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BioLiP
Download all results in tab-seperated text for 594392 receptor-ligand interactions, whose format is explained at readme.txt.
  • Hover over PDB to view the title of the structure. Click PDB to view the structure at the RCSB PDB database. Resolution -1.00 means the resolution is unavailable, e.g., for NMR structures.
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  • Hover over Ligand to view the full ligand name. Click Ligand to view the 2D diagram and other detail information of the ligand.
  • Hover over EC number to view the full name of enzymatic activity.
  • Hover over GO terms to view all GO terms.
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    # PDB
    (Resolution Å)
    Site # Ligand EC number GO terms UniProt PubMed Binding
    affinity
    135401 4keb:B (1.45) BS01 NDP 1.5.1.3 GO:0000900 ... P00374 24053334
    135402 4keg:A (2.5) BS01 MG ? GO:0002395 ... P0AEX9
    Q9NP55
    N/A
    135403 4keh:A (1.901) BS01 1R3 4.2.1.59
    5.3.3.14
    GO:0005737 ... P0A6Q3 24362570
    135404 4keh:A (1.901) BS02 1R3 4.2.1.59
    5.3.3.14
    GO:0005737 ... P0A6Q3 24362570
    135405 4keh:B (1.901) BS01 1R3 4.2.1.59
    5.3.3.14
    GO:0005737 ... P0A6Q3 24362570
    135406 4keh:B (1.901) BS02 1R3 4.2.1.59
    5.3.3.14
    GO:0005737 ... P0A6Q3 24362570
    135407 4kel:A (1.148) BS01 peptide 3.4.21.- GO:0004252 ... Q9Y5K2 31058493
    135408 4ken:B (1.89) BS01 1S7 3.5.2.6 GO:0008800 ... P00811 N/A
    135409 4kf6:A (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135410 4kf6:A (3.195) BS02 1T9 ? GO:0005543 ... Q5TA50 23863933
    135411 4kf6:B (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135412 4kf6:C (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135413 4kf6:D (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135414 4kf6:E (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135415 4kf6:F (3.195) BS01 1T9 ? GO:0005543 ... Q5TA50 23863933
    135416 4kfc:A (2.53) BS01 dna ? GO:0000156 ... P21866 24526190
    135417 4kfc:A (2.53) BS02 dna ? GO:0000156 ... P21866 24526190
    135418 4kfc:B (2.53) BS01 dna ? GO:0000156 ... P21866 24526190
    135419 4kfc:B (2.53) BS02 dna ? GO:0000156 ... P21866 24526190
    135420 4kfd:A (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135421 4kfd:B (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135422 4kfd:C (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135423 4kfd:D (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135424 4kfd:E (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135425 4kfd:F (1.69) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135426 4kfe:A (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135427 4kfe:B (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135428 4kfe:C (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135429 4kfe:D (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135430 4kfe:E (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135431 4kfe:F (2.1) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135432 4kff:A (2.15) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135433 4kff:B (2.15) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135434 4kff:C (2.15) BS01 CU 1.4.3.21 GO:0005507 ... P12807 N/A
