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Structure of PDB 1t74 Chain A Binding Site BS01

Receptor Information
>1t74 Chain A (length=249) Species: 9598 (Pan troglodytes) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWA
KALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLV
FNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVD
GLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPI
ARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHT
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB1t74 Recognition and accommodation at the androgen receptor coactivator binding interface.
Resolution2.0 Å
Binding residue
(original residue number in PDB)
L712 V716 K720 M734 I737 Q738 E893 M894
Binding residue
(residue number reindexed from 1)
L43 V47 K51 M65 I68 Q69 E224 M225
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:1t74, PDBe:1t74, PDBj:1t74
PDBsum1t74
PubMed15328534
UniProtO97775|ANDR_PANTR Androgen receptor (Gene Name=AR)

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