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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Adenosine receptor A3
Species	Mus musculus (Mouse)
Gene	Adora3
Synonym	A3 receptor A3AR Adenosine receptor A3 ARA3 TGPCR1
Disease	N/A for non-human GPCRs
Length	319
Amino acid sequence	MEADNTTETDWLNITYITMEAAIGLCAVVGNMLVIWVVKLNPTLRTTTVYFIVSLALADIAVGVLVIPLAIAVSLQVKMHFYACLFMSCVLLIFTHASIMSLLAIAVHRYLRVKLTVRYRTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKATLASSQNSSTLLCHFRSVVSLDYMVFFSFITWILVPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFLFALCWLPLSIINFVSYFDVKIPDVAMCLGILLSHANSMMNPIVYACKIKKFKETYFLILRAVRLCQTSDSLDSNMEQTTE
UniProt	Q61618
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL1075269
IUPHAR	21
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
1200	CHEMBL178846	C22H25ClN6O5	488.929	9 / 4	1.3	Yes
4749	CHEMBL27376	C20H20ClIN6O3	554.773	7 / 4	2.0	No
9822	CHEMBL2089350	C33H28ClN5O2	562.07	6 / 3	5.6	No
29001	CHEMBL2064639	C22H21FN6O3	436.447	8 / 4	1.1	Yes
443540	CHEMBL2064645	C22H20F2N6O3	454.438	9 / 4	1.2	Yes
468737	CHEMBL3612932	C22H23ClN6O3S	486.975	8 / 4	2.5	Yes
443589	CHEMBL3407788	C22H28N6O3	424.505	7 / 4	1.9	Yes
52516	CHEMBL2402025	C29H28N6O6S	588.639	10 / 5	1.7	No
53566	CHEMBL2064655	C28H24Cl2N6O3	563.439	7 / 4	3.7	No
553504	MRS5151	C26H27ClN6O5	538.989	9 / 5	1.6	No
60680	CHEMBL2064659	C29H25ClN6O5	573.006	9 / 5	2.6	No
471403	CHEMBL3612940	C22H22ClN5O3S	471.96	7 / 4	2.3	Yes
471532	CHEMBL3612939	C21H20ClN5O3S	457.933	7 / 4	2.0	Yes
82293	CHEMBL255907	C22H25IN6O5	580.383	9 / 4	1.0	No
90123	CHEMBL2089346	C27H25N5O2	451.53	6 / 3	3.5	Yes
92067	CHEMBL175543	C20H20Cl2N6O3	463.319	7 / 4	2.0	Yes
101160	CHEMBL283057	C14H17ClN6O3	352.779	7 / 4	-0.1	Yes
445708	CHEMBL3407776	C19H20N8O3	408.422	8 / 5	-0.7	Yes
104062	CHEMBL368872	C27H27ClN6O3	519.002	7 / 4	3.3	No
446271	CHEMBL3407774	C20H20N8O3	420.433	9 / 4	-1.1	Yes
446400	CHEMBL3407783	C20H20N6O3S	424.479	8 / 4	0.7	Yes
121529	CHEMBL256520	C26H27ClN6O5	538.989	9 / 5	1.9	No
123577	CHEMBL2064656	C28H24Cl2N6O3	563.439	7 / 4	3.7	No
124379	IB-MECA	C18H19IN6O4	510.292	8 / 4	0.9	No
126967	CHEMBL425741	C20H20BrClN6O3	507.773	7 / 4	2.1	No
127342	CHEMBL2064640	C22H21ClN6O3	452.899	7 / 4	1.6	Yes
525275	CHEMBL3747670	C20H21N11O3	463.462	11 / 4	-1.3	No
130397	CHEMBL402607	C14H17ClN6O4	368.778	8 / 4	-0.1	Yes
446928	CHEMBL2064636	C21H21N7O3	419.445	8 / 4	-0.1	Yes
133229	CHEMBL2089345	C32H26ClN5O2	548.043	6 / 3	5.3	No
