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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Gonadotropin-releasing hormone receptor
Species	Rattus norvegicus (Rat)
Gene	Gnrhr
Synonym	luteinizing hormone-releasing hormone (LHRH) receptor luliberin receptor LHRHR LHRH receptor GNRHR1 GnRHR GnRH1 receptor GnRH-R GnRH receptor GnRH I receptor Type I GnRHR [ Show all ]
Disease	N/A for non-human GPCRs
Length	327
Amino acid sequence	MANNASLEQDQNHCSAINNSIPLTQGKLPTLTLSGKIRVTVTFFLFLLSTAFNASFLVKLQRWTQKRKKGKKLSRMKVLLKHLTLANLLETLIVMPLDGMWNITVQWYAGEFLCKVLSYLKLFSMYAPAFMMVVISLDRSLAVTQPLAVQSKSKLERSMTSLAWILSIVFAGPQLYIFRMIYLADGSGPAVFSQCVTHCSFPQWWHEAFYNFFTFSCLFIIPLLIMLICNAKIIFALTRVLHQDPRKLQLNQSKNNIPRARLRTLKMTVAFGTSFVICWTPYYVLGIWYWFDPEMLNRVSEPVNHFFFLFAFLNPCFDPLIYGYFSL
UniProt	P30969
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3066
IUPHAR	256
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
441671	CHEMBL413066	C83H110ClN15O13	1561.33	16 / 14	7.3	No
445	CHEMBL266870	C61H85N15O11	1204.44	14 / 12	2.2	No
864	CHEMBL439697	C91H124ClN25O13	1811.6	24 / 20	7.1	No
1309	CHEMBL262235	C64H79FN12O10	1195.41	12 / 12	5.3	No
1310	CHEMBL408861	C64H79FN12O10	1195.41	12 / 12	5.3	No
1384	CHEMBL88293	C24H27ClN2O2	410.942	3 / 1	5.0	Yes
1573	CHEMBL112466	C29H30F2N4O3	520.581	7 / 0	4.0	No
2999	CHEMBL50283	C29H31ClN6O3	547.056	6 / 4	3.6	No
3672	CHEMBL468551	C28H24F5N3O3	545.51	9 / 1	4.5	No
3989	CHEMBL1091579	C28H34N6O2	486.62	5 / 1	4.2	Yes
4212	nafarelin 6NMe2Nal	C67H85N17O13	1336.52	15 / 15	1.0	No
4298	CHEMBL150228	C28H32N2O3	444.575	4 / 3	5.8	No
4351	CHEMBL11134	C24H25N3	355.485	2 / 2	4.7	Yes
4405	CHEMBL2370559	C67H85N17O13	1336.52	15 / 15	1.0	No
4697	CHEMBL404991	C68H91ClN16O15	1408.02	16 / 16	0.5	No
4698	CHEMBL2371556	C68H91ClN16O15	1408.02	16 / 16	0.5	No
4923	CHEMBL2371354	C76H102ClN19O13	1525.22	15 / 18	4.3	No
5136	CHEMBL2371484	C74H93ClN18O14	1494.12	16 / 15	1.2	No
5349	CHEMBL401418	C37H54N6O2S	646.939	7 / 3	4.8	No
5428	CHEMBL423215	C28H32N2O	412.577	2 / 3	6.6	No
5781	CHEMBL407225	C67H88ClN19O12	1387.01	16 / 15	0.3	No
5942	CHEMBL317843	C38H50N10O6	742.882	8 / 7	1.0	No
6024	CHEMBL3278371	C48H75N15O14	1086.22	15 / 15	-4.1	No
6605	CHEMBL413862	C69H84ClN13O12	1322.96	13 / 13	5.4	No
7091	CHEMBL428299	C64H85ClN14O11	1261.92	13 / 12	3.8	No
7426	CHEMBL372316	C24H31N5O4S	485.603	6 / 2	4.8	Yes
7482	CHEMBL48224	C33H42N4O	510.726	3 / 2	6.2	No
7622	CHEMBL3278580	C48H77N13O12	1028.22	13 / 13	-0.7	No
8582	CHEMBL411197	C64H85FN14O13	1277.47	15 / 13	1.4	No
9008	CHEMBL407023	C64H103N21O13	1374.66	18 / 18	-1.0	No
9400	CHEMBL10929	C28H33N3	411.593	2 / 3	6.3	No
9666	CHEMBL3272533	C72H93N13O16	1396.61	17 / 14	N/A	No
10378	Relugolix	C29H27F2N7O5S	623.636	11 / 2	3.2	No
11779	CHEMBL264332	C68H86ClN17O13	1384.99	14 / 15	1.1	No
12652	CHEMBL2371508	C73H92ClN19O14	1495.11	17 / 15	0.2	No
12855	CHEMBL405961	C57H83ClN16O14	1251.84	16 / 14	-1.2	No
13069	CHEMBL46060	C26H27Cl3N4O3	549.877	4 / 4	4.9	No
13559	CHEMBL3272874	C64H85ClN14O14	1309.92	15 / 16	N/A	No
13587	CHEMBL364933	C26H28N6O4S	520.608	7 / 2	4.1	No
13924	CHEMBL48763	C35H46N4O3S	602.838	5 / 3	6.5	No
14393	CHEMBL414350	C68H91ClN16O15	1408.02	16 / 16	0.5	No
14394	CHEMBL2371582	C68H91ClN16O15	1408.02	16 / 16	0.5	No
