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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	5-hydroxytryptamine receptor 5A
Species	Rattus norvegicus (Rat)
Gene	Htr5a
Synonym	5-HT5A receptor REC17 MR22 Htr5 5-HT-5A 5HT5- 5-HT5A 5-hydroxytryptamine (serotonin) receptor 5A, G protein-coupled 5-HT5alpha serotonin receptor 5A [ Show all ]
Disease	N/A for non-human GPCRs
Length	357
Amino acid sequence	MDLPINLTSFSLSTPSTLEPNRSLDTEALRTSQSFLSAFRVLVLTLLGFLAAATFTWNLLVLATILRVRTFHRVPHNLVASMAISDVLVAVLVMPLSLVHELSGRRWQLGRRLCQLWIACDVLCCTASIWNVTAIALDRYWSITRHLEYTLRARKRVSNVMILLTWALSAVISLAPLLFGWGETYSELSEECQVSREPSYTVFSTVGAFYLPLCVVLFVYWKIYKAAKFRMGSRKTNSVSPIPEAVEVKDASQHPQMVFTVRHATVTFQTEGDTWREQKEQRAALMVGILIGVFVLCWFPFFVTELISPLCSWDIPALWKSIFLWLGYSNSFFNPLIYTAFNRSYSSAFKVFFSKQQ
UniProt	P35364
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4655
IUPHAR	10
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
6268	CHEMBL76237	C19H22N2O3S	358.456	4 / 0	3.5	Yes
13648	8-OH-Dpat	C16H25NO	247.382	2 / 1	4.1	Yes
23173	1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine	C11H16INO2	321.158	3 / 1	2.5	Yes
26598	Yohimbine	C21H26N2O3	354.45	4 / 2	2.9	Yes
39124	CHEMBL334553	C16H25NO	247.382	2 / 0	4.0	Yes
67092	Melatonin	C13H16N2O2	232.283	2 / 2	0.8	Yes
71362	CHEMBL133020	C16H25NO	247.382	2 / 1	3.8	Yes
71363	CHEMBL133433	C16H25NO	247.382	2 / 1	3.8	Yes
76577	Zacopride	C15H20ClN3O2	309.794	4 / 2	1.7	Yes
97163	CHEMBL92139	C18H20N2O2S	328.43	3 / 0	3.5	Yes
148379	CHEMBL541993	C11H12ClF2N3	259.685	3 / 2	2.5	Yes
154027	Mesulergine	C18H26N4O2S	362.492	5 / 1	1.4	Yes
174885	methysergide	C21H27N3O2	353.466	3 / 2	2.3	Yes
182776	CHEMBL37844	C15H23NO	233.355	2 / 1	3.6	Yes
223307	CHEMBL34652	C16H25NO	247.382	2 / 0	4.0	Yes
223308	CHEMBL132580	C16H25NO	247.382	2 / 0	4.0	Yes
225632	CHEMBL93868	C18H20N2O2S	328.43	3 / 0	3.5	Yes
251091	CHEMBL127411	C20H22N2O3S	370.467	4 / 1	2.9	Yes
255410	CHEMBL126340	C25H24N2O3S	432.538	4 / 0	5.2	No
267364	CHEMBL133935	C17H27NO	261.409	2 / 0	4.2	Yes
267365	CHEMBL336124	C17H27NO	261.409	2 / 0	4.2	Yes
282243	CHEMBL132019	C16H25NO	247.382	2 / 1	3.8	Yes
282244	CHEMBL132123	C16H25NO	247.382	2 / 1	3.8	Yes
290313	serotonin	C10H12N2O	176.219	2 / 3	0.2	Yes
299026	methiothepin	C20H24N2S2	356.546	4 / 0	4.2	Yes
302412	abt-702	C22H19BrN6O	463.339	7 / 1	3.4	Yes
312996	dl-Arterenol	C8H11NO3	169.18	4 / 4	-1.2	Yes
313385	CHEMBL34653	C15H23NO	233.355	2 / 1	3.6	Yes
338101	CHEMBL263700	C19H20N2O2	308.381	3 / 1	3.5	Yes
359853	CHEMBL125745	C16H16N2O2S	300.376	3 / 1	2.5	Yes
367178	dopamine	C8H11NO2	153.181	3 / 3	-1.0	Yes
373706	CHEMBL135894	C17H27NO	261.409	2 / 0	4.2	Yes
373707	CHEMBL134331	C17H27NO	261.409	2 / 0	4.2	Yes
375966	5-Carboxamidotryptamine	C11H13N3O	203.245	2 / 3	-0.6	Yes
386160	metergoline	C25H29N3O2	403.526	3 / 1	3.8	Yes
388259	ERGOTAMINE	C33H35N5O5	581.673	6 / 3	2.0	No
390516	CHEMBL404372	C9H10ClN3	195.65	1 / 2	1.2	Yes
390714	Skf 83566	C17H18BrNO	332.241	2 / 1	4.0	Yes
402971	CHEMBL341373	C14H21NO	219.328	2 / 1	2.8	Yes
424618	CHEMBL423527	C15H23NO	233.355	2 / 0	3.1	Yes

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