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BioLiP

Structure of PDB 9f9m Chain C

Receptor sequence
>9f9mC (length=183) Species: 9606 (Homo sapiens) [Search protein sequence]
PLELRPGEYRVLLCVDIGETRGPELLRELQRLHVTHTVRKLHVGDFVWVA
QETNPRDPANPGELVLDHIVERKRLDDLCSSIIDGRFREQKFRLKRCGLE
RRVYLVEELSLPESTLLQAVTNTQVIDGFFVKRTADIKESAAYLALLTRG
LQRLYQGHTLRSRPWGTPNPLCSLLTFSDFNAG
3D structure
PDB9f9m Fragment-Based Discovery of Novel MUS81 Inhibitors.
ChainC
Resolution2.469 Å
3D
structure
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Interaction with ligand
Site
#
Ligand Ligand
chain
Binding residues on receptor
(original residue number in PDB)
Binding residues on receptor
(residue number reindexed from 1)
Binding affinity
BS01 MG C D307 E333 R334 D45 E71 R72
BS02 A1IA4 C D307 E333 K335 D339 R348 D45 E71 K73 D77 R86
External links
PDB RCSB:9f9m, PDBe:9f9m, PDBj:9f9m
PDBsum9f9m
PubMed39015284
UniProtQ96NY9|MUS81_HUMAN Crossover junction endonuclease MUS81 (Gene Name=MUS81)

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