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| Name | Vasopressin V1a receptor |
|---|---|
| Species | Rattus norvegicus (Rat) |
| Gene | Avpr1a |
| Synonym | AVPR AVPR V1a AVPR1 antidiuretic hormone receptor 1a V1A receptor [ Show all ] |
| Disease | N/A for non-human GPCRs |
| Length | 424 |
| Amino acid sequence | MSFPRGSQDRSVGNSSPWWPLTTEGSNGSQEAARLGEGDSPLGDVRNEELAKLEIAVLAVIFVVAVLGNSSVLLALHRTPRKTSRMHLFIRHLSLADLAVAFFQVLPQLCWDITYRFRGPDWLCRVVKHLQVFAMFASAYMLVVMTADRYIAVCHPLKTLQQPARRSRLMIATSWVLSFILSTPQYFIFSVIEIEVNNGTKTQDCWATFIQPWGTRAYVTWMTSGVFVAPVVVLGTCYGFICYHIWRNIRGKTASSRHSKGDKGSGEAVGPFHKGLLVTPCVSSVKSISRAKIRTVKMTFVIVSAYILCWAPFFIVQMWSVWDENFIWTDSENPSITITALLASLNSCCNPWIYMFFSGHLLQDCVQSFPCCHSMAQKFAKDDSDSMSRRQTSYSNNRSPTNSTGMWKDSPKSSKSIRFIPVST |
| UniProt | P30560 |
| Protein Data Bank | N/A |
| GPCR-HGmod model | N/A |
| 3D structure model | No available structures or models |
| BioLiP | N/A |
| Therapeutic Target Database | N/A |
| ChEMBL | CHEMBL2868 |
| IUPHAR | 366 |
| DrugBank | N/A |
You can:
| GLASS ID | Molecule | Formula | Molecular weight | H-bond acceptor / donor | XlogP | Lipinski's druglikeness |
|---|---|---|---|---|---|---|
| 9487 |  CHEMBL332060 | C24H22N2O3 | 386.451 | 3 / 1 | 4.2 | Yes |
| 10059 |  Phenypressin | C46H65N15O11S2 | 1068.24 | 15 / 13 | -4.5 | No |
| 12342 |  CHEMBL2372415 | C57H76N12O13S2 | 1201.43 | 16 / 11 | 2.3 | No |
| 12633 |  CHEMBL72945 | C28H22N2O2 | 418.496 | 2 / 1 | 5.3 | No |
| 12882 |  CHEMBL143341 | C25H30N4O4 | 450.539 | 4 / 2 | 2.0 | Yes |
| 12898 |  CHEMBL266264 | C61H80N20O13 | 1301.44 | 17 / 15 | -0.8 | No |
| 13172 |  CHEMBL338018 | C46H61N7O6 | 808.037 | 7 / 4 | 5.1 | No |
| 14873 |  CHEMBL385062 | C51H73N13O10S2 | 1092.35 | 13 / 11 | 0.1 | No |
| 14875 |  CHEMBL266643 | C51H73N13O10S2 | 1092.35 | 13 / 11 | 0.1 | No |
| 442221 |  CHEMBL3350125 | C51H73N13O10S2 | 1092.35 | 13 / 11 | 0.1 | No |
| 17424 |  CHEMBL129089 | C43H58N6O6 | 754.973 | 6 / 2 | 5.1 | No |
| 17816 |  CHEMBL350090 | C24H19FN4O2S | 446.5 | 5 / 2 | 3.9 | Yes |
| 19942 |  CHEMBL339493 | C36H52N6O6 | 664.848 | 6 / 2 | 3.2 | No |
| 20112 |  CHEMBL75489 | C40H42N6O4 | 670.814 | 6 / 1 | 5.5 | No |
| 22490 |  CHEMBL1807276 | C24H28ClFN2O3 | 446.947 | 4 / 3 | 4.3 | Yes |
| 24466 |  CHEMBL339450 | C42H54N8O6 | 766.944 | 7 / 4 | 3.9 | No |
| 27013 |  CHEMBL76763 | C37H40N4O5 | 620.75 | 6 / 1 | 5.7 | No |
| 27365 |  CHEMBL332685 | C25H25N3O2 | 399.494 | 3 / 1 | 4.4 | Yes |
| 28090 |  CHEMBL59896 | C22H24N2O2 | 348.446 | 2 / 0 | 3.3 | Yes |
| 28139 |  CHEMBL418692 | C26H33N3O3 | 435.568 | 4 / 1 | 3.1 | Yes |
| 29227 |  CHEMBL333139 | C23H20N2O2 | 356.425 | 2 / 1 | 4.2 | Yes |
| 29780 |  CHEMBL119551 | C23H19ClN2O2 | 390.867 | 2 / 1 | 4.8 | Yes |
| 30436 |  CHEMBL2372421 | C46H64N18O12S2 | 1125.25 | 18 / 14 | -3.9 | No |
