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●BioLiP ●HPmod ●E. coli ●GLASS ●GPCR-HGmod ●GPCR-RD ●GPCR-EXP ●Tara-3D ●TM-fold ●DECOYS ●POTENTIAL ●RW/RWplus ●EvoEF ●HPSF ●THE-DB ●ADDRESS ●Alpaca-Antibody ●CASP7 ●CASP8 ●CASP9 ●CASP10 ●CASP11 ●CASP12 ●CASP13 ●CASP14

You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Glucagon receptor
Species	Mus musculus (Mouse)
Gene	Gcgr
Synonym	GGR GL-R glucagon receptor GR
Disease	N/A for non-human GPCRs
Length	485
Amino acid sequence	MPLTQLHCPHLLLLLLVLSCLPEAPSAQVMDFLFEKWKLYSDQCHHNLSLLPPPTELVCNRTFDKYSCWPDTPPNTTANISCPWYLPWYHKVQHRLVFKRCGPDGQWVRGPRGQPWRNASQCQLDDEEIEVQKGVAKMYSSQQVMYTVGYSLSLGALLLALVILLGLRKLHCTRNYIHGNLFASFVLKAGSVLVIDWLLKTRYSQKIGDDLSVSVWLSDGAMAGCRVATVIMQYGIIANYCWLLVEGVYLYSLLSLATFSERSFFSLYLGIGWGAPLLFVIPWVVVKCLFENVQCWTSNDNMGFWWILRIPVFLALLINFFIFVHIIHLLVAKLRAHQMHYADYKFRLARSTLTLIPLLGVHEVVFAFVTDEHAQGTLRSTKLFFDLFLSSFQGLLVAVLYCFLNKEVQAELMRRWRQWQEGKALQEERLASSHGSHMAPAGPCHGDPCEKLQLMSAGSSSGTGCVPSMETSLASSLPRLADSPT
UniProt	Q61606
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4773
IUPHAR	N/A
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
31167	CHEMBL348555	C24H22ClN3	387.911	2 / 2	6.1	No
50145	643011-22-7	C27H21ClF3N3O3S	559.988	9 / 2	6.4	No
62741	CHEMBL350255	C21H14BrClN2	409.711	1 / 1	5.9	No
64646	MK 0893	C32H27Cl2N3O4	588.485	5 / 2	6.8	No
77349	CHEMBL347663	C25H23ClN2O	402.922	2 / 1	6.5	No
95077	CHEMBL158671	C21H15FN2	314.363	2 / 1	4.7	Yes
114786	L-168,049	C24H20BrClN2O	467.791	2 / 1	6.8	No
115016	aminothiazole, 10	C30H27Cl2N3O3S	580.524	6 / 2	7.5	No
129012	glucagon receptor antagonists-4	C26H28F3N3O4	503.522	8 / 2	5.0	No
132424	CHEMBL1644183	C27H20Cl2F3N3O4	578.369	8 / 2	6.4	No
151872	CHEMBL328126	C21H14ClFN2	348.805	2 / 1	5.3	No
174425	aminothiazole, 16	C27H21ClF3N3O3S	559.988	9 / 2	6.4	No
179331	CHEMBL348401	C21H21FN2	320.411	2 / 1	5.2	No
182887	CHEMBL155686	C24H20Cl2N2O	423.337	2 / 1	6.7	No
202842	CHEMBL346698	C23H19ClN2O	374.868	2 / 1	5.6	No
210352	CHEMBL158535	C24H19ClN2O	386.879	2 / 1	5.8	No
216743	CHEMBL160561	C24H21ClN2O	388.895	2 / 1	6.0	No
232570	CHEMBL351104	C23H17ClN2O2	388.851	3 / 1	4.9	Yes
233418	CHEMBL158989	C22H14FN3	339.373	3 / 1	4.4	Yes
238453	CHEMBL345834	C27H27ClN2O	430.976	2 / 1	7.5	No
271926	CHEMBL156458	C24H21ClN2O	388.895	2 / 1	6.1	No
286050	CHEMBL157529	C21H14F2N2	332.354	3 / 1	4.8	Yes
289599	CHEMBL158676	C25H23ClN2O	402.922	2 / 1	6.4	No
308065	CHEMBL347462	C27H27ClN2O2	446.975	3 / 1	6.9	No
317401	CHEMBL160380	C22H17ClN2O	360.841	2 / 1	5.2	No
324258	aminothiazole, 6	C34H26F3N3O4S	629.654	10 / 2	7.7	No
324917	CHEMBL160638	C21H13Cl2FN2	383.247	2 / 1	5.9	No
345680	CHEMBL160735	C21H21ClN2	336.863	1 / 1	6.1	No
352494	aminothiazole, 19	C28H21F6N3O4S	609.543	13 / 2	7.0	No
372260	aminothiazole, 7	C30H26F3N3O3S	565.611	9 / 2	6.6	No
378633	CHEMBL158548	C18H17ClN2	296.798	1 / 1	4.7	Yes
389205	CHEMBL160287	C24H20BrClN2O	467.791	2 / 1	6.8	No
389545	aminothiazole, 17	C27H21ClF3N3O4S	575.987	10 / 2	6.7	No
393869	CHEMBL155694	C22H17ClN2O	360.841	2 / 1	5.2	No
398107	CHEMBL160372	C15H11ClN2	254.717	1 / 1	3.6	Yes
401176	CHEMBL160490	C21H14Cl2N2	365.257	1 / 1	5.8	No
415232	CHEMBL160281	C21H14ClFN2	348.805	2 / 1	5.3	No
421525	CHEMBL345863	C18H15ClN2O2	326.78	3 / 1	3.8	Yes
423283	aminothiazole, 8	C30H26F3N3O4S	581.61	10 / 2	6.9	No

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