    135435 4kfj:A (1.76) BS01 NDP 1.5.1.3 GO:0000900 ... P00374 24053334
    135436 4kfj:A (1.76) BS02 1R0 1.5.1.3 GO:0000900 ... P00374 24053334 MOAD: ic50=60nM
    BindingDB: IC50=60nM
    135437 4kfj:A (1.76) BS03 MG 1.5.1.3 GO:0000900 ... P00374 24053334
    135438 4kfj:A (1.76) BS04 MG 1.5.1.3 GO:0000900 ... P00374 24053334
    135439 4kfj:B (1.76) BS01 NDP 1.5.1.3 GO:0000900 ... P00374 24053334
    135440 4kfj:B (1.76) BS02 MG 1.5.1.3 GO:0000900 ... P00374 24053334
    135441 4kfm:A (3.45) BS01 PIO ? GO:0005242 ... P48542 23739333
    135442 4kfn:A (1.6) BS01 1QR 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=9.0nM
    135443 4kfn:B (1.6) BS01 1QR 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=9.0nM
    135444 4kfo:A (1.6) BS01 1QS 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=5.0nM, EC50=1.1nM
    135445 4kfo:A (1.6) BS02 1QS 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=5.0nM, EC50=1.1nM
    135446 4kfo:B (1.6) BS01 1QS 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=5.0nM, EC50=1.1nM
    135447 4kfo:B (1.6) BS02 1QS 2.4.2.12 GO:0005125 ... P43490 23617784 BindingDB: IC50=5.0nM, EC50=1.1nM
    135448 4kfp:A (1.84) BS01 1R7 2.4.2.12 GO:0005125 ... P43490 23899614 MOAD: ic50=0.01uM
    PDBbind: -logKd/Ki=8.00, IC50=10nM
    135449 4kfp:B (1.84) BS01 1R7 2.4.2.12 GO:0005125 ... P43490 23899614 MOAD: ic50=0.01uM
    PDBbind: -logKd/Ki=8.00, IC50=10nM
    135450 4kfq:A (2.2) BS01 KFQ ? GO:0015276 ... P35439 24072709 PDBbind: -logKd/Ki=8.23, Kd=5.86nM
    135451 4kfq:B (2.2) BS01 KFQ ? GO:0015276 ... P35439 24072709
    135452 4kfz:A (2.8) BS01 ZN ? GO:0001221 ... P25791 24407558
    135453 4kfz:A (2.8) BS02 ZN ? GO:0001221 ... P25791 24407558
    135454 4kfz:A (2.8) BS03 ZN ? GO:0001221 ... P25791 24407558
    135455 4kfz:A (2.8) BS04 ZN ? GO:0001221 ... P25791 24407558
    135456 4kfz:B (2.8) BS01 ZN ? GO:0001221 ... P25791 24407558
    135457 4kfz:B (2.8) BS02 ZN ? GO:0001221 ... P25791 24407558
    135458 4kfz:B (2.8) BS03 ZN ? GO:0001221 ... P25791 24407558
    135459 4kfz:B (2.8) BS04 ZN ? GO:0001221 ... P25791 24407558
    135460 4kg2:A (1.89) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135461 4kg2:B (1.89) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135462 4kg5:A (2.11) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135463 4kg5:B (2.11) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135464 4kg5:C (2.11) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135465 4kg5:D (2.11) BS01 CEF 3.5.2.6 GO:0008800 ... P00811 N/A
    135466 4kga:A (2.32) BS01 NI 3.4.21.- GO:0004252 ... Q9Y5K2 27767076
    135467 4kga:A (2.32) BS02 NI 3.4.21.- GO:0004252 ... Q9Y5K2 27767076
    135468 4kga:B (2.32) BS01 NI 3.4.21.- GO:0004252 ... Q9Y5K2 27767076
    135469 4kga:B (2.32) BS02 NI 3.4.21.- GO:0004252 ... Q9Y5K2 27767076
    135470 4kgc:A (2.69) BS01 dna ? GO:0000786 ... P84233 24637564
    135471 4kgc:A (2.69) BS02 dna ? GO:0000786 ... P84233 24637564
    135472 4kgc:B (2.69) BS01 dna ? GO:0000786 ... P62799 24637564
    135473 4kgc:B (2.69) BS02 dna ? GO:0000786 ... P62799 24637564