| 30437 |  CHEMBL2372422 | C46H64N18O12S2 | 1125.25 | 18 / 14 | -3.9 | No |
| 32339 |  CHEMBL331956 | C18H18N2O2 | 294.354 | 2 / 1 | 2.5 | Yes |
| 32455 |  CHEMBL59947 | C21H22N2O2 | 334.419 | 2 / 0 | 3.0 | Yes |
| 32565 |  CHEMBL64046 | C23H24N2O4 | 392.455 | 4 / 0 | 2.7 | Yes |
| 32596 |  CHEMBL117566 | C25H24N2O2 | 384.479 | 2 / 1 | 4.9 | Yes |
| 34010 |  CHEMBL1807278 | C21H24Cl2N2O3 | 423.334 | 3 / 3 | 3.8 | Yes |
| 35880 |  CHEMBL1817698 | C44H69N13O12S2 | 1036.23 | 16 / 13 | -4.4 | No |
| 36183 |  CHEMBL558950 | C57H77N13O10S2 | 1168.44 | 13 / 11 | 1.5 | No |
| 36185 |  CHEMBL558950 | C57H77N13O10S2 | 1168.44 | 13 / 11 | 1.5 | No |
| 36647 |  CHEMBL333201 | C24H22N2O2 | 370.452 | 2 / 1 | 4.5 | Yes |
| 37058 |  d[Cha4,Orn8]VP | C49H69N11O11S2 | 1052.28 | 14 / 11 | 0.5 | No |
| 39753 |  Relcovaptan | C28H27Cl2N3O7S | 620.498 | 8 / 2 | 3.8 | No |
| 40102 |  CHEMBL159823 | C32H25N3O2 | 483.571 | 2 / 1 | 5.3 | No |
| 41395 |  CHEMBL1807281 | C23H26Cl2N2O3 | 449.372 | 3 / 3 | 4.4 | Yes |
| 46799 |  CHEMBL417458 | C31H46N4O4S | 570.793 | 7 / 1 | 3.4 | No |
| 53748 |  d[Leu4]AVP | C47H67N13O11S2 | 1054.25 | 14 / 12 | -1.5 | No |
| 54582 |  CHEMBL2112898 | C27H44N4O5S2 | 568.792 | 8 / 2 | 2.6 | No |
| 54588 |  CHEMBL2391300 | C27H44N4O5S2 | 568.792 | 8 / 2 | 2.6 | No |
| 54625 |  CHEMBL119591 | C27H27N3O3 | 441.531 | 3 / 2 | 3.8 | Yes |
| 56285 |  CHEMBL64695 | C25H30N2O3 | 406.526 | 3 / 0 | 4.2 | Yes |
| 58613 |  CHEMBL1817692 | C41H63N13O11S2 | 978.155 | 15 / 12 | -4.5 | No |
| 60105 |  (Phe2,Orn8)-oxytocin | C42H65N13O11S2 | 992.182 | 15 / 12 | -4.1 | No |
| 61654 |  CHEMBL442743 | C26H20FN3O2 | 425.463 | 3 / 1 | 3.8 | Yes |
| 62542 |  CHEMBL59397 | C22H23N3O3 | 377.444 | 3 / 1 | 1.8 | Yes |
| 63497 |  CHEMBL334082 | C27H29N3O3 | 443.547 | 4 / 1 | 4.1 | Yes |
| 65500 |  CHEMBL308741 | C29H24N2O2 | 432.523 | 2 / 1 | 5.8 | No |
| 65701 |  CHEMBL311230 | C26H18Cl3N3O2 | 510.799 | 2 / 1 | 5.6 | No |
| 65997 |  d[Cha4,Dab8]VP | C48H67N11O11S2 | 1038.25 | 14 / 11 | 0.1 | No |
| 68195 |  CHEMBL121455 | C23H19ClN2O2 | 390.867 | 2 / 1 | 4.8 | Yes |
| 68443 |  CHEMBL1817749 | C40H61N13O11S2 | 964.128 | 15 / 12 | -4.8 | No |
| 68776 |  CHEMBL119318 | C26H25Cl2N3O2 | 482.405 | 3 / 1 | 5.4 | No |
| 70070 |  CHEMBL60096 | C27H33N3O4 | 463.578 | 4 / 1 | 3.0 | Yes |
| 444451 |  CHEMBL3349464 | C46H68N10O11S2 | 1001.23 | 14 / 11 | -1.4 | No |
| 444455 |  CHEMBL3349466 | C46H68N10O11S2 | 1001.23 | 14 / 11 | -1.4 | No |
| 70862 |  CHEMBL1790307 | C46H68N10O11S2 | 1001.23 | 14 / 11 | -1.4 | No |
| 70866 |  CHEMBL1790312 | C46H68N10O11S2 | 1001.23 | 14 / 11 | -1.4 | No |
| 71835 |  CHEMBL1790938 | C41H55N9O6 | 769.948 | 7 / 4 | 3.1 | No |
| 73575 |  CHEMBL299440 | C28H26N4O5 | 498.539 | 6 / 1 | 2.9 | Yes |
| 444630 |  CHEMBL406533 | C53H73N11O11S2 | 1104.35 | 13 / 8 | 0.6 | No |
