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BioLiP

Structure of PDB 8wu1 Chain R

Receptor sequence
>8wu1R (length=280) Species: 9606 (Homo sapiens) [Search protein sequence]
MVLNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGS
LAVADLLGSVIFVYSFIDFHVFHRKDSRNVFLFKLGGVTASFTASVGSLF
LTAIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCC
SDIFPHIDETYLMFWIGVTSVLLLFIVYAYMYILWKAHSHAVRMIQDIRL
AKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNST
VNPIIYALRSKDLRHAFESCTTASSSLAKD
3D structure
PDB8wu1 Cryo-EM structure of CB1-beta-arrestin1 complex
ChainR
Resolution3.2 Å
3D
structure
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Enzymatic activity
Enzyme Commision number ?
Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 KCA R F170 F174 L193 V196 T197 F200 F268 Y275 L276 W279 F379 S383 F62 F66 L85 V88 T89 F92 F154 Y161 L162 W165 F238 S242
Gene Ontology
Molecular Function
GO:0004930 G protein-coupled receptor activity
GO:0004949 cannabinoid receptor activity
Biological Process
GO:0007186 G protein-coupled receptor signaling pathway
Cellular Component
GO:0016020 membrane

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Molecular Function

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Biological Process

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Cellular Component
External links
PDB RCSB:8wu1, PDBe:8wu1, PDBj:8wu1
PDBsum8wu1
PubMed
UniProtP21554|CNR1_HUMAN Cannabinoid receptor 1 (Gene Name=CNR1);
P30518|V2R_HUMAN Vasopressin V2 receptor (Gene Name=AVPR2)

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