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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Lysophosphatidic acid receptor 2
Species	Mus musculus (Mouse)
Gene	Lpar2
Synonym	Pbx4 Lysophosphatidic acid receptor Edg-4 LPA2 receptor LPA-2 LPA receptor 2 endothelial differentiation gene 4, lysophosphatidic acid G-protein-coupled receptor 4 Edg4 pre-B-cell leukemia transcription factor 4 [ Show all ]
Disease	N/A for non-human GPCRs
Length	348
Amino acid sequence	MGQCYYNETIGFFYNNSGKELSLHWRPKDVVVVALGLTVSVLVLLTNLLVIAAIASNRRFHQPIYYLLGNLAAADLFAGMAYLFLMFHTGPPHCQALHQRLVPATGPAGHQPHGVSGHTAGIAVERHRSVMAVQLHSRLPRGRVVTLIVGVWAAALGLGLLPAHFWHCLCDLDSCSRMVPLFSRSYLAAWALSSLLVFLLMVAVYTRIFFYVRRRVERMAEHVSCHPRYRETTLSLVKTVVIILGAFVVCWTPGQVVLLLDGLDCKTCNVLAVEKYFLLLAEANSLVNAVVYSCRDAEMRRTFRRLLCCMCLRWSSHKSARYSASAQTGASTRIMLPENGRPLMDSTL
UniProt	Q9JL06
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	N/A
IUPHAR	273
DrugBank	N/A

Ligand

Name	NAEPA
Molecular formula	C20H40NO5P
IUPAC name	2-[[(E)-octadec-9-enoyl]amino]ethyl dihydrogen phosphate
Molecular weight	405.516
Hydrogen bond acceptor	5
Hydrogen bond donor	3
XlogP	5.2
Synonyms	NAEPA, >=98 (TLC), solid D0R8LB N-acyl ethanolamide phosphate 2-{[(9E)-Octadec-9-enoyl]amino}ethyl dihydrogen phosphate NCGC00165839-01 API0008297 DTXSID00590850 (Z)-N-[2-(Phosphonooxy)ethyl]-9-octadecenamide 24435-25-4 ZINC17654921 CHEMBL1574292 GTPL6982 2-[[(E)-octadec-9-enoyl]amino]ethyl dihydrogen phosphate [ Show all ]
Inchi Key	BCSUWOZFWWBYSX-MDZDMXLPSA-N
Inchi ID	InChI=1S/C20H40NO5P/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-15-16-17-20(22)21-18-19-26-27(23,24)25/h9-10H,2-8,11-19H2,1H3,(H,21,22)(H2,23,24,25)/b10-9+
PubChem CID	17757220
ChEMBL	N/A
IUPHAR	6982
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand has a partition coefficient log P greater than 5.

Experimental Data

Parameter	Value	Reference	Database source
EC50	30.0 nM	PMID18781939	IUPHAR

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