3k23 A 3.0 BS01 peptide D 0 V575 K579 M593 Q597 E751 M752 E755 V50 K54 M68 Q72 E220 M221 E224 ? P04150 19822747 743 ~ 751 LPQLTPTLVSLLEVIEPEVLYAGYDSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 A 3.0 BS02 peptide E 0 Y648 E652 K720 Y118 E122 K190 ? P04150 19822747 742 ~ 751 LPQLTPTLVSLLEVIEPEVLYAGYDSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 A 3.0 BS03 JZN A 1 P541 M560 L563 N564 L566 Q570 M601 L603 M604 A605 A607 L608 F623 C736 P17 M35 L38 N39 L41 Q45 M76 L78 M79 A80 A82 L83 F98 C206 ? -logKd/Ki=8.20, IC50=6.3nM IC50=6.3nM P04150 19822747 1 LPQLTPTLVSLLEVIEPEVLYAGYDSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 B 3.0 BS01 peptide E 0 V575 K579 M593 E751 M752 V49 K53 M67 E222 M223 ? P04150 19822747 742 ~ 751 QLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKRESQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 B 3.0 BS02 JZN B 1 P541 M560 L563 N564 L566 Q570 M604 A607 R611 F623 Q642 M646 L732 Y735 P15 M34 L37 N38 L40 Q44 M78 A81 R85 F97 Q116 M120 L203 Y206 ? IC50=6.3nM P04150 19822747 2 QLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVKRESQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQ 3k23 C 3.0 BS01 peptide F 0 K579 M593 Q597 E751 M752 E755 N759 K55 M69 Q73 E225 M226 E229 N233 ? P04150 19822747 741 ~ 750 LPQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMIEFPEMLAEIITNQIPKYNIKKLLFH 3k23 C 3.0 BS02 JZN C 1 M560 L563 N564 L566 Q570 M604 A605 A607 L608 R611 F623 M646 L732 M36 L39 N40 L42 Q46 M80 A81 A83 L84 R87 F99 M122 L207 ? IC50=6.3nM P04150 19822747 3 LPQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMIEFPEMLAEIITNQIPKYNIKKLLFH