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BioLiP Library
Download all results in tab-seperated text for 3964 receptor-ligand interactions, whose format is explained at readme.txt.
  • Hover over PDB to view the title of the structure. Click PDB to view the structure at the RCSB PDB database. Resolution -1.00 means the resolution is unavailable, e.g., for NMR structures.
  • Click Site # to view the binding site structure. Hover over Site # to view the binding residues.
  • Hover over Ligand to view the full ligand name. Click Ligand to view the 2D diagram and other detail information of the ligand.
  • Hover over EC number to view the full name of enzymatic activity.
  • Hover over GO terms to view all GO terms.
  • Hover over UniProt to view the protein name.
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    # PDB
    (Resolution Å)
    Site # Ligand EC number GO terms UniProt PubMed Binding
    affinity
    1401 4fpa:A (2.48) BS01 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1402 4fpa:A (2.48) BS03 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1403 4fpa:B (2.48) BS01 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1404 4fpa:B (2.48) BS03 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1405 4fpb:A (3.0) BS01 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1406 4fpb:A (3.0) BS03 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1407 4fpb:B (3.0) BS01 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1408 4fpb:B (3.0) BS03 BGC 2.7.1.1 GO:0001678 ... P19367 N/A
    1409 4fus:A (1.75) BS01 BGC 3.2.1.4 GO:0004553 ... Q2SJA2 23055526
    1410 4fus:A (1.75) BS02 BGC 3.2.1.4 GO:0004553 ... Q2SJA2 23055526
    1411 4gal:B (1.95) BS01 BGC ? GO:0005515 ... P47929 9760227
    1412 4gbz:A (2.894) BS01 BGC ? GO:0005886 ... P0AGF4 23075985
    1413 4gey:A (2.7) BS01 BGC ? GO:0008643 ... A5VZA8 23066028
    1414 4gn9:A (2.0) BS02 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1415 4gn9:A (2.0) BS03 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1416 4gn9:A (2.0) BS04 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1417 4gn9:B (2.0) BS02 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1418 4gn9:B (2.0) BS03 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1419 4gn9:B (2.0) BS04 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1420 4gn9:B (2.0) BS05 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1421 4gn9:B (2.0) BS06 BGC 3.1.1.17 GO:0001822 ... Q64374 23349732
    1422 4gpn:B (2.291) BS01 BGC 3.2.1.86 GO:0004553 ... Q8DT00 23519420
    1423 4gzi:A (1.68) BS01 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1424 4gzi:A (1.68) BS02 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1425 4gzi:A (1.68) BS03 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1426 4gzj:A (1.55) BS01 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1427 4gzj:A (1.55) BS02 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1428 4gzj:A (1.55) BS03 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1429 4gzj:A (1.55) BS04 BGC 3.2.1.39 GO:0004553 ... Q70C53 23275163
    1430 4hap:A (1.6) BS01 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1431 4hap:A (1.6) BS02 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1432 4hap:B (1.6) BS01 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1433 4hap:B (1.6) BS02 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1434 4haq:A (1.9) BS01 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1435 4haq:A (1.9) BS02 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1436 4haq:B (1.9) BS01 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1437 4haq:B (1.9) BS02 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1438 4hg6:A (3.25) BS01 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1439 4hg6:A (3.25) BS02 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1440 4hg6:A (3.25) BS03 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1441 