYDTVSAEKHLSGTPISFILLLSYTSSCVNPIIYCFMNKRFRLGFMATFPCCPNPGPPGVRGEVGEEEDGRTIRALLSRYSYSHMSTSAPPP |
| UniProt | P30551 |
| Protein Data Bank | N/A |
| GPCR-HGmod model | N/A |
| 3D structure model | No available structures or models |
| BioLiP | N/A |
| Therapeutic Target Database | N/A |
| ChEMBL | CHEMBL2871 |
| IUPHAR | 76 |
| DrugBank | N/A |
You can:
| GLASS ID | Molecule | Formula | Molecular weight | H-bond acceptor / donor | XlogP | Lipinski's druglikeness |
|---|---|---|---|---|---|---|
| 118 |  CHEMBL343158 | C21H18FN3OS | 379.453 | 5 / 2 | 3.8 | Yes |
| 402 |  diazepam | C16H13ClN2O | 284.743 | 2 / 0 | 3.0 | Yes |
| 628 |  CHEMBL37699 | C25H20BrN3O2 | 474.358 | 3 / 1 | 5.1 | No |
| 903 |  CHEMBL115612 | C27H28N6O3 | 484.56 | 6 / 3 | 3.2 | Yes |
| 1093 |  CHEMBL140749 | C22H22FN3OS | 395.496 | 5 / 2 | 3.7 | Yes |
| 441717 |  CHEMBL3349028 | C29H39N3O5 | 509.647 | 5 / 5 | N/A | No |
| 441720 |  CHEMBL3350686 | C29H39N3O5 | 509.647 | 5 / 5 | N/A | No |
| 1350 |  CHEMBL2111203 | C29H39N3O5 | 509.647 | 5 / 5 | N/A | No |
| 1679 |  CHEMBL124917 | C20H29ClN2O4 | 396.912 | 4 / 3 | 4.2 | Yes |
| 1847 |  CHEMBL336690 | C22H26FN3O2 | 383.467 | 5 / 1 | 4.4 | Yes |
| 3215 |  CHEMBL354049 | C33H40N4O5 | 572.706 | 6 / 5 | 4.8 | No |
| 4026 |  CHEMBL2110202 | C25H29N9O2 | 487.568 | 7 / 4 | 3.2 | Yes |
| 4044 |  CHEMBL339115 | C22H31ClN2O4 | 422.95 | 4 / 3 | 4.6 | Yes |
| 4491 |  CHEMBL575161 | C25H20N2O4S | 444.505 | 5 / 3 | 5.5 | No |
| 4787 |  CHEMBL124719 | C42H50N8O13S2 | 939.025 | 14 / 11 | 0.6 | No |
| 5015 |  CHEMBL432266 | C33H32FN9O3 | 621.677 | 8 / 3 | 3.8 | No |
| 5561 |  CHEMBL140495 | C24H22FN3O2 | 403.457 | 5 / 2 | 4.4 | Yes |
| 6548 |  CHEMBL424076 | C25H20N4O2 | 408.461 | 3 / 2 | 3.7 | Yes |
| 7047 |  CHEMBL9083 | C24H21N7O2 | 439.479 | 5 / 3 | 3.0 | Yes |
| 7998 |  CHEMBL573562 | C25H21N3O4 | 427.46 | 4 / 4 | 4.3 | Yes |
| 8259 |  CHEMBL86879 | C39H44N4O5S | 680.864 | 6 / 5 | 6.7 | No |
| 553286 |  rebamipide | C19H15ClN2O4 | 370.789 | 4 / 3 | 2.4 | Yes |
| 553290 |  (3S)-4-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-[[(2S)-2-[[(2S)-3-(1H-indol-3-yl)-2-[3-(2-methylpropoxycarbonylamino)propanoylamino]propanoyl]amino]-4-methylsulfanylbutanoyl]amino]-4-oxobutanoic acid | C37H49N7O9S | 767.899 | 10 / 8 | 2.2 | No |
| 8943 |  CHEMBL137208 | C25H24N4O2 | 412.493 | 3 / 2 | 3.8 | Yes |
| 9325 |  CHEMBL336749 | C23H19FN4O2 | 402.429 | 4 / 2 | 3.0 | Yes |
| 9805 |  CHEMBL1933109 | C26H23N3O4 | 441.487 | 4 / 4 | 5.0 | Yes |
| 10008 |  CHEMBL102867 | C27H26Cl2N4O3 | 525.43 | 3 / 2 | 5.2 | No |