    135474 4kgc:C (2.69) BS01 dna ? GO:0000786 ... Q6AZJ8 24637564
    135475 4kgc:C (2.69) BS02 dna ? GO:0000786 ... Q6AZJ8 24637564
    135476 4kgc:D (2.69) BS01 dna ? GO:0000786 ... P02281 24637564
    135477 4kgc:D (2.69) BS02 dna ? GO:0000786 ... P02281 24637564
    135478 4kgc:E (2.69) BS01 dna ? GO:0000786 ... P84233 24637564
    135479 4kgc:E (2.69) BS02 dna ? GO:0000786 ... P84233 24637564
    135480 4kgc:F (2.69) BS01 dna ? GO:0000786 ... P62799 24637564
    135481 4kgc:F (2.69) BS02 dna ? GO:0000786 ... P62799 24637564
    135482 4kgc:G (2.69) BS01 dna ? GO:0000786 ... Q6AZJ8 24637564
    135483 4kgc:G (2.69) BS02 dna ? GO:0000786 ... Q6AZJ8 24637564
    135484 4kgc:G (2.69) BS03 HRU ? GO:0000786 ... Q6AZJ8 24637564
    135485 4kgc:H (2.69) BS01 dna ? GO:0000786 ... P02281 24637564
    135486 4kgc:H (2.69) BS02 dna ? GO:0000786 ... P02281 24637564
    135487 4kgn:A (2.15) BS01 SAH 2.1.1.207 GO:0001510 ... Q3JWH1 N/A
    135488 4kgn:C (2.15) BS01 SAH 2.1.1.207 GO:0001510 ... Q3JWH1 N/A
    135489 4kgn:E (2.15) BS01 SAH 2.1.1.207 GO:0001510 ... Q3JWH1 N/A
    135490 4kgn:G (2.15) BS01 SAH 2.1.1.207 GO:0001510 ... Q3JWH1 N/A
    135491 4kgv:B (2.1) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135492 4kgv:B (2.1) BS02 ATP N/A GO:0006207 ... N/A 24138583
    135493 4kgv:D (2.1) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135494 4kgv:D (2.1) BS02 ATP N/A GO:0006207 ... N/A 24138583
    135495 4kgx:B (2.202) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135496 4kgx:B (2.202) BS02 CTP N/A GO:0006207 ... N/A 24138583
    135497 4kgx:D (2.202) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135498 4kgx:D (2.202) BS02 CTP N/A GO:0006207 ... N/A 24138583
    135499 4kgz:B (2.4) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135500 4kgz:B (2.4) BS02 UTP N/A GO:0006207 ... N/A 24138583
    135501 4kgz:B (2.4) BS03 UTP N/A GO:0006207 ... N/A 24138583
    135502 4kgz:D (2.4) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135503 4kgz:D (2.4) BS02 UTP N/A GO:0006207 ... N/A 24138583
    135504 4kgz:D (2.4) BS03 UTP N/A GO:0006207 ... N/A 24138583
    135505 4kh0:B (2.25) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135506 4kh0:B (2.25) BS02 ATP N/A GO:0006207 ... N/A 24138583
    135507 4kh0:B (2.25) BS03 ATP N/A GO:0006207 ... N/A 24138583
    135508 4kh0:B (2.25) BS04 ATP N/A GO:0006207 ... N/A 24138583
    135509 4kh0:B (2.25) BS05 ATP N/A GO:0006207 ... N/A 24138583
    135510 4kh0:D (2.25) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135511 4kh0:D (2.25) BS02 ATP N/A GO:0006207 ... N/A 24138583
    135512 4kh0:D (2.25) BS03 ATP N/A GO:0006207 ... N/A 24138583
    135513 4kh1:B (2.2) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135514 4kh1:B (2.2) BS02 CTP N/A GO:0006207 ... N/A 24138583
    135515 4kh1:B (2.2) BS03 UTP N/A GO:0006207 ... N/A 24138583
    135516 4kh1:D (2.2) BS01 ZN N/A GO:0006207 ... N/A 24138583
    135517 4kh1:D (2.2) BS02 CTP N/A GO:0006207 ... N/A 24138583
    135518 4kh1:D (2.2) BS03 UTP N/A GO:0006207 ... N/A 24138583
    135519 4kh4:A (3.0) BS01 ANP 3.6.1.15 GO:0005576 ... Q27895 24115522
    135520 4kh4:B (3.0) BS01 ANP 3.6.1.15 GO:0005576 ... Q27895 24115522