4hg6:A (3.25) BS04 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1442 4hg6:A (3.25) BS05 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1443 4hg6:A (3.25) BS06 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1444 4hg6:A (3.25) BS07 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1445 4hg6:A (3.25) BS08 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1446 4hg6:A (3.25) BS09 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1447 4hg6:A (3.25) BS10 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1448 4hg6:A (3.25) BS11 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1449 4hg6:A (3.25) BS12 BGC 2.4.1.12 GO:0000166 ... Q3J125 23222542
    1450 4hg6:B (3.25) BS01 BGC ? GO:0005515 ... Q3J126 23222542
    1451 4hg6:B (3.25) BS02 BGC ? GO:0005515 ... Q3J126 23222542
    1452 4hoa:A (2.0) BS01 BGC 3.2.2.22 GO:0000166 ... D9J2T9 N/A
    1453 4hql:A (2.241) BS01 BGC ? N/A Q9TVF0 23236185
    1454 4hqn:A (2.196) BS01 BGC ? N/A Q9TVF0 23236185
    1455 4hu0:A (2.38) BS01 BGC ? GO:0000272 ... I6PLH5 N/A
    1456 4hu0:A (2.38) BS02 BGC ? GO:0000272 ... I6PLH5 N/A
    1457 4hu0:A (2.38) BS03 BGC ? GO:0000272 ... I6PLH5 N/A
    1458 4hz7:A (2.0) BS01 BGC 3.2.1.21 GO:0004553 ... Q0GMU3 20005197
    1459 4hz8:A (1.14) BS01 BGC 3.2.1.21 GO:0004553 ... Q0GMU3 20005197
    1460 4i3g:A (1.4) BS01 BGC ? GO:0004553 ... C5IXN7 23225731
    1461 4i3g:B (1.4) BS01 BGC ? GO:0004553 ... C5IXN7 23225731
    1462 4i8d:A (2.48) BS02 BGC 3.2.1.21 GO:0000272 ... Q12715 25164811
    1463 4i8d:B (2.48) BS01 BGC 3.2.1.21 GO:0000272 ... Q12715 25164811
    1464 4ibl:L (1.8) BS01 BGC 3.4.21.21 GO:0005509 ... P08709 N/A
    1465 4iig:A (2.3) BS08 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1466 4iig:A (2.3) BS09 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1467 4iig:B (2.3) BS08 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1468 4iig:B (2.3) BS09 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1469 4iih:A (2.0) BS09 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1470 4iih:B (2.0) BS09 BGC 3.2.1.21 GO:0004553 ... P48825 23537284
    1471 4ipm:A (1.14) BS02 BGC 3.2.1.91 GO:0004553 ... D4HRL0 23733951
    1472 4jcw:A (1.75) BS01 BGC 3.2.1.4 N/A A5CLK3 N/A
    1473 4jcw:A (1.75) BS02 BGC 3.2.1.4 N/A A5CLK3 N/A
    1474 4jcw:A (1.75) BS03 BGC 3.2.1.4 N/A A5CLK3 N/A
    1475 4jcw:B (1.75) BS01 BGC 3.2.1.4 N/A A5CLK3 N/A
    1476 4jcw:B (1.75) BS02 BGC 3.2.1.4 N/A A5CLK3 N/A
    1477 4jcw:B (1.75) BS03 BGC 3.2.1.4 N/A A5CLK3 N/A
    1478 4jcw:B (1.75) BS04 BGC 3.2.1.4 N/A A5CLK3 N/A
    1479 4jjj:A (1.6) BS01 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1480 4jjj:A (1.6) BS02 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1481 4jjj:A (1.6) BS04 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1482 4jjj:A (1.6) BS05 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1483 4jjj:A (1.6) BS06 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1484 4jjj:A (1.6) BS07 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1485 4jjj:A (1.6) BS08 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1486 4jjj:A (1.6) BS09 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1487 4jjj:A (1.6) BS10 BGC 3.2.1.91 GO:0004553 ... Q47NH7 24264519
    1488 4jsd:A (2.05) BS01 BGC ? GO:0015833 ... Q9WXN8 24090243
    1489 4jsd:A (2.05) BS02 BGC ? GO:0015833 ... Q9WXN8 24090243
    1490 4jso:A (2.07) BS01 BGC ? GO:0015833 ... Q9WXN8 24090243
    1491 4jso:A (2.07) BS02 BGC ? GO:0015833 ... Q9WXN8 24090243
    1492 4jso:A (2.07) BS03 BGC ? GO:0015833 ... Q9WXN8 24090243
    1493 4jso:A (2.07) BS04 BGC ? GO:0015833 ... Q9WXN8 24090243
    1494 4jso:A (2.07) BS05 BGC ? GO:0015833 ... Q9WXN8 24090243
    1495 4kbb:A (2.3) BS04 BGC 3.4.24.69 GO:0005576 ... P10844 23807078
    1496 4kbb:B (2.3) BS02 BGC 3.4.24.69 GO:0005576 ... P10844 23807078
    1497 4kkv:A (1.74) BS01 BGC 2.7.7.2 GO:0000287 ... Q6FNA9 23663086