| 74384 |  CHEMBL2372414 | C57H76N14O11S2 | 1197.44 | 16 / 11 | 3.4 | No |
| 74766 |  CHEMBL2372419 | C53H70N14O11S2 | 1143.35 | 16 / 11 | 2.0 | No |
| 74866 |  CHEMBL416505 | C20H21N3O2 | 335.407 | 3 / 0 | 1.9 | Yes |
| 76086 |  CHEMBL310416 | C27H22ClN3O2 | 455.942 | 2 / 1 | 4.7 | Yes |
| 444711 |  CHEMBL3350126 | C48H74N12O12S2 | 1075.31 | 15 / 11 | -1.9 | No |
| 76267 |  CHEMBL261914 | C48H74N12O12S2 | 1075.31 | 15 / 11 | -1.9 | No |
| 76272 |  CHEMBL263521 | C48H74N12O12S2 | 1075.31 | 15 / 11 | -1.9 | No |
| 76402 |  d[Arg4,Orn8]VP | C46H66N14O11S2 | 1055.24 | 15 / 13 | -3.4 | No |
| 77302 |  CHEMBL293863 | C24H28N2O2 | 376.5 | 2 / 0 | 4.3 | Yes |
| 77313 |  CHEMBL307487 | C37H40N4O4 | 604.751 | 5 / 1 | 5.8 | No |
| 78665 |  CHEMBL293922 | C22H21N3O2 | 359.429 | 3 / 0 | 2.7 | Yes |
| 80037 |  CHEMBL1807264 | C20H22Cl2N2O3 | 409.307 | 3 / 3 | 3.4 | Yes |
| 80733 |  CHEMBL70981 | C27H22FN3O2 | 439.49 | 3 / 1 | 4.2 | Yes |
| 81723 |  CHEMBL293177 | C21H21ClN2O2 | 368.861 | 2 / 0 | 3.6 | Yes |
| 81933 |  CHEMBL118595 | C23H20N2O2 | 356.425 | 2 / 1 | 4.2 | Yes |
| 83389 |  CHEMBL201889 | C24H18F3N5O | 449.437 | 7 / 1 | 4.6 | Yes |
| 84086 |  CHEMBL71283 | C28H22N2O3 | 434.495 | 3 / 1 | 5.2 | No |
| 85782 |  CHEMBL61578 | C21H21N3O4 | 379.416 | 4 / 0 | 2.8 | Yes |
| 86859 |  CHEMBL331424 | C23H19N3O4 | 401.422 | 4 / 1 | 4.0 | Yes |
| 86953 |  CHEMBL553710 | C51H73N13O11S2 | 1108.34 | 14 / 12 | -0.3 | No |
| 86956 |  CHEMBL553710 | C51H73N13O11S2 | 1108.34 | 14 / 12 | -0.3 | No |
| 88535 |  CHEMBL299532 | C25H19BrN4O2 | 487.357 | 3 / 1 | 3.7 | Yes |
| 88544 |  d[Leu4,Orn8]VP | C46H65N11O11S2 | 1012.21 | 14 / 11 | -0.9 | No |
| 88689 |  CHEMBL77105 | C37H48N4O5 | 628.814 | 6 / 1 | 5.5 | No |
| 88731 |  CHEMBL405289 | C40H53N9O6 | 755.921 | 7 / 5 | 3.0 | No |
| 91111 |  CHEMBL2112250 | C42H54N8O6 | 766.944 | 7 / 4 | 4.0 | No |
| 92274 |  CHEMBL118760 | C24H22N2O3 | 386.451 | 3 / 1 | 4.8 | Yes |
| 92456 |  CHEMBL307271 | C29H24N2O2 | 432.523 | 2 / 1 | 5.6 | No |
| 93098 |  CHEMBL129733 | C41H54N6O6 | 726.919 | 6 / 3 | 4.6 | No |
| 94128 |  CHEMBL71355 | C26H20BrN3O2 | 486.369 | 2 / 1 | 4.4 | Yes |
| 96506 |  CHEMBL305309 | C15H20N2O | 244.338 | 2 / 0 | 1.8 | Yes |
| 96530 |  CHEMBL304060 | C27H23N3O2S | 453.56 | 3 / 1 | 4.2 | Yes |
| 96597 |  CHEMBL1819439 | C45H69N13O13S2 | 1064.24 | 16 / 13 | -4.0 | No |
| 96831 |  CHEMBL61947 | C23H27N3O3 | 393.487 | 4 / 1 | 2.0 | Yes |
| 100313 |  CHEMBL304486 | C24H29N3O3 | 407.514 | 4 / 1 | 2.3 | Yes |
| 102169 |  CHEMBL118220 | C24H22N2O2 | 370.452 | 2 / 1 | 4.5 | Yes |
| 445766 |  CHEMBL412539 | C47H68N14O11S2 | 1069.27 | 15 / 12 | -2.6 | No |
| 104164 |  CHEMBL324935 | C20H22N2O2 | 322.408 | 2 / 1 | 3.5 | Yes |
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