3nyx A 2.5 BS01 TZ1 A 1 F908 K930 I960 Y962 L976 M978 V981 L1030 D1041 F1042 G1043 F20 K40 I70 Y72 L85 M87 V90 L139 D150 F151 G152 N1023 A1025 R1027 N1028 D1041 P1064 N132 A134 R136 N137 D150 P173 2.7.10.2 0004672,0005524,0006468 Ki=32nM -logKd/Ki=7.49, Ki=32nM P29597 21117080 1 PTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGEMVAVKALKADCGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDQEKSLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHSQHYIHRNLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYRH