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Structure of PDB 6ggg Chain A Binding Site BS01

Receptor Information
>6ggg Chain A (length=233) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
IVYAGYDKPDTAENLLSTLNRLAGKQMIQVVKWAKVLPGFKNLPLEDQIT
LIQYSWMSLLSFALSWRSYKHTNSQFLYFAPDLVFNEEKMHQSAMYELCQ
GMHQISLQFVRLQLTFEEYTIMKVLLLLSTIPKDGLKSQAAFEEMRTNYI
KELRKMVTKSPNNSGQSWQRFYQLTKLLDSMHDLVSDLLEFCFYTFRESH
ALKVEFPAMLVEIISDQLPKVESGNAKPLYFHR
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB6ggg Identification of Mineralocorticoid Receptor Modulators with Low Impact on Electrolyte Homeostasis but Maintained Organ Protection.
Resolution1.71 Å
Binding residue
(original residue number in PDB)
V781 K785 L795 I799 I802 M959 E962
Binding residue
(residue number reindexed from 1)
V31 K35 L45 I49 I52 M209 E212
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:6ggg, PDBe:6ggg, PDBj:6ggg
PDBsum6ggg
PubMed30596500
UniProtP08235|MCR_HUMAN Mineralocorticoid receptor (Gene Name=NR3C2)

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