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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Beta-1 adrenergic receptor
Species	Sus scrofa (Pig)
Gene	ADRB1
Synonym	Beta-1 adrenoceptor Beta-1 adrenoreceptor
Disease	N/A for non-human GPCRs
Length	468
Amino acid sequence	MGAGALALGASEPCNLSSAAPLPDGAATAARLLVPASPPASLLTPASEGSVQLSQQWTAGMGLLMALIVLLIVAGNVLVIVAIAKTPRLQTLTNLFIMSLASADLVMGLLVVPFGATIVVWGRWEYGSFFCELWTSVDVLCVTASIETLCVIALDRYLAITSPFRYQSLLTRAARALVCTVWAISALVSFLPILMHWWRDKGAEARRCYNDPKCCDFVTNRAYAIASSVVSFYVPLCIMAFVYLRVFREAQKQVKKIDSCERRFLGSPARPPSPAPSPGSPLPAAAAAAPVANGRTSKRRPSRLVALREQKALKTLGIIMGVFTLCWLPFFLANVVKAFHRDLVPDRLFVFFNWLGYANSAFNPIIYCRSPDFRKAFQRLLCCARRVARGSCAAAGDGPRASGCLAVARPPPSPGAASDDDDDEEDVGAAPPAPLLEPWAGYNGGAARDSDSSLDERTPGGRASESKV
UniProt	Q28998
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL4351
IUPHAR	N/A
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
11746	propranolol	C16H21NO2	259.349	3 / 2	3.0	Yes
23511	CHEMBL2443000	C20H30FN5O3	407.49	8 / 0	1.1	Yes
50012	CHEMBL1203618	C27H32ClNO3	454.007	4 / 3	N/A	N/A
50018	CHEMBL1203604	C22H27ClN2O3S	434.979	6 / 3	N/A	N/A
81398	CHEMBL2443010	C18H26FN5O2	363.437	7 / 0	1.3	Yes
81766	CHEMBL1203621	C27H32ClNO3	454.007	4 / 3	N/A	N/A
106708	CHEMBL2443007	C25H32FN5O3	469.561	8 / 0	3.3	Yes
178968	CHEMBL1203599	C23H29ClN2O3	416.946	4 / 4	N/A	N/A
187964	CHEMBL2443004	C22H26FN5O2	411.481	7 / 0	3.1	Yes
188238	CHEMBL348274	C27H29NO4	431.532	4 / 2	4.3	Yes
203399	CHEMBL1203620	C29H36ClNO3	482.061	4 / 3	N/A	N/A
225115	CHEMBL2443006	C26H34FN5O4	499.587	9 / 0	2.8	Yes
232875	CHEMBL1202033	C30H35NO7	521.61	8 / 3	N/A	No
242863	CHEMBL1203607	C28H34ClNO3	468.034	4 / 3	N/A	N/A
243231	CHEMBL1203605	C22H30ClNO3	391.936	4 / 3	N/A	N/A
257223	CHEMBL1203608	C26H30ClNO3	439.98	4 / 3	N/A	N/A
269381	CHEMBL1203606	C21H28ClNO3	377.909	4 / 3	N/A	N/A
280787	CHEMBL1203619	C25H28ClNO	393.955	2 / 3	N/A	N/A
313954	VERAPAMIL	C27H38N2O4	454.611	6 / 0	3.8	Yes
322273	CHEMBL1203640	C29H34ClNO4	496.044	5 / 2	N/A	N/A
322344	CHEMBL2443002	C20H28FN5O5	437.472	10 / 3	-0.1	Yes
330135	CHEMBL160317	C28H33NO3	431.576	4 / 1	5.4	No
343087	CHEMBL2443009	C20H30FN5O	375.492	6 / 0	2.8	Yes
349011	CHEMBL2443008	C29H38FN5O7	587.649	12 / 3	1.9	No
373216	CHEMBL2443003	C20H28FN5O5	437.472	10 / 3	-0.6	Yes
381731	CHEMBL2443001	C22H34FN5O4	451.543	9 / 0	1.0	Yes
390540	CHEMBL1203610	C27H32ClNO2	438.008	3 / 2	N/A	N/A
401281	CHEMBL2443005	C23H28FN5O2	425.508	7 / 0	3.5	Yes
405016	CHEMBL155739	C20H25NO3	327.424	4 / 2	3.1	Yes
417716	CHEMBL1203617	C26H28ClNO3	437.964	4 / 3	N/A	N/A

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