# | PDB (Resolution Å) |
Site # | Ligand | EC number | GO terms | UniProt | PubMed | Binding affinity |
---|---|---|---|---|---|---|---|---|
1 | 2qyk:A (2.1) | BS01 | NPV | 3.1.4.53 | GO:0004114 ... | P27815 | 17727341 | MOAD: ic50=3.3uM PDBbind: -logKd/Ki=5.48, IC50=3.3uM BindingDB: IC50=3300nM, EC50=20nM |
2 | 2qyk:B (2.1) | BS01 | NPV | 3.1.4.53 | GO:0004114 ... | P27815 | 17727341 | MOAD: ic50=3.3uM BindingDB: IC50=3300nM, EC50=20nM |
3 | 2qyl:A (1.95) | BS03 | NPV | 3.1.4.53 | GO:0004114 ... | Q07343 | 17727341 | MOAD: ic50=0.65uM PDBbind: -logKd/Ki=6.19, IC50=0.65uM BindingDB: IC50=650nM |
4 | 2qyn:A (1.57) | BS01 | NPV | 3.1.4.53 | GO:0004114 ... | Q08499 | 17727341 | MOAD: ic50=0.57uM PDBbind: -logKd/Ki=6.24, IC50=0.57uM BindingDB: IC50=1nM |
5 | 2qyn:B (1.57) | BS01 | NPV | 3.1.4.53 | GO:0004114 ... | Q08499 | 17727341 | MOAD: ic50=0.57uM BindingDB: IC50=1nM |