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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	C-X-C chemokine receptor type 4
Species	Homo sapiens (Human)
Gene	CXCR4
Synonym	LESTR LESTR {ECO:0000303\|PubMed:8276799} Stromal cell-derived factor 1 receptor LCR1 LAP-3 Leukocyte-derived seven transmembrane domain receptor Lipopolysaccharide-associated protein 3 LPS-associated protein 3 NPY3R NPYRL NPYY3R SDF-1 receptor HUMSTSR HSY3RR CD184 chemokine (C-X-C motif) receptor 4 Cmkar4 CXC-R4 CXCR-4 CXCR4 FB22 fusin HM89 [ Show all ]
Disease	N/A
Length	352
Amino acid sequence	MEGISIYTSDNYTEEMGSGDYDSMKEPCFREENANFNKIFLPTIYSIIFLTGIVGNGLVILVMGYQKKLRSMTDKYRLHLSVADLLFVITLPFWAVDAVANWYFGNFLCKAVHVIYTVNLYSSVLILAFISLDRYLAIVHATNSQRPRKLLAEKVVYVGVWIPALLLTIPDFIFANVSEADDRYICDRFYPNDLWVVVFQFQHIMVGLILPGIVILSCYCIIISKLSHSKGHQKRKALKTTVILILAFFACWLPYYIGISIDSFILLEIIKQGCEFENTVHKWISITEALAFFHCCLNPILYAFLGAKFKTSAQHALTSVSRGSSLKILSKGKRGGHSSVSTESESSSFHSS
UniProt	P61073
Protein Data Bank	3oe9, 3oe8, 3oe6, 3odu
GPCR-HGmod model	P61073
3D structure model	This structure is from PDB ID 3oe9.
BioLiP	BL0187218, BL0187262,BL0187263, BL0187259,BL0187260,BL0187261, BL0187197,BL0187198
Therapeutic Target Database	N/A
ChEMBL	CHEMBL2107
IUPHAR	71
DrugBank	BE0000919

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
535928	CHEMBL3972873	C27H32N6O	456.594	5 / 2	2.2	Yes
535929	CHEMBL3981053	C27H32N6O	456.594	5 / 2	2.2	Yes
1801	CHEMBL536302	C14H21IN6	400.268	2 / 5	N/A	N/A
2038	CHEMBL218806	C37H49N11O6	743.87	8 / 9	0.2	No
2039	CHEMBL374421	C37H49N11O6	743.87	8 / 9	0.2	No
547933	CHEMBL3933958	C26H36N8O2S	524.688	5 / 4	0.8	No
547934	CHEMBL3897010	C26H36N8O2S	524.688	5 / 4	0.8	No
3716	CHEMBL2031828	C39H42FN7O2	659.81	6 / 4	4.7	No
3717	CHEMBL2031696	C39H42FN7O2	659.81	6 / 4	4.7	No
547943	CHEMBL3969980	C19H17F2N3	325.363	5 / 2	4.1	Yes
5566	CHEMBL2180085	C37H46F3N9O8	801.825	13 / 10	N/A	No
7028	CHEMBL1956255	C36H47N11O5	713.844	7 / 9	0.4	No
7980	CHEMBL460483	C20H30N2S	330.534	2 / 1	5.7	No
536234	CHEMBL3958178	C24H27N5	385.515	4 / 2	2.3	Yes
536245	CHEMBL3946745	C27H31N5	425.58	4 / 2	3.7	Yes
536247	CHEMBL3935318	C28H36N6	456.638	5 / 2	2.5	Yes
536248	CHEMBL3911032	C28H36N6	456.638	5 / 2	2.5	Yes
536254	CHEMBL3974711	C31H39N5O2	513.686	6 / 1	4.2	No
