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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Lysophosphatidic acid receptor 4
Species	Mus musculus (Mouse)
Gene	Lpar4
Synonym	P2Y9 P2Y5-like receptor P2Y purinoceptor 9 P2RY9 LPA4 receptor LPA4 LPA-4 LPA receptor 4 GPR23 G-protein coupled receptor 23 G protein-coupled receptor 23 Purinergic receptor 9 [ Show all ]
Disease	N/A for non-human GPCRs
Length	370
Amino acid sequence	MGDRRFIDFQFQDLNSSLRPRLGNATANNTCIVDDSFKYNLNGAVYSVVFILGLITNSASLFVFCFRMKMRSETAIFITNLALSDLLFVCTLPFKIFYNFNRHWPFGDTLCKISGTAFLTNIYGSMLFLTCISVDRFLAIVYPFRSRTIRTRRNSAIVCAGVWILVLSGGISASLFSTTNVNNATTTCFEGFSKRVWKTYLSKITIFIEVVGFIIPLILNVSCSSVVLRTLRKPATLSQIGTNKKKVLKMITVHMAVFVVCFVPYNSVLFLYALVRSQAITNCLLERFAKIMYPITLCLATLNCCFDPFIYYFTLESFQKSFYINTHIRMESLFKTETPLTPKPSLPAIQEEVSDQTTNNGGELMLESTF
UniProt	Q8BLG2
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3321650
IUPHAR	94
DrugBank	N/A

Ligand

Name	lysophosphatidic acid
Molecular formula	C21H41O7P
IUPAC name	(2-hydroxy-3-phosphonooxypropyl) (Z)-octadec-9-enoate
Molecular weight	436.526
Hydrogen bond acceptor	7
Hydrogen bond donor	3
XlogP	5.2
Synonyms	WRGQSWVCFNIUNZ-KTKRTIGZSA-N (2-hydroxy-3-phosphonooxypropyl) (E)-octadec-9-enoate 1-Oleoyl-lyso-phosphatidate 22002-87-5 CMC_8485 Lysophosphophatidic acid [3H]LPA 1-(9Z-octadecenoyl)-phosphatidic acid 1-oleoyl-lysophosphatidic acid 9-Octadecenoic acid (Z)-, 2-hydroxy-3-(phosphonooxy)propyl ester DTXSID5041061 Olein, 1-mono-, 3-(dihydrogen phosphate) (8CI) 1-oleoyl-glycero-3-phosphate 2-hydroxy-3-(phosphonooxy)propyl (9Z)-octadec-9-enoate AKOS030561932 GTPL5395 Oleoyl lysophosphatidic acid [3H]-LPA (2-hydroxy-3-phosphonooxypropyl) (E)-octadec-9-enoic acid 1-Oleoyl-lyso-phosphatidic acid D0X0UR monooleylphosphatidate [3H]lysophosphatidic acid 1-monooleoylglycerol 3-phosphate 1-Oleyllysophosphatidate 9-octadecenoic acid, 2-hydroxy-3-(phosphonooxy)propyl ester, (9Z)- EINECS 244-710-0 Olein, 1-mono-, 3-phosphate (7CI) SCHEMBL1548 1-oleoyl-LPA 2-Hydroxy-3-(phosphonooxy)propyl oleate cis-9-Octadecenoic acid 2-hydroxy-3-phosphonooxypropyl ester [3H]1-oleoyl-LPA (2-hydroxy-3-phosphonooxypropyl) (Z)-octadec-9-enoate 1-Oleoyl-lysophosphatidate 9-Octadecenoic acid (9Z)-, 2-hydroxy-3-(phosphonooxy)propyl ester (9CI) D0Z9FO Monooleylphosphatidic acid {2-hydroxy-3-[(9Z)-octadec-9-enoyloxy]propoxy}phosphonic acid 1-Oleoyl-2-lysophosphatidic acid 1-Oleyllysophosphatidic acid AC1NUZKL GTPL2906 Oleoyl lysophosphatidate [ Show all ]
Inchi Key	WRGQSWVCFNIUNZ-KTKRTIGZSA-N
Inchi ID	InChI=1S/C21H41O7P/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16-17-21(23)27-18-20(22)19-28-29(24,25)26/h9-10,20,22H,2-8,11-19H2,1H3,(H2,24,25,26)/b10-9-
PubChem CID	5497152
ChEMBL	N/A
IUPHAR	2906
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand has a partition coefficient log P greater than 5.

Experimental Data

Parameter	Value	Reference	Database source
Kd	45.0 nM	PMID12724320	IUPHAR

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