1vcu A 2.85 BS01 DAN A 1 R21 D46 M85 E111 Y179 Y181 L217 R237 R304 Y334 R21 D46 M85 E111 Y179 Y181 L217 R234 R297 Y327 D46 E218 D46 E218 3.2.1.18 0004308,0005515,0005737,0005764,0005829,0006516,0006689,0009313,0016020,0016042,0016798,0046479,0052794,0052795,0052796,1902494 -logKd/Ki=3.85, Ki=0.14mM Ki=25000nM, IC50=37000nM Q9Y3R4 15501818 381 MASLPVLQKESVFQSGAHAYRIPALLYLPGQQSLLAFAEQRASKKDEHAELIVLRRGDYDAPTHQVQWQAQEVVAQARLDGHRSMNPCPLYDAQTGTLFLFFIAIPGQVTEQQQLQTRANVTRLCQVTSTDHGRTWSSPRDLTDAAIGPAYREWSTFAVGPGHCLQLNDRARSLVVPAYAYRKLHPIQRPIPSAFCFLSHDHGRTWARGHFVAQDTLECQVAEVEQRVVTLNARSHLRARVQAQSTNDGLDFQESQLVKKLVEPPPQGCQGSVISFPSPRSPAQWLLYTHPTHSWQRADLGAYLNPRPPAPEAWSEPVLLAKGSCAYSDLQSMGTGPDGSPLFGCLYEANDYEEIVFLMFTLKQAFPAEY 1vcu B 2.85 BS01 DAN B 1 R21 D46 M85 E111 Y181 L217 R237 R304 Y334 R21 D46 M85 E111 Y181 L217 R237 R300 Y330 D46 E218 D46 E218 3.2.1.18 0004308,0005515,0005737,0005764,0005829,0006516,0006689,0009313,0016020,0016042,0016798,0046479,0052794,0052795,0052796,1902494 Ki=25000nM, IC50=37000nM Q9Y3R4 15501818 381 MASLPVLQKESVFQSGAHAYRIPALLYLPGQQSLLAFAEQRASKKDEHAELIVLRRGDYDAPTHQVQWQAQEVVAQARLDGHRSMNPCPLYDAQTGTLFLFFIAIPGQVTEQQQLQTRANVTRLCQVTSTDHGRTWSSPRDLTDAAIGPAYREWSTFAVGPGHCLQLNDRARSLVVPAYAYRKLHPIQRPIPSAFCFLSHDHGRTWARGHFVAQDTLECQVAEVETGEQRVVTLNARSHLRARVQAQSTNDGLDFQESQLVKKLVEPPPQGCQGSVISFPSPRSPAQWLLYTHPTHSWQRADLGAYLNPRPPAPEAWSEPVLLAKGSCAYSDLQSMGTGPDGSPLFGCLYEANDYEEIVFLMFTLKQAFPAEY