10756	CHEMBL1682855	C20H28N4	324.472	4 / 1	2.1	Yes
11468	SCHEMBL6012808	C23H35N3O2	385.552	3 / 1	3.7	Yes
536302	CHEMBL3925646	C34H44N6O2	568.766	7 / 1	4.1	No
12760	CID 56647929	C98H134N24O22	2000.3	28 / 23	-5.8	No
12804	CHEMBL462588	C23H38N4S2	434.705	4 / 1	5.3	No
13274	Spermidine tris-PheG	C28H37N9	499.667	3 / 5	2.9	Yes
548029	CHEMBL3941019	C23H27N3	345.49	3 / 2	5.5	No
14347	BDBM50363969	C77H98N18O14	1499.74	16 / 16	2.1	No
14571	CHEMBL2029608	C37H48N10O5	712.856	7 / 9	1.2	No
464763	CHEMBL3581265	C39H51N11O6	769.908	8 / 9	0.7	No
464766	CHEMBL3581273	C39H51N11O6	769.908	8 / 9	0.7	No
464768	CHEMBL3581264	C39H51N11O6	769.908	8 / 9	0.7	No
464769	CHEMBL3581271	C39H51N11O6	769.908	8 / 9	0.7	No
464772	CHEMBL3581272	C39H51N11O6	769.908	8 / 9	0.7	No
464773	CHEMBL3581270	C39H51N11O6	769.908	8 / 9	0.7	No
16719	CHEMBL1682990	C18H26N4	298.434	4 / 1	1.7	Yes
548089	CHEMBL3902257	C26H36N8O2S	524.688	5 / 4	0.7	No
21342	CHEMBL3091682	C26H38N4	406.618	4 / 2	3.8	Yes
536519	CHEMBL3901600	C27H33N5	427.596	4 / 2	4.1	Yes
536520	CHEMBL3944558	C27H33N5	427.596	4 / 2	4.1	Yes
442543	CHEMBL2031832	C40H42FN7O3	687.82	6 / 4	4.9	No
22673	CHEMBL2031701	C40H42FN7O3	687.82	6 / 4	4.9	No
23489	CHEMBL3091690	C29H37N5	455.65	5 / 1	3.3	Yes
25413	CHEMBL1682864	C22H32N4	352.526	4 / 1	2.9	Yes
536670	CHEMBL3976878	C31H34N6	490.655	5 / 2	4.2	Yes
536718	CHEMBL3947926	C31H38N6O2S	558.745	7 / 1	1.6	No
536722	CHEMBL434161	C20H25N3O2S	371.499	5 / 1	3.9	Yes
29267	CHEMBL235309	C24H22N2	338.454	2 / 2	6.1	No
536739	CHEMBL3947569	C36H37N5O2	571.725	5 / 0	5.7	No
30010	CHEMBL2370126	C80H135N33O18S2	1911.29	28 / 30	-11.2	No
30111	1,4-benzenedimethanamine, 2,3,5,6-tetramethyl-	C12H20N2	192.306	2 / 2	1.1	Yes
30391	CHEMBL2031838	C41H46FN7O2	687.864	6 / 4	5.7	No
30392	CHEMBL2031821	C41H46FN7O2	687.864	6 / 4	5.7	No
30602	AC1LA88L	C37H43N5O4	621.782	5 / 2	5.7	No
536826	CHEMBL3897039	C21H23N3	317.436	3 / 2	4.6	Yes
32251	m-Terephthalanisidide	C22H20N2O4	376.412	4 / 2	3.5	Yes
466877	CHEMBL3581285	C30H47N11O6	657.777	8 / 8	-1.9	No
33742	CHEMBL2370132	C90H140N32O19S2	2038.44	28 / 30	-8.0	No
548311	CHEMBL3923084	C139H221N45O31S2	3082.7	43 / 50	-7.0	No
36447	CHEMBL105659	C34H40N4O2	536.72	4 / 0	6.7	No
36525	CHEMBL2434978	C32H36N4O4S	572.724	7 / 1	2.1	No