| 10558 |  CHEMBL3143146 | C45H58N8O7S | 855.068 | 8 / 7 | 5.5 | No |
| 10560 |  CHEMBL341403 | C45H58N8O7S | 855.068 | 8 / 7 | 5.5 | No |
| 10683 |  CHEMBL413654 | C97H126N20O32S | 2116.24 | 34 / 27 | -3.9 | No |
| 11507 |  CHEMBL135988 | C21H24N4O2 | 364.449 | 3 / 2 | 2.4 | Yes |
| 11570 |  CHEMBL9312 | C23H22N2O | 342.442 | 1 / 2 | 5.3 | No |
| 12695 |  CHEMBL8949 | C26H21NO | 363.46 | 1 / 1 | 6.5 | No |
| 12711 |  CHEMBL1907850 | C23H17BrFN3O2 | 466.31 | 4 / 1 | 3.6 | Yes |
| 12713 |  CHEMBL70984 | C23H17BrFN3O2 | 466.31 | 4 / 1 | 3.6 | Yes |
| 13596 |  CHEMBL355319 | C27H29N3O4 | 459.546 | 4 / 2 | 4.6 | Yes |
| 14380 |  CHEMBL342614 | C24H19ClN4O4 | 462.89 | 5 / 3 | 3.7 | Yes |
| 14454 |  CHEMBL70883 | C28H23FN4O4 | 498.514 | 6 / 2 | 4.5 | Yes |
| 15269 |  CHEMBL332595 | C28H30N4O3 | 470.573 | 3 / 2 | 5.1 | No |
| 16380 |  CHEMBL22630 | C21H16FN3O4 | 393.374 | 6 / 2 | 2.5 | Yes |
| 16633 |  CHEMBL313756 | C40H47N5O6S | 725.905 | 7 / 5 | 5.4 | No |
| 16636 |  CHEMBL313756 | C40H47N5O6S | 725.905 | 7 / 5 | 5.4 | No |
| 17110 |  CHEMBL1907839 | C23H18IN3O2 | 495.32 | 3 / 1 | 4.4 | Yes |
| 17111 |  CHEMBL306166 | C23H18IN3O2 | 495.32 | 3 / 1 | 4.4 | Yes |
| 17244 |  CHEMBL1907842 | C24H18F3N3O2 | 437.422 | 6 / 1 | 4.1 | Yes |
| 17245 |  CHEMBL2092865 | C24H18F3N3O2 | 437.422 | 6 / 1 | 4.1 | Yes |
| 17247 |  CHEMBL73699 | C24H18F3N3O2 | 437.422 | 6 / 1 | 4.1 | Yes |
| 17921 |  CHEMBL575200 | C26H22N2O5S | 474.531 | 6 / 3 | 5.1 | No |
| 19303 |  CHEMBL342415 | C27H25FN4O | 440.522 | 4 / 2 | 4.4 | Yes |
| 20006 |  CHEMBL306958 | C23H19FN4O2 | 402.429 | 4 / 2 | 3.5 | Yes |
| 20213 |  CHEMBL53234 | C23H17ClN6O | 428.88 | 4 / 2 | 3.7 | Yes |
| 20270 |  CHEMBL430516 | C28H29N5O3 | 483.572 | 5 / 3 | 3.9 | Yes |
| 20501 |  CHEMBL371019 | C33H40N6O6S | 648.779 | 7 / 5 | 3.3 | No |
| 20503 |  CHEMBL436123 | C33H40N6O6S | 648.779 | 7 / 5 | 3.3 | No |
| 20505 |  CHEMBL371288 | C33H40N6O6S | 648.779 | 7 / 5 | 3.3 | No |
| 20507 |  CHEMBL200490 | C33H40N6O6S | 648.779 | 7 / 5 | 3.3 | No |
| 21057 |  CHEMBL576021 | C26H23N3O4 | 441.487 | 4 / 4 | 5.0 | Yes |
| 21279 |  CHEMBL277661 | C22H18N2O4 | 374.396 | 4 / 2 | 3.4 | Yes |
| 21282 |  CHEMBL22918 | C22H18N2O4 | 374.396 | 4 / 2 | 3.4 | Yes |
| 21369 |  CHEMBL350853 | C23H27N5O2 | 405.502 | 3 / 2 | 2.7 | Yes |
| 22011 |  CHEMBL34335 | C24H29N3O4 | 423.513 | 4 / 2 | 3.7 | Yes |
| 22615 |  CHEMBL420459 | C32H42N4O3 | 530.713 | 3 / 2 | 7.4 | No |
| 22642 |  CHEMBL74170 | C27H27N3O2 | 425.532 | 3 / 2 | 5.9 | No |
| 22887 |  CHEMBL484590 | C20H17N3O6 | 395.371 | 6 / 5 | 2.2 | Yes |