14421	CHEMBL399857	C37H50N4O3S	630.892	5 / 1	6.2	No
14758	CHEMBL120834	C33H43ClN4O2	563.183	5 / 2	9.0	No
14867	CHEMBL343658	C28H26F6N2O	520.519	8 / 3	7.6	No
15232	WAY-207024	C30H32N6	476.628	5 / 1	5.5	No
16002	nafarelin 5NMeTyr	C67H85N17O13	1336.52	15 / 15	1.0	No
16083	CHEMBL2371351	C80H118ClN21O12	1601.41	15 / 18	4.1	No
16363	CHEMBL3272539	C65H89N13O16S	1340.56	18 / 14	N/A	No
16673	CHEMBL506877	C31H30F3N3O5	581.592	9 / 2	1.8	No
16845	CHEMBL417726	C32H38N4O2	510.682	4 / 2	5.0	No
17041	CHEMBL265169	C63H79ClN14O14	1291.86	16 / 12	1.6	No
17183	CHEMBL116246	C27H33N3O2	431.58	4 / 1	5.8	No
17212	CHEMBL416286	C36H39N3O2	545.727	3 / 4	7.4	No
19093	CHEMBL181864	C23H21ClFN3O3S	473.947	6 / 1	4.9	Yes
19214	CHEMBL2370320	C59H74N12O11	1127.31	12 / 12	3.0	No
19383	CHEMBL2371555	C64H84ClN13O15	1310.9	15 / 13	1.7	No
19384	CHEMBL410198	C64H84ClN13O15	1310.9	15 / 13	1.7	No
20078	BDBM50022926	C68H87ClN20O12	1412.02	16 / 17	0.4	No
20246	CHEMBL297927	C35H45N3O4S	603.822	6 / 3	7.0	No
20307	CHEMBL395225	C37H37F4N5O	643.731	8 / 2	6.4	No
20410	BDBM50085774	C71H91ClN18O14	1456.07	15 / 17	1.2	No
20470	CHEMBL3144569	C40H43Cl2N7O6	788.727	9 / 4	5.1	No
21193	CHEMBL86365	C22H23ClN2O2	382.888	3 / 1	4.2	Yes
21812	CHEMBL487627	C21H18F6N6	468.407	10 / 2	4.3	Yes
22015	CHEMBL91311	C25H30N2O2	390.527	3 / 1	4.5	Yes
22133	BDBM50085799	C69H87ClN18O14	1428.02	15 / 17	0.5	No
22134	CID 44380271	C69H87ClN18O14	1428.02	15 / 16	0.1	No
23203	CHEMBL268108	C60H91ClN18O14	1323.95	16 / 17	-2.0	No
23204	CHEMBL2371584	C60H91ClN18O14	1323.95	16 / 17	-2.0	No
23442	CHEMBL364246	C28H31N5O4S	533.647	6 / 2	5.5	No
24740	CHEMBL262977	C61H77N13O10	1152.37	11 / 13	3.8	No
25167	CHEMBL131665	C41H42FN5O4	687.816	9 / 0	7.2	No
25361	CHEMBL11087	C27H31N3	397.566	2 / 2	5.9	No
27450	CHEMBL410818	C81H103ClN16O15	1576.26	17 / 14	4.7	No
27451	CHEMBL408335	C81H103ClN16O15	1576.26	17 / 14	4.7	No
27866	CHEMBL342396	C31H31ClF3N5O5	646.064	11 / 4	N/A	No
28350	CHEMBL305358	C22H17Cl2N3O4	458.295	5 / 0	4.0	Yes
28462	CHEMBL359370	C27H30N2O5	462.546	6 / 4	4.2	Yes
28463	CHEMBL149189	C27H30N2O5	462.546	6 / 4	4.2	Yes
29328	CHEMBL2370313	C34H50N8O5	650.825	6 / 6	2.2	No
29937	CHEMBL197317	C26H35N7O5S	557.67	8 / 4	2.7	No
29944	CHEMBL90726	C26H30N2O4	434.536	5 / 1	4.0	Yes
30222	CID 44379956	C71H91ClN18O14	1456.07	15 / 16	0.8	No
30223	CID 44380257	C71H91ClN18O14	1456.07	15 / 16	0.8	No
31286	CHEMBL401349	C36H49N5O2S	615.881	5 / 1	6.1	No
31287	CHEMBL2370317	C30H44N8O5	596.733	6 / 7	1.1	No
31601	CHEMBL119856	C29H36N2O2	444.619	3 / 2	6.4	No
31812	CHEMBL45661	C23H24ClN3O4	441.912	5 / 2	4.3	Yes
32169	CHEMBL407615	C80H101ClN16O15	1562.23	17 / 15	4.4	No
32170	CHEMBL267642	C80H101ClN16O15	1562.23	17 / 15	4.4	No
32323	CHEMBL262373	C64H88ClN19O14	1382.98	17 / 15	-2.1	No
33079	CHEMBL3272879	C66H88N14O15	1317.51	16 / 15	N/A	No
33685	CHEMBL429723	C63H84FN19O12	1318.48	16 / 18	-1.1	No
33862	CHEMBL407073	C64H80FN13O10	1210.42	12 / 12	4.5	No
34440	CHEMBL123301	C33H38N4O2	522.693	5 / 2	7.6	No
34474	CHEMBL2371522	C74H92Cl2N18O14	1528.56	16 / 15	1.9	No
34506	CHEMBL413896	C57H81ClN18O14	1277.84	16 / 15	-3.4	No
443035	CHEMBL263488	C81H106ClN15O13	1533.28	16 / 14	6.5	No
35016	CHEMBL3272882	C73H94N14O15	1407.64	16 / 15	N/A	No

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