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Go to the GPCR, ligand, or experimental data tables.
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GPCR

Name	Trace amine-associated receptor 1
Species	Mus musculus (Mouse)
Gene	Taar1
Synonym	TA1 receptor TaR-1 TAR1 trace amine receptor 1 TRAR1
Disease	N/A for non-human GPCRs
Length	332
Amino acid sequence	MHLCHAITNISHRNSDWSREVQASLYSLMSLIILATLVGNLIVIISISHFKQLHTPTNWLLHSMAIVDFLLGCLIMPCSMVRTVERCWYFGEILCKVHTSTDIMLSSASIFHLAFISIDRYCAVCDPLRYKAKINISTILVMILVSWSLPAVYAFGMIFLELNLKGVEELYRSQVSDLGGCSPFFSKVSGVLAFMTSFYIPGSVMLFVYYRIYFIAKGQARSINRTNVQVGLEGKSQAPQSKETKAAKTLGIMVGVFLVCWCPFFLCTVLDPFLGYVIPPSLNDALYWFGYLNSALNPMVYAFFYPWFRRALKMVLLGKIFQKDSSRSKLFL
UniProt	Q923Y8
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4908
IUPHAR	364
DrugBank	N/A

Ligand

Name	SCHEMBL3619998
Molecular formula	C10H9F3N2O
IUPAC name	4-methyl-4-(3,4,5-trifluorophenyl)-5H-1,3-oxazol-2-amine
Molecular weight	230.19
Hydrogen bond acceptor	5
Hydrogen bond donor	1
XlogP	1.4
Synonyms	US8604061, 273 CHEMBL3684860 BDBM109515
Inchi Key	BKWLTLWYHNRYMM-UHFFFAOYSA-N
Inchi ID	InChI=1S/C10H9F3N2O/c1-10(4-16-9(14)15-10)5-2-6(11)8(13)7(12)3-5/h2-3H,4H2,1H3,(H2,14,15)
PubChem CID	59323688
ChEMBL	CHEMBL3684860
IUPHAR	N/A
BindingDB	109515
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Experimental Data

Parameter	Value	Reference	Database source
Ki	9.5 nM	, None	BindingDB,ChEMBL

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