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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Probable G-protein coupled receptor 34
Species	Mus musculus (Mouse)
Gene	Gpr34
Synonym	GPR34
Disease	N/A for non-human GPCRs
Length	375
Amino acid sequence	MTTTSVDSWLCSSHGMHFITNYSDQASQNFSGVPNVTSCPMDEKLLSTVLTTFYSVIFLVGLVGNIIALYVFLGIHRKRNSIQIYLLNVAVADLLLIFCLPFRIMYHINQNKWTLGVILCKVVGTLFYMNMYISIILLGFISLDRYIKINRSIQQRRAITTKQSIYVCCIVWTVALAGFLTMIILTLKKGGHNSTMCFHYRDRHNAKGEAIFNFVLVVMFWLIFLLIILSYIKIGKNLLRISKRRSKFPNSGKYATTARNSFIVLIIFTICFVPYHAFRFIYISSQLNVSSCYWKEIIHKTNEIMLVFSSFNSCLDPVMYFLMSSNIRKIMCQLLFRRFQSEASRSESTSEFKPGHSLHDLSVTVKMPQYSTKGN
UniProt	Q9R1K6
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL1075291
IUPHAR	101
DrugBank	N/A

Ligand

Name	CHEMBL3815090
Molecular formula	C30H44NO9P
IUPAC name	(2S)-2-amino-3-[hydroxy-[2-[3-(2-undecoxyphenyl)propanoyloxymethyl]phenoxy]phosphoryl]oxypropanoic acid
Molecular weight	593.654
Hydrogen bond acceptor	10
Hydrogen bond donor	3
XlogP	3.8
Synonyms	BDBM50177123 SCHEMBL19136019
Inchi Key	UDMRSZRXXMZWJZ-SANMLTNESA-N
Inchi ID	InChI=1S/C30H44NO9P/c1-2-3-4-5-6-7-8-9-14-21-37-27-17-12-10-15-24(27)19-20-29(32)38-22-25-16-11-13-18-28(25)40-41(35,36)39-23-26(31)30(33)34/h10-13,15-18,26H,2-9,14,19-23,31H2,1H3,(H,33,34)(H,35,36)/t26-/m0/s1
PubChem CID	127051792
ChEMBL	CHEMBL3815090
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand is heavier than 500 daltons.

Experimental Data

Parameter	Value	Reference	Database source
EC50	700.0 nM	PMID27077565	ChEMBL
EC50	707.95 nM	PMID27077565	ChEMBL
Emax	5.9 %	PMID27077565	ChEMBL
Intrinsic activity	0.2 -	PMID27077565	ChEMBL

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