3hfb A 1.92 BS01 FE A 1 H272 H277 E317 H153 H158 E198 H272 H277 E317 S336 H153 H158 E198 S217 1.14.16.4 0004497,0005506,0009072,0016714 P17752 20556201 400 SVPWFPKKISDLDHCANRDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFRELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI 3hfb A 1.92 BS02 ML4 A 1 P238 R257 Y264 T265 P266 H272 Q306 A309 F313 E317 S336 S337 C364 P119 R138 Y145 T146 P147 H153 Q187 A190 F194 E198 S217 S218 C245 H272 H277 E317 S336 H153 H158 E198 S217 1.14.16.4 0004497,0005506,0009072,0016714 Ki=0.03uM -logKd/Ki=7.52, Ki=0.03uM IC50=40nM P17752 20556201 401 SVPWFPKKISDLDHCANRDNVYRKRRKYFADLAMNYKHGDPIPKVEFTEEEIKTWGTVFRELNKLYPTHACREYLKNLPLLSKYCGYREDNIPQLEDVSNFLKERTGFSIRPVAGYLSPRDFLSGLAFRVFHCTQYVRHSSDPFYTPEPDTCHELLGHVPLLAEPSFAQFSQEIGLASLGASEEAVQKLATCYFFTVEFGLCKQDGQLRVFGAGLLSSISELKHALSGHAKVKPFDPKITCKQECLITTFQDVYFVSESFEDAKEKMREFTKTI