    1498 4kqm:C (2.77) BS02 BGC 2.4.1.11 GO:0004373 ... P27472 24324135
    1499 4ktp:A (1.9) BS01 BGC 2.4.1.332 GO:0003824 ... D6XZ22 24828502
    1500 4ktp:B (1.9) BS01 BGC 2.4.1.332 GO:0003824 ... D6XZ22 24828502
    1501 4kwu:A (1.9) BS03 BGC ? GO:0003824 ... Q8Y4J2 N/A
    1502 4kwu:A (1.9) BS04 BGC ? GO:0003824 ... Q8Y4J2 N/A
    1503 4kwu:A (1.9) BS05 BGC ? GO:0003824 ... Q8Y4J2 N/A
    1504 4kwu:A (1.9) BS06 BGC ? GO:0003824 ... Q8Y4J2 N/A
    1505 4l0g:A (2.0) BS01 BGC 3.2.1.4 GO:0004553 ... B9MKU7 N/A
    1506 4l0g:A (2.0) BS02 BGC 3.2.1.4 GO:0004553 ... B9MKU7 N/A
    1507 4l48:A (2.1) BS01 BGC 3.2.1.4 N/A A5CLK3 N/A
    1508 4l48:A (2.1) BS02 BGC 3.2.1.4 N/A A5CLK3 N/A
    1509 4l48:A (2.1) BS03 BGC 3.2.1.4 N/A A5CLK3 N/A
    1510 4l48:A (2.1) BS04 BGC 3.2.1.4 N/A A5CLK3 N/A
    1511 4l48:C (2.1) BS01 BGC 3.2.1.4 N/A A5CLK3 N/A
    1512 4l48:C (2.1) BS02 BGC 3.2.1.4 N/A A5CLK3 N/A
    1513 4l48:C (2.1) BS03 BGC 3.2.1.4 N/A A5CLK3 N/A
    1514 4lbj:A (1.8) BS01 BGC ? GO:0030246 ... P17931 24326249
    1515 4lbk:A (1.6) BS01 BGC ? GO:0030246 ... P17931 24326249
    1516 4lbl:A (1.58) BS01 BGC ? GO:0030246 ... P17931 24326249 PDBbind: -logKd/Ki=4.96, Kd=11uM
    1517 4lbm:A (1.55) BS01 BGC ? GO:0030246 ... P17931 24326249
    1518 4lbo:A (1.65) BS01 BGC ? GO:0030246 ... P17931 24326249 PDBbind: -logKd/Ki=5.77, Kd=1.7uM
    1519 4le4:D (1.8) BS01 BGC ? N/A J7K096 N/A
    1520 4lef:B (1.842) BS03 BGC 3.1.-.- GO:0008270 ... P45548 N/A
    1521 4lef:C (1.842) BS03 BGC 3.1.-.- GO:0008270 ... P45548 N/A
    1522 4lpc:B (2.39) BS01 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1523 4lpc:B (2.39) BS03 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1524 4lpc:B (2.39) BS08 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1525 4lpc:B (2.39) BS10 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1526 4lpc:D (2.39) BS05 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1527 4lq1:A (2.55) BS01 BGC 2.4.1.18 GO:0003824 ... P07762 26280198
    1528 4m24:A (1.386) BS01 BGC 3.2.1.4 GO:0000272 ... C1JI15 N/A
    1529 4m24:A (1.386) BS02 BGC 3.2.1.4 GO:0000272 ... C1JI15 N/A
    1530 4m82:A (1.592) BS02 BGC 2.4.1.-
    3.2.1.58
    GO:0000272 ... P29717 24804868
    1531 4n2z:A (1.8) BS02 BGC 3.2.1.55 GO:0005576 ... E2GHW5 24394409
    1532 4n2z:A (1.8) BS03 BGC 3.2.1.55 GO:0005576 ... E2GHW5 24394409
    1533 4nfu:A (2.21) BS01 BGC 3.-.-.- GO:0005634 ... Q9XF23 24331460
    1534 4no4:A (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1535 4no4:B (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1536 4no4:C (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1537 4no4:D (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1538 4no4:E (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1539 4no4:F (1.399) BS01 BGC ? GO:0002317 ... P11762 N/A
    1540 4ojl:A (2.0) BS01 BGC ? GO:0019058 ... G3M189 24671238
    1541 4ojl:B (2.0) BS01 BGC ? GO:0019058 ... G3M189 24671238
    1542 4ojl:C (2.0) BS01 BGC ? GO:0019058 ... G3M189 24671238
    1543 4ojl:C (2.0) BS02 BGC ? GO:0019058 ... G3M189 24671238
    1544 4p00:A (3.2) BS01 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1545 4p00:A (3.2) BS02 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1546 4p00:A (3.2) BS03 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1547 4p00:A (3.2) BS04 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1548 4p00:A (3.2) BS05 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1549 4p00:A (3.2) BS06 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1550 4p00:A (3.2) BS07 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1551 4p00:A (3.2) BS08 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1552 4p00:A (3.2) BS09 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1553 4p00:B (3.2) BS01 BGC ? GO:0006011 ... Q3J126 24704788
    1554 4p00:B (3.2) BS02 BGC ? GO:0006011 ... Q3J126 24704788
    1555 4p00:B (3.2) BS03 BGC ? GO:0006011 ... Q3J126 24704788
