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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Prostaglandin F2-alpha receptor
Species	Mus musculus (Mouse)
Gene	Ptgfr
Synonym	prostaglandin F2-alpha receptor prostaglandin F receptor (FP) prostaglandin F receptor PGF2-alpha receptor PGF2 alpha receptor PGF receptor PF2AR FP receptor Prostanoid FP receptor [ Show all ]
Disease	N/A for non-human GPCRs
Length	366
Amino acid sequence	MSMNSSKQPVSPAAGLIANTTCQTENRLSVFFSIIFMTVGILSNSLAIAILMKAYQRFRQKSKASFLLLASGLVITDFFGHLINGGIAVFVYASDKDWIRFDQSNILCSIFGISMVFSGLCPLFLGSAMAIERCIGVTNPIFHSTKITSKHVKMILSGVCMFAVFVAVLPILGHRDYQIQASRTWCFYNTEHIEDWEDRFYLLFFSFLGLLALGVSFSCNAVTGVTLLRVKFRSQQHRQGRSHHLEMIIQLLAIMCVSCVCWSPFLVTMANIAINGNNSPVTCETTLFALRMATWNQILDPWVYILLRKAVLRNLYKLASRCCGVNIISLHIWELSSIKNSLKVAAISESPAAEKESQQASSEAGL
UniProt	P43117
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL5000
IUPHAR	344
DrugBank	N/A

Ligand

Name	CHEMBL2326219
Molecular formula	C20H26N4O6S
IUPAC name	(Z)-7-[(1R,2S,3R,5S)-3,5-dihydroxy-2-[1-(4-sulfamoylphenyl)triazol-4-yl]cyclopentyl]hept-5-enoic acid
Molecular weight	450.51
Hydrogen bond acceptor	9
Hydrogen bond donor	4
XlogP	0.2
Synonyms	N/A
Inchi Key	SSXZVAUTSNINDY-DKIGCFPISA-N
Inchi ID	InChI=1S/C20H26N4O6S/c21-31(29,30)14-9-7-13(8-10-14)24-12-16(22-23-24)20-15(17(25)11-18(20)26)5-3-1-2-4-6-19(27)28/h1,3,7-10,12,15,17-18,20,25-26H,2,4-6,11H2,(H,27,28)(H2,21,29,30)/b3-1-/t15-,17-,18+,20-/m0/s1
PubChem CID	71552665
ChEMBL	CHEMBL2326219
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Experimental Data

Parameter	Value	Reference	Database source
EC50	1995.26 nM	PMID23317571	ChEMBL
Intrinsic activity	<1.0 -	PMID23317571	ChEMBL

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