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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
Go back to previous page.

GPCR

Name	CX3C chemokine receptor 1
Species	Homo sapiens (Human)
Gene	CX3CR1
Synonym	Beta chemokine receptor-like 1 Rbs11 GPR13 G-protein coupled receptor 13 Fractalkine receptor CX3CR1 CMKDR1 CMKBRL1 CMK-BRL1 CMK-BRL-1 chemokine (C-X3-C motif) receptor 1 CCRL1 C-X3-C CKR-1 V28 [ Show all ]
Disease	N/A
Length	355
Amino acid sequence	MDQFPESVTENFEYDDLAEACYIGDIVVFGTVFLSIFYSVIFAIGLVGNLLVVFALTNSKKPKSVTDIYLLNLALSDLLFVATLPFWTHYLINEKGLHNAMCKFTTAFFFIGFFGSIFFITVISIDRYLAIVLAANSMNNRTVQHGVTISLGVWAAAILVAAPQFMFTKQKENECLGDYPEVLQEIWPVLRNVETNFLGFLLPLLIMSYCYFRIIQTLFSCKNHKKAKAIKLILLVVIVFFLFWTPYNVMIFLETLKLYDFFPSCDMRKDLRLALSVTETVAFSHCCLNPLIYAFAGEKFRRYLYHLYGKCLAVLCGRSVHVDFSSSESQRSRHGSVLSSNFTYHTSDGDALLLL
UniProt	P49238
Protein Data Bank	N/A
GPCR-HGmod model	P49238
3D structure model	This predicted structure model is from GPCR-EXP P49238.
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4843
IUPHAR	N/A
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
19237	CHEMBL2349332	C18H21BrFN5OS2	486.422	9 / 3	5.2	No
26012	CHEMBL2349182	C19H25N5OS2	403.563	8 / 3	4.8	Yes
46892	CHEMBL2349318	C19H21N5O2S2	415.53	8 / 3	3.7	Yes
50220	CHEMBL2349309	C17H22N6OS2	390.524	9 / 3	3.3	Yes
61382	CHEMBL2349314	C19H24BrN5OS2	482.459	8 / 3	5.5	No
61384	CHEMBL2349315	C19H24BrN5OS2	482.459	8 / 3	5.5	No
65645	CHEMBL2349306	C18H20F2N4O2S2	426.501	9 / 3	4.2	Yes
88399	CHEMBL2349328	C18H22BrN5OS2	468.432	8 / 3	5.1	No
93213	CHEMBL2349330	C18H22BrN5OS2	468.432	8 / 3	5.1	No
95583	CHEMBL2349187	C20H27N5OS2	417.59	8 / 3	5.0	Yes
96252	CHEMBL271013	C15H17N5OS2	347.455	8 / 3	3.1	Yes
98885	CHEMBL2349325	C19H25N5OS2	403.563	8 / 3	4.7	Yes
106977	CHEMBL2349301	C19H24ClN5OS2	438.005	8 / 3	5.9	No
124790	CHEMBL2349324	C18H22FN5OS2	407.526	9 / 3	4.5	Yes
128390	CHEMBL2349312	C19H24N4O2S2	404.547	7 / 3	4.4	Yes
128391	CHEMBL2349313	C19H24N4O2S2	404.547	7 / 3	4.4	Yes
134839	CHEMBL2349333	C18H21F2N5OS2	425.517	10 / 3	4.6	Yes
137833	CHEMBL2349179	C18H23ClN6OS2	438.993	9 / 3	4.4	Yes
150778	CHEMBL2349305	C18H21N5O2S2	403.519	9 / 3	4.6	Yes
169685	CHEMBL10309	C23H25BrN2O2	441.369	3 / 1	3.8	Yes
170419	CHEMBL2349186	C18H22N4O3S	374.459	7 / 3	3.5	Yes
184489	CHEMBL2349304	C18H22N6OS2	402.535	8 / 3	4.0	Yes
192657	CHEMBL2349321	C18H22N4O2S2	390.52	7 / 3	4.0	Yes
199812	CHEMBL2349339	C17H21N5OS2	375.509	8 / 3	3.9	Yes
214471	CHEMBL2349338	C17H21N5OS2	375.509	8 / 3	4.0	Yes
221251	CHEMBL2349329	C19H22N6OS2	414.546	9 / 3	4.1	Yes
229036	CHEMBL274737	C16H19N5OS2	361.482	8 / 3	3.6	Yes
247623	CHEMBL2349323	C18H22ClN5OS2	423.978	8 / 3	5.0	Yes
254134	CHEMBL2349308	C17H22N6OS2	390.524	9 / 3	3.3	Yes
264090	CHEMBL2349317	C19H22N6OS2	414.546	9 / 3	4.1	Yes
266646	CHEMBL2349316	C19H24FN5OS2	421.553	9 / 3	4.9	Yes
283274	CHEMBL2349185	C18H22N4O3S2	406.519	8 / 3	2.7	Yes
290213	CHEMBL2349302	C19H22ClN5O2S2	451.988	9 / 2	5.6	No
309477	CHEMBL2349184	C18H22N4O4S2	422.518	8 / 3	2.7	Yes
329787	CHEMBL2349307	C17H22N6OS2	390.524	9 / 3	3.3	Yes
331529	CHEMBL2349337	C20H19N5OS2	409.526	8 / 3	4.1	Yes
333495	az599	C25H35N3O4S	473.632	5 / 0	3.1	Yes
334066	CHEMBL2349180	C18H22ClN5O2S2	439.977	8 / 3	4.0	Yes
351196	CHEMBL2349331	C19H22N6OS2	414.546	9 / 3	4.1	Yes
356422	CHEMBL2349322	C18H22BrN5OS2	468.432	8 / 3	5.1	No
359802	CHEMBL2349334	C16H18N4O2S2	362.466	7 / 3	3.2	Yes
372081	CHEMBL2349303	C19H23N5O2S2	417.546	9 / 2	4.9	Yes
375626	CHEMBL2349181	C17H20ClN5O2S2	425.95	8 / 3	3.5	Yes
388678	CHEMBL2349335	C18H23N5OS2	389.536	8 / 3	4.4	Yes
388680	CHEMBL2349336	C18H23N5OS2	389.536	8 / 3	4.4	Yes
391999	CHEMBL2349183	C20H27N5OS2	417.59	8 / 3	5.2	No
402344	CHEMBL2349326	C19H22N6OS2	414.546	9 / 3	4.1	Yes
410950	CHEMBL2349327	C19H25N5O2S2	419.562	9 / 3	4.3	Yes
430182	CHEMBL2349319	C20H27N5O3S3	481.648	10 / 3	4.0	Yes
430685	CHEMBL2349320	C18H23N5OS2	389.536	8 / 3	4.4	Yes
432329	AZD8797	C19H25N5OS2	403.563	8 / 3	4.8	Yes
432332	CHEMBL2349311	C19H25N5OS2	403.563	8 / 3	4.8	Yes
440996	CHEMBL402986	C15H16N4O2S2	348.439	7 / 3	2.7	Yes

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