    1556 4p02:A (2.65) BS01 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1557 4p02:A (2.65) BS02 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1558 4p02:A (2.65) BS03 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1559 4p02:A (2.65) BS04 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1560 4p02:A (2.65) BS05 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1561 4p02:A (2.65) BS06 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1562 4p02:A (2.65) BS07 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1563 4p02:A (2.65) BS08 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1564 4p02:A (2.65) BS09 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1565 4p02:A (2.65) BS10 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1566 4p02:A (2.65) BS11 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1567 4p02:A (2.65) BS12 BGC 2.4.1.12 GO:0000166 ... Q3J125 24704788
    1568 4p02:B (2.65) BS02 BGC ? GO:0006011 ... Q3J126 24704788
    1569 4p02:B (2.65) BS03 BGC ? GO:0006011 ... Q3J126 24704788
    1570 4p02:B (2.65) BS04 BGC ? GO:0006011 ... Q3J126 24704788
    1571 4pex:B (1.75) BS01 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1572 4pey:A (1.5) BS01 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1573 4pey:A (1.5) BS02 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1574 4pey:A (1.5) BS03 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1575 4pey:A (1.5) BS04 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1576 4pey:A (1.5) BS05 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1577 4pey:A (1.5) BS06 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1578 4pez:A (1.9) BS01 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1579 4pez:A (1.9) BS02 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1580 4pez:A (1.9) BS03 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1581 4pez:A (1.9) BS04 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1582 4pf0:A (1.75) BS01 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1583 4pf0:A (1.75) BS02 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1584 4pf0:A (1.75) BS03 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1585 4pf0:A (1.75) BS04 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1586 4pf0:A (1.75) BS05 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1587 4pf0:A (1.75) BS06 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1588 4pf0:A (1.75) BS07 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1589 4pf0:A (1.75) BS08 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1590 4pf0:B (1.75) BS01 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1591 4pf0:B (1.75) BS02 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1592 4pf0:B (1.75) BS03 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1593 4pf0:B (1.75) BS04 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1594 4pf0:B (1.75) BS05 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1595 4pf0:B (1.75) BS06 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1596 4pf0:B (1.75) BS07 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1597 4pf0:B (1.75) BS08 BGC 3.2.1.58 GO:0000272 ... G2NFJ9 25752603
    1598 4ptv:A (1.85) BS02 BGC 3.2.1.21 GO:0004553 ... B8CYA8 25173693
    1599 4ptv:B (1.85) BS02 BGC 3.2.1.21 GO:0004553 ... B8CYA8 25173693
    1600 4ptx:A (1.8) BS01 BGC 3.2.1.21 GO:0004553 ... B8CYA8 25173693

    Reference:
    • Chengxin Zhang, Xi Zhang, Peter L Freddolino, and Yang Zhang. BioLiP2: an updated structure database for biologically relevent ligand-protein interactions, Nucleic Acids Research, gkad630 (2023)(download the PDF file).
    • Jianyi Yang, Ambrish Roy, and Yang Zhang. BioLiP: a semi-manually curated database for biologically relevant ligand-protein interactions, Nucleic Acids Research, 41: D1096-D1103 (2013) (download the PDF file).

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