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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Lysophosphatidic acid receptor 4
Species	Homo sapiens (Human)
Gene	LPAR4
Synonym	Purinergic receptor 9 P2Y9 P2Y5-like receptor P2Y purinoceptor 9 P2RY9 G-protein coupled receptor 23 G protein-coupled receptor 23 LPA4 LPA-4 LPA receptor 4 GPR23 LPA4 receptor [ Show all ]
Disease	N/A
Length	370
Amino acid sequence	MGDRRFIDFQFQDSNSSLRPRLGNATANNTCIVDDSFKYNLNGAVYSVVFILGLITNSVSLFVFCFRMKMRSETAIFITNLAVSDLLFVCTLPFKIFYNFNRHWPFGDTLCKISGTAFLTNIYGSMLFLTCISVDRFLAIVYPFRSRTIRTRRNSAIVCAGVWILVLSGGISASLFSTTNVNNATTTCFEGFSKRVWKTYLSKITIFIEVVGFIIPLILNVSCSSVVLRTLRKPATLSQIGTNKKKVLKMITVHMAVFVVCFVPYNSVLFLYALVRSQAITNCFLERFAKIMYPITLCLATLNCCFDPFIYYFTLESFQKSFYINAHIRMESLFKTETPLTTKPSLPAIQEEVSDQTTNNGGELMLESTF
UniProt	Q99677
Protein Data Bank	N/A
GPCR-HGmod model	Q99677
3D structure model	This predicted structure model is from GPCR-EXP Q99677.
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL5968
IUPHAR	94
DrugBank	N/A

Ligand

Name	Farnesyl monophosphate
Molecular formula	C15H27O4P
IUPAC name	[(2Z,6Z)-3,7,11-trimethyldodeca-2,6,10-trienyl] dihydrogen phosphate
Molecular weight	302.351
Hydrogen bond acceptor	4
Hydrogen bond donor	2
XlogP	3.7
Synonyms	15416-91-8 [(2Z,6Z)-3,7,11-trimethyldodeca-2,6,10-trienyl] dihydrogen phosphate AC1O5T7O GTPL2911 2,6,10-Dodecatrien-1-ol, 3,7,11-trimethyl-, dihydrogen phosphate, (E,E)- (2z,6z)-3,7,11-Trimethyldodeca-2,6,10-Trien-1-Yl Dihydrogen Phosphate SCHEMBL2506806 FFT [ Show all ]
Inchi Key	ALEWCKXBHSDCCT-FBXUGWQNSA-N
Inchi ID	InChI=1S/C15H27O4P/c1-13(2)7-5-8-14(3)9-6-10-15(4)11-12-19-20(16,17)18/h7,9,11H,5-6,8,10,12H2,1-4H3,(H2,16,17,18)/b14-9-,15-11-
PubChem CID	6440220
ChEMBL	N/A
IUPHAR	2911
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Experimental Data

Parameter	Value	Reference	Database source
IC50	1445.44 nM	PMID19366702	IUPHAR

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