467452	CHEMBL3187346	C27H35N3O5	481.593	6 / 2	4.0	Yes
37006	CHEMBL2170444	C26H46N4	414.682	4 / 2	4.0	Yes
37007	CHEMBL2170299	C26H46N4	414.682	4 / 2	4.0	Yes
37008	CHEMBL2170443	C26H46N4	414.682	4 / 2	4.0	Yes
38617	CHEMBL2031837	C40H44FN7O2	673.837	6 / 4	5.2	No
38618	CHEMBL2031820	C40H44FN7O2	673.837	6 / 4	5.2	No
39800	CHEMBL2031835	C39H40FN7O3	673.793	6 / 4	4.4	No
39801	CHEMBL2031818	C39H40FN7O3	673.793	6 / 4	4.4	No
41254	CHEMBL2180078	C32H38N8O6	630.706	7 / 8	0.8	No
41781	CHEMBL480114	C27H34N10O2	530.637	4 / 7	0.0	No
42529	CHEMBL2372996	C89H137N31O20S2	2025.39	28 / 30	-8.0	No
522800	CHEMBL3828236	C29H35N3	425.62	3 / 0	5.0	Yes
43637	CHEMBL2180077	C38H48F3N11O8	843.866	13 / 11	N/A	No
43638	CHEMBL2180076	C38H48F3N11O8	843.866	13 / 11	N/A	No
522811	CHEMBL3827585	C24H26F2N2	380.483	4 / 0	4.8	Yes
548393	CHEMBL3914095	C136H215N43O31S2	3012.61	43 / 48	-7.9	No
443497	CHEMBL3357471	C27H39N7O	477.657	3 / 4	2.4	Yes
46432	CHEMBL1682860	C19H27N5	325.46	5 / 2	1.4	Yes
47791	CHEMBL516480	C20H28N4S2	388.592	4 / 1	4.0	Yes
48581	CHEMBL1092629	C21H25N5O	363.465	4 / 2	1.4	Yes
522956	CHEMBL3827508	C15H23N3O2	277.368	5 / 0	-0.2	Yes
48721	CHEMBL450815	C30H40N10O2	572.718	4 / 7	2.0	No
48722	CHEMBL501494	C30H40N10O2	572.718	4 / 7	2.0	No
48723	CHEMBL450041	C30H40N10O2	572.718	4 / 7	2.0	No
48968	CHEMBL1802280	C18H16F2N4	326.351	6 / 2	3.6	Yes
49070	CHEMBL545063	C30H57BrN6	581.732	6 / 5	N/A	No
49332	CHEMBL3091692	C29H41N5O2	491.68	6 / 1	2.1	Yes
49607	CHEMBL1802283	C18H18N4	290.37	4 / 2	3.5	Yes
469074	CHEMBL3188149	C27H35N3O6	497.592	7 / 2	3.6	Yes
50313	CHEMBL2370134	C87H134N30O18S2	1952.34	27 / 28	-7.1	No
50978	CHEMBL1088916	C23H31N5	377.536	4 / 2	3.1	Yes
537259	CHEMBL3957139	C31H40N6O	512.702	6 / 1	2.8	No
537260	CHEMBL3975192	C31H40N6O	512.702	6 / 1	2.8	No
537265	CHEMBL3918137	C33H31N5O2	529.644	5 / 0	4.3	No
537275	CHEMBL3965697	C19H17N5O4	379.376	7 / 2	3.5	Yes
52109	NSC 66832	C10H16Cl2N8	319.194	4 / 6	N/A	No
52140	AMD 3465	C24H38N6	410.61	6 / 4	0.8	Yes
53240	PharmaGSID_48521	C31H49N5O4	555.764	7 / 0	4.1	No
54309	CHEMBL545532	C28H51ClN4O4	543.19	8 / 3	N/A	No
469637	CHEMBL3627799	C26H37N5O2	451.615	6 / 2	2.1	Yes
54824	BDBM50363983	C103H142N26O24	2128.43	30 / 23	-8.0	No

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