1eb3 A 1.75 BS01 DSB A 1 S179 K210 Y216 F219 R220 K263 Y287 V289 S290 Y329 S179 K210 Y216 F219 R220 K263 Y287 V289 S290 Y329 K210 K263 K210 K263 4.2.1.24 0004655,0005634,0005737,0005829,0006782,0006783,0008270,0016829,0033014,0046872 P05373 11513881 1341 MHTAEFLETEPTEISSVLAGGYNHPLLRQWQSERQLTKNMLIFPLFISDNPDDFTEIDSLPNINRIGVNRLKDYLKPLVAKGLRSVILFGVPLIPGTKDPVGTAADDPAGPVIQGIKFIREYFPELYIICDVCLCEYTSHGHCGVLYDDGTINRERSVSRLAAVAVNYAKAGAHCVAPSDMIDGRIRDIKRGLINANLAHKTFVLSYAAKFSGNLYGPFRDAACSAPSNGDRKCYQLPPAGRGLARRALERDMSEGADGIIVKPSTFYLDIMRDASEICKDLPICAYHVSGEYAMLHAAAEKGVVDLKTIAFESHQGFLRAGARLIITYLAPEFLDWLDE 1i8j A 1.9 BS02 DSB A 1 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 -logKd/Ki=4.41, IC50=39uM P0ACB2 11444968 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1i8j B 1.9 BS02 DSB B 1 S164 Y191 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 S164 Y191 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 P0ACB2 11444968 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1l6s A 1.7 BS02 DSB A 1 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 -logKd/Ki=4.41, IC50=39uM P0ACB2 11909869 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 1l6s B 1.7 BS02 DSB B 1 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 Y200 F203 R204 R215 Q219 K246 Y269 V271 S272 Y311 K194 K246 K194 K246 4.2.1.24 0000287,0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 P0ACB2 11909869 350 TDLIQRPRRLRKSPALRAMFEETTLSLNDLVLPIFVEEEIDDYKAVEAMPGVMRIPEKHLAREIERIANAGIRSVMTFGISHHTDETGSDAWREDGLVARMSRICKQTVPEMIVMSDTCFCEYTSHGHCGVLCEHGVDNDATLENLGKQAVVAAAAGADFIAPSAAMDGQVQAIRQALDAAGFKDTAIMSYSTKFASSFYGPFREAAGSALKGDRKSYQMNPMNRREAIRESLLDEAQGADCLMVKPAGAYLDIVRELRERTELPIGAYQVSGEYAMIKFAALAGAIDEEKVVLESLGSIKRAGADLIFSYFALDLAEKKILR 2c1h A 2.6 BS01 DSB A 1 S170 K200 Y206 F209 R210 K222 K253 Y276 V278 S279 Y318 S161 K191 Y197 F200 R201 K213 K244 Y267 V269 S270 Y309 K200 K253 K191 K244 4.2.1.24 0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 Q59334 16304458 1330 VHRPRRLRRTAALRNLVQENTLTVNDLVFPLFVMPGTNAVEEVSSMPGSFRFTIDRAVEECKELYDLGIQGIDLFGIPEQKTEDGSEAYNDNGILQQAIRAIKKAVPELCIMTDVALDPFTPFGHDGLVKDGIILNDETVEVLQKMAVSHAEAGADFVSPSDMMDGRIGAIREALDETDHSDVGILSYAAKYASSFYGPFRDALHSAPQFGDKSTYQMNPANTEEAMKEVELDIVEGADIVMVKPGLAYLDIVWRTKERFDVPVAIYHVSGEYAMVKAAAAKGWIDEDRVMMESLLCMKRAGADIIFTYYAKEAAKKLR 2c1h B 2.6 BS02 DSB B 1 S170 K200 Y206 F209 R210 K222 K253 Y276 V278 S279 Y318 S161 K191 Y197 F200 R201 K213 K244 Y267 V269 S270 Y309 K200 K253 K191 K244 4.2.1.24 0004655,0005829,0006782,0006783,0008270,0016829,0033014,0046872 Q59334 16304458 1330 VHRPRRLRRTAALRNLVQENTLTVNDLVFPLFVMPGTNAVEEVSSMPGSFRFTIDRAVEECKELYDLGIQGIDLFGIPEQKTEDGSEAYNDNGILQQAIRAIKKAVPELCIMTDVALDPFTPFGHDGLVKDGIILNDETVEVLQKMAVSHAEAGADFVSPSDMMDGRIGAIREALDETDHSDVGILSYAAKYASSFYGPFRDALHSAPQFGDKSTYQMNPANTEEAMKEVELDIVEGADIVMVKPGLAYLDIVWRTKERFDVPVAIYHVSGEYAMVKAAAAKGWIDEDRVMMESLLCMKRAGADIIFTYYAKEAAKKLR