    135521 4kh5:A (3.0) BS01 AU1 3.6.1.15 GO:0005576 ... Q27895 24115522
    135522 4kh5:B (3.0) BS01 AU1 3.6.1.15 GO:0005576 ... Q27895 24115522
    135523 4kh6:A (2.4) BS01 AU1 3.6.1.15 GO:0005576 ... Q27895 24115522
    135524 4kh6:B (2.4) BS01 AU1 3.6.1.15 GO:0005576 ... Q27895 24115522
    135525 4kho:A (2.0) BS01 CA ? GO:0035101 ... G0SDN1 23698368
    135526 4kho:B (2.0) BS01 CA ? GO:0035101 ... G0SDN1 23698368
    135527 4khp:B (3.1) BS01 rna ? GO:0003735 ... P80371 23702293
    135528 4khp:D (3.1) BS01 rna ? GO:0003723 ... P80373 23702293
    135529 4khp:D (3.1) BS02 MG ? GO:0003723 ... P80373 23702293
    135530 4khp:E (3.1) BS01 rna ? GO:0003723 ... Q5SHQ5 23702293
    135531 4khp:F (3.1) BS01 rna ? GO:0003735 ... Q5SLP8 23702293
    135532 4khp:G (3.1) BS01 rna ? GO:0000028 ... P17291 23702293
    135533 4khp:G (3.1) BS02 rna ? GO:0000028 ... P17291 23702293
    135534 4khp:H (3.1) BS01 rna N/A GO:0003735 ... N/A 23702293
    135535 4khp:I (3.1) BS01 rna ? GO:0000049 ... P80374 23702293
    135536 4khp:J (3.1) BS01 rna ? GO:0000049 ... Q5SHN7 23702293
    135537 4khp:K (3.1) BS01 rna ? GO:0003735 ... P80376 23702293
    135538 4khp:K (3.1) BS02 MG ? GO:0003735 ... P80376 23702293
    135539 4khp:L (3.1) BS01 rna ? GO:0000049 ... Q5SHN3 23702293
    135540 4khp:L (3.1) BS02 MG ? GO:0000049 ... Q5SHN3 23702293
    135541 4khp:M (3.1) BS01 rna ? GO:0000049 ... P80377 23702293
    135542 4khp:N (3.1) BS01 rna N/A GO:0003735 ... N/A 23702293
    135543 4khp:O (3.1) BS01 rna ? GO:0003735 ... Q5SJ76 23702293
    135544 4khp:P (3.1) BS01 rna ? GO:0003735 ... Q5SJH3 23702293
    135545 4khp:Q (3.1) BS01 rna N/A GO:0003735 ... N/A 23702293
    135546 4khp:R (3.1) BS01 rna ? GO:0003735 ... Q5SLQ0 23702293
    135547 4khp:S (3.1) BS01 rna ? GO:0003723 ... Q5SHP2 23702293
    135548 4khp:S (3.1) BS02 MG ? GO:0003723 ... Q5SHP2 23702293
    135549 4khp:T (3.1) BS01 rna ? GO:0003723 ... P80380 23702293
    135550 4khz:E (2.9) BS01 GLC ? GO:0005515 ... P0AEX9 24145421
    135551 4khz:E (2.9) BS02 GLC ? GO:0005515 ... P0AEX9 24145421
    135552 4khz:E (2.9) BS03 GLC ? GO:0005515 ... P0AEX9 24145421
    135553 4khz:E (2.9) BS04 GLC ? GO:0005515 ... P0AEX9 24145421
    135554 4khz:F (2.9) BS01 GLC ? GO:0005515 ... P02916 24145421
    135555 4khz:F (2.9) BS02 GLC ? GO:0005515 ... P02916 24145421
    135556 4ki0:A (2.38) BS01 MG 7.5.2.1 GO:0005515 ... P68187 24145421
    135557 4ki0:A (2.38) BS02 ANP 7.5.2.1 GO:0005515 ... P68187 24145421
    135558 4ki0:A (2.38) BS03 ANP 7.5.2.1 GO:0005515 ... P68187 24145421
    135559 4ki0:B (2.38) BS01 ANP 7.5.2.1 GO:0005515 ... P68187 24145421
    135560 4ki0:B (2.38) BS02 MG 7.5.2.1 GO:0005515 ... P68187 24145421
    135561 4ki0:B (2.38) BS03 ANP 7.5.2.1 GO:0005515 ... P68187 24145421
    135562 4ki0:F (2.38) BS01 GLC ? GO:0005515 ... P02916 24145421
    135563 4ki0:F (2.38) BS02 GLC ? GO:0005515 ... P02916 24145421
