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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Platelet-activating factor receptor
Species	Rattus norvegicus (Rat)
Gene	Ptafr
Synonym	AGEPC receptor PAF receptor PAF-R PAFr
Disease	N/A for non-human GPCRs
Length	341
Amino acid sequence	MEQNGSFRVDSEFRYTLFPIVYSVIFVLGVVANGYVLWVFATLYPSKKLNEIKIFMVNLTVADLLFLMTLPLWIVYYSNEGDWIVHKFLCNLAGCLFFINTYCSVAFLGVITYNRYQAVAYPIKTAQATTRKRGITLSLVIWISIAATASYFLATDSTNVVPKKDGSGNITRCFEHYEPYSVPILVVHIFITSCFFLVFFLIFYCNMVIIHTLLTRPVRQQRKPEVKRRALWMVCTVLAVFVICFVPHHVVQLPWTLAELGYQTNFHQAINDAHQITLCLLSTNCVLDPVIYCFLTKKFRKHLSEKFYSMRSSRKCSRATSDTCTEVMMPANQTPVLPLKN
UniProt	P46002
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4127
IUPHAR	N/A
DrugBank	N/A

Ligand

Name	CHEMBL52369
Molecular formula	C31H38O8S2
IUPAC name	(5S)-2-[3-methoxy-4-(2-phenylsulfanylethoxy)-5-propylsulfonylphenyl]-5-(3,4,5-trimethoxyphenyl)oxolane
Molecular weight	602.757
Hydrogen bond acceptor	9
Hydrogen bond donor	0
XlogP	5.8
Synonyms	N/A
Inchi Key	CUHVOXPURFBJHZ-SKCDSABHSA-N
Inchi ID	InChI=1S/C31H38O8S2/c1-6-16-41(32,33)29-20-22(19-28(36-4)31(29)38-14-15-40-23-10-8-7-9-11-23)25-13-12-24(39-25)21-17-26(34-2)30(37-5)27(18-21)35-3/h7-11,17-20,24-25H,6,12-16H2,1-5H3/t24-,25?/m0/s1
PubChem CID	44297811
ChEMBL	CHEMBL52369
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand is heavier than 500 daltons. This ligand has a partition coefficient log P greater than 5.

Experimental Data

Parameter	Value	Reference	Database source
Inhibition	84.0 %	Bioorg. Med. Chem. Lett., (1992) 2:2:181	ChEMBL
Inhibition	95.0 %	Bioorg. Med. Chem. Lett., (1992) 2:2:181	ChEMBL

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