525382	CHEMBL3746886	C26H23Cl2N9O3S	612.49	10 / 4	3.1	No
525399	CHEMBL3798200	C20H18ClN5O3S	443.906	7 / 3	1.7	Yes
553959	ATL802	C24H22F3N7O3	513.481	9 / 1	2.9	No
137491	CHEMBL178644	C23H23ClN6O4	482.925	8 / 5	0.9	Yes
138946	2-Cl-IB-Meca	C18H18ClIN6O4	544.734	8 / 4	1.9	No
549649	CHEMBL3955519	C21H26ClN5O4	447.92	8 / 3	2.4	Yes
525655	CHEMBL3745851	C23H24ClN9O3S	542.015	10 / 4	1.9	No
539713	NECA	C12H16N6O4	308.298	8 / 4	-0.7	Yes
447756	CHEMBL3407777	C20H22N8O3	422.449	8 / 4	-0.7	Yes
448302	CHEMBL3407773	C20H20N8O3	420.433	9 / 4	-0.7	Yes
172068	CHEMBL256312	C28H33ClN8O4	581.074	9 / 6	0.7	No
550070	CHEMBL3970041	C20H24ClN5O4	433.893	8 / 3	2.0	Yes
182179	CHEMBL2064653	C28H25ClN6O3	528.997	7 / 4	3.1	No
188776	CHEMBL2089340	C21H20ClN5O2	409.874	6 / 3	2.6	Yes
196792	CHEMBL402574	C22H21ClN6O3	452.899	7 / 4	1.3	Yes
199449	MRS 5698	C28H23ClF2N6O3	564.978	9 / 4	3.3	No
221197	CHEMBL2064654	C28H24ClFN6O3	546.987	8 / 4	3.2	No
528214	CHEMBL3612944	C21H22ClN9O3S	515.977	10 / 4	1.4	No
238309	CHEMBL2402023	C27H25N5O5S	531.587	9 / 4	2.3	No
253418	CHEMBL2089335	C20H19N5O2	361.405	6 / 3	1.6	Yes
551262	CHEMBL3976121	C20H25ClN6O3	432.909	7 / 4	1.4	Yes
274618	CHEMBL175444	C20H20ClIN6O3	554.773	7 / 4	1.7	No
452720	CHEMBL3407775	C20H20N8O3	420.433	9 / 4	-1.1	Yes
497444	CHEMBL3612931	C21H21ClN6O3S	472.948	8 / 4	2.0	Yes
279243	CHEMBL2064658	C28H26ClN7O3	544.012	8 / 5	2.4	No
529471	CHEMBL3799738	C19H16ClN5O3S	429.879	7 / 3	1.3	Yes
293840	CHEMBL257405	C25H29ClN6O3Si	525.081	7 / 4	N/A	No
453336	CHEMBL3407778	C20H20N6O4	408.418	8 / 4	0.1	Yes
453817	CHEMBL3407784	C20H19ClN6O3S	458.921	8 / 4	1.7	Yes
314972	CHEMBL436649	C27H29ClN6O5	553.016	9 / 4	1.9	No
327782	CHEMBL175814	C21H23ClN6O3S	474.964	8 / 4	1.9	Yes
350086	CHEMBL411861	C22H23ClN6O3	454.915	7 / 4	1.8	Yes
351324	CHEMBL2401954	C28H25ClN6O6S	609.054	10 / 5	1.8	No
359728	CHEMBL2064661	C38H29ClN6O3	653.139	7 / 4	6.2	No
365915	CHEMBL257833	C26H27ClN6O5	538.989	9 / 5	1.6	No
375339	CHEMBL257573	C30H35ClN8O5	623.111	9 / 6	1.0	No
569367	CHEMBL3800106	C29H25N5O4	507.55	7 / 4	2.4	No
392275	CHEMBL2402024	C29H28N6O3	508.582	7 / 4	2.9	No
392917	CHEMBL258421	C25H27ClN6O3	494.98	7 / 4	2.8	Yes
532642	CHEMBL3800048	C22H21N5O3	403.442	6 / 3	1.1	Yes
395905	CHEMBL2064660	C34H29ClN6O3	605.095	7 / 4	4.7	No
417308	CHEMBL257785	C28H33ClN8O4	581.074	9 / 6	0.4	No
430313	CHEMBL2401955	C28H25ClN6O6S	609.054	10 / 5	1.8	No
431158	CHEMBL2089339	C21H21N5O2	375.432	6 / 3	1.9	Yes

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