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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Endothelin-1 receptor
Species	Mus musculus (Mouse)
Gene	Ednra
Synonym	ETA receptor ET-AR ET-A endothelin-1 receptor Endothelin receptor type A {ECO:0000312\|MGI:MGI:105923} endothelin A receptor ENDOR Gpcr10 [ Show all ]
Disease	N/A for non-human GPCRs
Length	427
Amino acid sequence	MSIFCLAAYFWLTMVGGVMADNPERYSANLSSHMEDFTPFPGTEINFLGTTHRPPNLALPSNGSMHGYCPQQTKITTAFKYINTVISCTIFIVGMVGNATLLRIIYQNKCMRNGPNALIASLALGDLIYVVIDLPINVFKLLAGRWPFDHNDFGVFLCKLFPFLQKSSVGITVLNLCALSVDRYRAVASWSRVQGIGIPLITAIEIVSIWILSFILAIPEAIGFVMVPFEYKGELHRTCMLNATSKFMEFYQDVKDWWLFGFYFCMPLVCTAIFYTLMTCEMLNRRNGSLRIALSEHLKQRREVAKTVFCLVVIFALCWFPLHLSRILKKTVYDEMDKNRCELLSFLLLMDYIGINLATMNSCINPIALYFVSKKFKNCFQSCLCCCCHQSKSLMTSVPMNGTSIQWKNQEQNNHNTERSSHKDSMN
UniProt	Q61614
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL2286
IUPHAR	N/A
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
57818	CHEMBL347948	C43H57N7O10	831.968	10 / 8	3.3	No
80617	CHEMBL1672882	C51H61FN4O17	1021.06	21 / 1	3.2	No
94423	CHEMBL594265	C29H27BrO9	599.43	9 / 1	4.7	No
100815	CHEMBL359235	C47H59N7O10	882.028	10 / 9	4.5	No
100818	CHEMBL356864	C47H59N7O10	882.028	10 / 9	4.5	No
111864	CHEMBL147510	C43H60N8O11	864.998	12 / 11	-0.7	No
114606	CHEMBL611626	C36H34O12S	690.716	12 / 1	4.9	No
137896	CHEMBL151361	C42H56N8O11	848.955	11 / 10	1.0	No
141186	CHEMBL433893	C48H61N7O10	896.055	10 / 9	5.3	No
143624	CHEMBL149091	C41H55N7O10	805.93	10 / 9	2.6	No
169218	CHEMBL148751	C47H59N7O10	882.028	10 / 8	4.6	No
189351	CHEMBL594482	C29H27FO9	538.524	10 / 1	4.3	No
210057	CHEMBL1672881	C38H42FN3O12	751.761	15 / 1	3.1	No
219044	CHEMBL146866	C49H60N8O10	921.065	10 / 10	5.1	No
225259	CHEMBL603635	C29H27BrO9	599.43	9 / 1	4.7	No
225689	CHEMBL1672880	C35H39FO12	670.683	13 / 1	3.9	No
254584	CHEMBL147058	C47H59N7O11	898.027	11 / 10	3.8	No
255236	CHEMBL593928	C36H34O12S	690.716	12 / 1	4.9	No
266505	CHEMBL1672883	C46H51FN4O13	886.927	17 / 1	5.0	No
270496	CI 1020	C28H26O9	506.507	9 / 1	4.0	No
326324	CHEMBL1672885	C44H47FN4O14S	906.932	18 / 2	3.5	No
341479	CHEMBL604286	C29H27FO9	538.524	10 / 1	4.3	No
342767	CHEMBL1672886	C38H42FN3O12	751.761	15 / 1	3.1	No
354807	CHEMBL444274	C47H60N8O10	897.043	11 / 10	0.7	No
374269	CHEMBL1672884	C45H49FN4O14S	920.959	18 / 1	3.7	No
385025	CHEMBL423941	C43H60N8O10	848.999	11 / 10	0.5	No
385728	CHEMBL279259	C43H60N8O10	848.999	11 / 10	-0.4	No
385729	CHEMBL21253	C43H60N8O10	848.999	11 / 10	-0.4	No
385730	CHEMBL262782	C43H60N8O10	848.999	11 / 10	-0.4	No
432589	CHEMBL150719	C45H61N9O10	888.036	11 / 11	0.6	No

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