| 22954 |  CHEMBL1808416 | C33H41N5O4 | 571.722 | 5 / 2 | 3.9 | No |
| 23230 |  CHEMBL43345 | C17H17NO2 | 267.328 | 3 / 3 | 2.5 | Yes |
| 23689 |  CHEMBL303386 | C30H32N4O4 | 512.61 | 5 / 2 | 4.8 | No |
| 23702 |  CHEMBL9888 | C24H21BrN4O3 | 493.361 | 4 / 2 | 4.9 | Yes |
| 24619 |  CHEMBL168253 | C26H31N9O2 | 501.595 | 7 / 3 | 3.8 | No |
| 24990 |  CHEMBL59985 | C37H50N2O3 | 570.818 | 3 / 2 | 8.9 | No |
| 25068 |  CHEMBL338056 | C41H48N8O13S2 | 924.998 | 14 / 11 | 0.4 | No |
| 25076 |  CHEMBL536938 | C27H41Cl3N4O3 | 576.0 | 4 / 3 | N/A | No |
| 25169 |  CHEMBL435587 | C21H28BrN3O4 | 466.376 | 5 / 3 | 1.6 | Yes |
| 25266 |  CHEMBL301331 | C31H22FN5 | 483.55 | 4 / 1 | 6.1 | No |
| 25888 |  CHEMBL331413 | C21H31ClN2O4 | 410.939 | 4 / 3 | 4.8 | Yes |
| 26162 |  CHEMBL314846 | C29H33IN6O3 | 640.526 | 5 / 2 | N/A | No |
| 26194 |  CHEMBL309017 | C26H19N3O2 | 405.457 | 3 / 2 | 4.8 | Yes |
| 26435 |  CHEMBL1808417 | C33H40FN5O4 | 589.712 | 6 / 2 | 4.0 | No |
| 27776 |  CHEMBL266376 | C23H21N5O3 | 415.453 | 4 / 3 | 3.5 | Yes |
| 27836 |  CHEMBL40668 | C26H21ClFN3O4 | 493.919 | 6 / 1 | 4.7 | Yes |
| 28169 |  CHEMBL152306 | C31H27N5O3 | 517.589 | 5 / 2 | 4.8 | No |
| 28202 |  CHEMBL268197 | C22H18ClNO | 347.842 | 1 / 1 | 5.8 | No |
| 28329 |  CHEMBL351891 | C25H20N6O4 | 468.473 | 6 / 3 | 2.9 | Yes |
| 28331 |  CHEMBL163610 | C25H20N6O4 | 468.473 | 6 / 3 | 2.9 | Yes |
| 29066 |  CHEMBL1808409 | C27H35N5O5 | 509.607 | 6 / 3 | 2.4 | No |
| 29115 |  CHEMBL406978 | C36H47N7O10S | 769.871 | 11 / 9 | 1.3 | No |
| 29327 |  CHEMBL8779 | C24H22N2O | 354.453 | 1 / 2 | 5.8 | No |
| 29332 |  CHEMBL469974 | C25H23N3O2 | 397.478 | 2 / 3 | 5.4 | No |
| 29798 |  CHEMBL331929 | C30H26N4O3 | 490.563 | 3 / 2 | 4.9 | Yes |
| 30324 |  CHEMBL135371 | C30H32N6O4 | 540.624 | 6 / 2 | 2.7 | No |
| 30417 |  CHEMBL330773 | C29H32N4O3S | 516.66 | 4 / 2 | 5.5 | No |
| 30737 |  CHEMBL136412 | C24H20N4O4 | 428.448 | 5 / 3 | 3.0 | Yes |
| 30920 |  CHEMBL308111 | C24H16F2N4O2 | 430.415 | 5 / 3 | 4.2 | Yes |
| 31113 |  CHEMBL1808413 | C27H37N5O3 | 479.625 | 4 / 2 | 3.8 | Yes |
| 31895 |  CHEMBL407530 | C48H61N9O11S3 | 1036.25 | 13 / 9 | 1.8 | No |
| 32453 |  CHEMBL344211 | C28H38N4O3 | 478.637 | 4 / 3 | 5.1 | No |
| 32735 |  CHEMBL70549 | C26H20FN3O2 | 425.463 | 4 / 2 | 4.5 | Yes |
| 32776 |  CHEMBL166168 | C28H28N4O5 | 500.555 | 6 / 2 | 4.2 | No |
| 32827 |  CHEMBL268382 | C26H24N2O3 | 412.489 | 3 / 2 | 6.0 | No |
| 33673 |  CHEMBL9308 | C22H19ClN2O | 362.857 | 1 / 2 | 5.6 | No |
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