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You can:

Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	FLUPERLAPINE
Molecular formula	C19H20FN3
IUPAC name	3-fluoro-6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine
Molecular weight	309.388
Hydrogen bond acceptor	3
Hydrogen bond donor	0
XlogP	2.9
Synonyms	NB-106689 PDSP2_000470 UNII-EWG253M961 BRD-K15715913-001-01-5 CTK8F9821 Fluperlapina [INN-Spanish] HMS2052M07 NCGC00160388-02 SMR000449303 3-Fluoro-6-(4-methyl-piperazin-1-yl)-11H-dibenzo[b,e]azepine AC1L2LPB CCG-101093 DSSTox_GSID_46123 Fluperlapinum L000256 MLS001424156 OBWGMKKHCLHVIE-UHFFFAOYSA-N Tox21_111780 3-fluoro-6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine Biomol-NT_000093 CHEMBL63756 EWG253M961 FT-0651061 NC00343 SAM001247034 ZINC26247473 67121-76-0 C10967 D0F8TG HMS2090H12 NCGC00160388-03 SR-01000759288 3-Fluoro-6-(4-methyl-piperazin-1-yl)-11H-dibenzo[b,e]azepine(fluperlapine) API0006718 CHEBI:5122 DSSTox_RID_81359 Fluperlapinum [INN-Latin] LS-176575 NB 106-689 PDSP1_000472 Tox21_111780_1 (E)-3-fluoro-6-(4-methylpiperazin-1-yl)-11H-dibenzo[b,e]azepine 3-fluoro-6-(4-methylpiperazinyl)-11H-dibenz(b,e)azepine BPBio1_001099 CPD000449303 Fluperlapina GTPL279 NCGC00160388-01 SCHEMBL142558 3-Fluoro-6-(4-methyl-1-piperazinyl)morphanthridine AB00639914-06 CAS-67121-76-0 DSSTox_CID_26123 Fluperlapine [INN] HMS3394M07 NCGC00160388-04 SR-01000759288-4 3-fluoro-6-(4-methyl-piperazinyl)-11h-dibenz-(b,e)-azepine BDBM50040241 DTXSID2046123 FT-0081219 MLS000758217 [ Show all ]
Inchi Key	OBWGMKKHCLHVIE-UHFFFAOYSA-N
Inchi ID	InChI=1S/C19H20FN3/c1-22-8-10-23(11-9-22)19-17-5-3-2-4-14(17)12-15-6-7-16(20)13-18(15)21-19/h2-7,13H,8-12H2,1H3
PubChem CID	49381
ChEMBL	CHEMBL63756
IUPHAR	279
BindingDB	50040241
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
556405	5-hydroxytryptamine receptor 2A	P14842	Htr2a	Rattus norvegicus (Rat)	471
237428	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
237430	5-hydroxytryptamine receptor 2C	P08909	Htr2c	Rattus norvegicus (Rat)	460
237421	5-hydroxytryptamine receptor 6	P31388	Htr6	Rattus norvegicus (Rat)	436
237422	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
554459	5-hydroxytryptamine receptor 7	P32305	Htr7	Rattus norvegicus (Rat)	448
554460	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
237423	D(1A) dopamine receptor	P21728	DRD1	Homo sapiens (Human)	446
237429	D(1A) dopamine receptor	P18901	Drd1	Rattus norvegicus (Rat)	446
237435	D(1A) dopamine receptor	Q61616	Drd1	Mus musculus (Mouse)	446
237433	D(1B) dopamine receptor	P25115	Drd5	Rattus norvegicus (Rat)	475
237425	D(2) dopamine receptor	P61169	Drd2	Rattus norvegicus (Rat)	444
556406	D(2) dopamine receptor	P61168	Drd2	Mus musculus (Mouse)	444
556407	D(3) dopamine receptor	P19020	Drd3	Rattus norvegicus (Rat)	446
237419	D(4) dopamine receptor	P21917	DRD4	Homo sapiens (Human)	467
237431	D(4) dopamine receptor	P30729	Drd4	Rattus norvegicus (Rat)	387
237432	Muscarinic acetylcholine receptor M1	P11229	CHRM1	Homo sapiens (Human)	460
237420	Muscarinic acetylcholine receptor M2	P08172	CHRM2	Homo sapiens (Human)	466
237426	Muscarinic acetylcholine receptor M3	P20309	CHRM3	Homo sapiens (Human)	590
237427	Muscarinic acetylcholine receptor M4	P08173	CHRM4	Homo sapiens (Human)	479

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