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Structure of PDB 1kv6 Chain B Binding Site BS01

Receptor Information
>1kv6 Chain B (length=222) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
NKIVSHLLVAEPEKIYAMPDPTVPDSDIKALTTLCDLADRELVVIIGWAK
HIPGFSTLSLADQMSLLQSAWMEILILGVVYRSLSFEDELVYADDYIMDE
DQSKLAGLLDLNNAILQLVKKYKSMKLEKEEFVTLKAIALANSDSMHIED
VEAVQKLQDVLHEALQDYEAGQHMEDPRRAGKMLMTLPLLRQTSTKAVQH
FYNIKLEGKVPMHKLFLEMLEA
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB1kv6 Structural and Functional Evidence for Ligand-Independent Transcriptional Activation by the Estrogen-Related Receptor 3
Resolution2.7 Å
Binding residue
(original residue number in PDB)
I280 K284 M298 K448 L449 E452
Binding residue
(residue number reindexed from 1)
I46 K50 M64 K214 L215 E218
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:1kv6, PDBe:1kv6, PDBj:1kv6
PDBsum1kv6
PubMed11864604
UniProtP62508|ERR3_HUMAN Estrogen-related receptor gamma (Gene Name=ESRRG)

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