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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	G-protein coupled estrogen receptor 1
Species	Homo sapiens (Human)
Gene	GPER1
Synonym	Chemoattractant receptor-like 2 Gpr41 IL8-related receptor DRY12 LERGU LERGU2 LYGPR Lymphocyte-derived G-protein coupled receptor Membrane estrogen receptor mER GPR30 GPGR GPER chemokine receptor-like 2 CMKRL2 DRY12 FEG-1 Flow-induced endothelial G-protein coupled receptor 1 G protein-coupled estrogen receptor 1 G-protein coupled receptor 30 CEPR GPCR-BR [ Show all ]
Disease	N/A
Length	375
Amino acid sequence	MDVTSQARGVGLEMYPGTAQPAAPNTTSPELNLSHPLLGTALANGTGELSEHQQYVIGLFLSCLYTIFLFPIGFVGNILILVVNISFREKMTIPDLYFINLAVADLILVADSLIEVFNLHERYYDIAVLCTFMSLFLQVNMYSSVFFLTWMSFDRYIALARAMRCSLFRTKHHARLSCGLIWMASVSATLVPFTAVHLQHTDEACFCFADVREVQWLEVTLGFIVPFAIIGLCYSLIVRVLVRAHRHRGLRPRRQKALRMILAVVLVFFVCWLPENVFISVHLLQRTQPGAAPCKQSFRHAHPLTGHIVNLAAFSNSCLNPLIYSFLGETFRDKLRLYIEQKTNLPALNRFCHAALKAVIPDSTEQSDVRFSSAV
UniProt	Q99527
Protein Data Bank	N/A
GPCR-HGmod model	Q99527
3D structure model	This predicted structure model is from GPCR-EXP Q99527.
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL5872
IUPHAR	221
DrugBank	BE0003446

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
523196	CHEMBL3798728	C17H16N2O3	296.326	4 / 1	3.1	Yes
548810	Femring	C20H26O3	314.425	3 / 1	2.8	Yes
553795	raloxifene	C28H27NO4S	473.587	6 / 2	6.1	No
127868	CHEMBL566178	C19H15BrINO2	496.142	3 / 1	5.5	No
526616	CHEMBL3799544	C17H17N3O2	295.342	4 / 2	2.8	Yes
460875	E2-NMe3+	C29H36NO2+	430.612	2 / 2	5.4	No
550328	MK-0354	C7H8N6	176.183	4 / 2	0.2	Yes
527308	AC1O72D3	C17H17NO	251.329	2 / 1	3.3	Yes
527693	SCHEMBL4274851	C17H18N2	250.345	2 / 2	3.0	Yes
527840	CHEMBL3800024	C17H16N2O3	296.326	4 / 1	3.1	Yes
554397	tamoxifen	C26H29NO	371.524	2 / 0	7.1	No
528045	CHEMBL3797605	C18H19NO	265.356	2 / 1	3.6	Yes
461242	E2-NB	C32H39NO4	501.667	4 / 3	5.9	No
249172	CHEMBL569277	C21H18INO3	459.283	4 / 1	4.5	Yes
461369	E2-COO-	C27H27O4-	415.509	4 / 2	5.6	No
550973	UNII-65C72P1860	C32H48O4	496.732	4 / 0	8.3	No
268396	CHEMBL583633	C21H17BrINO3	538.179	4 / 1	5.2	No
554693	G-36	C22H22BrNO2	412.327	3 / 1	6.0	No
529742	CHEMBL3798571	C18H20N2	264.372	2 / 2	3.4	Yes
297259	CHEMBL584524	C19H15BrINO2	496.142	3 / 1	5.5	No
551686	estradiol valerate	C23H32O3	356.506	3 / 1	6.0	No
530522	CHEMBL3798085	C17H18N2O	266.344	3 / 3	2.6	Yes
530654	CHEMBL3797846	C17H17N3O2	295.342	4 / 2	2.8	Yes
552036	genistein	C15H10O5	270.24	5 / 3	2.7	Yes
552153	estradiol cypionate	C26H36O3	396.571	3 / 1	7.1	No
552281	estradiol benzoate	C25H28O3	376.496	3 / 1	4.5	Yes
462272	BDBM36490	C27H32NO2+	402.558	2 / 3	4.3	Yes
355535	G-1	C21H18BrNO3	412.283	4 / 1	4.6	Yes
360592	estradiol	C18H24O2	272.388	2 / 2	4.0	Yes
555125	Fulvestrant	C32H47F5O3S	606.777	9 / 2	9.2	No
531897	CHEMBL3798007	C17H17NO2	267.328	3 / 2	2.9	Yes
373492	CHEMBL571691	C28H24BrIN2O3	643.319	4 / 2	6.8	No
532375	CHEMBL3799283	C17H18N2O	266.344	3 / 3	2.6	Yes
415411	CHEMBL583543	C19H16BrNO2	370.246	3 / 1	4.9	Yes
423532	CHEMBL585707	C26H22BrIN4O2	629.296	6 / 2	6.6	No
423719	CHEMBL569504	C28H25BrIN3O3	658.334	4 / 3	6.5	No

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