    135564 4ki7:A (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135565 4ki7:B (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135566 4ki7:C (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135567 4ki7:D (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135568 4ki7:E (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135569 4ki7:F (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135570 4ki7:G (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135571 4ki7:H (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135572 4ki7:I (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135573 4ki7:J (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135574 4ki7:K (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135575 4ki7:L (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135576 4ki7:N (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135577 4ki7:O (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135578 4ki7:P (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135579 4ki7:Q (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135580 4ki7:R (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135581 4ki7:S (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135582 4ki7:T (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135583 4ki7:U (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135584 4ki7:V (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135585 4ki7:W (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135586 4ki7:X (2.8) BS01 1R2 4.2.1.10 GO:0003855 ... P9WPX7 25234229
    135587 4ki8:A (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135588 4ki8:B (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135589 4ki8:C (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135590 4ki8:D (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135591 4ki8:E (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135592 4ki8:F (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135593 4ki8:G (2.722) BS01 ADP 5.6.1.7 GO:0005524 ... Q548M1 23861496
    135594 4kii:A (1.85) BS01 RHL ? GO:0005515 ... P02754 N/A PDBbind: -logKd/Ki=6.23, Kd=0.59uM
    135595 4kij:A (2.8) BS01 KIJ 4.2.1.10 GO:0003855 ... P9WPX7 25234229 PDBbind: -logKd/Ki=4.30, Ki=50uM
    135596 4kin:A (1.97) BS01 1M8 2.7.11.24 GO:0000077 ... Q16539 23746475 MOAD: ic50=4.8nM
    PDBbind: -logKd/Ki=8.32, IC50=4.8nM
    BindingDB: IC50=4.8nM
    135597 4kin:B (1.97) BS01 1M8 2.7.11.24 GO:0000077 ... Q16539 23746475 MOAD: ic50=4.8nM
    BindingDB: IC50=4.8nM
    135598 4kin:C (1.97) BS01 1M8 2.7.11.24 GO:0000077 ... Q16539 23746475 MOAD: ic50=4.8nM
    BindingDB: IC50=4.8nM
    135599 4kin:D (1.97) BS01 1M8 2.7.11.24 GO:0000077 ... Q16539 23746475 MOAD: ic50=4.8nM
    BindingDB: IC50=4.8nM
    135600 4kip:A (2.27) BS01 1R9 2.7.11.24 GO:0000077 ... Q16539 23746475 MOAD: ic50=7nM
    PDBbind: -logKd/Ki=8.15, IC50=7nM
    BindingDB: IC50=7.0nM

    Reference:
  • Chengxin Zhang, Xi Zhang, Peter L Freddolino, and Yang Zhang. BioLiP2: an updated structure database for biologically relevent ligand-protein interactions, Nucleic Acids Research, gkad630 (2023)(download the PDF file).
  • Jianyi Yang, Ambrish Roy, and Yang Zhang. BioLiP: a semi-manually curated database for biologically relevant ligand-protein interactions, Nucleic Acids Research, 41: D1096-D1103 (2013) (download the PDF file).
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