2qrk A 1.75 BS01 AMP A 1 L202 G203 R204 C205 D227 I228 T231 I250 L200 G201 R202 C203 D225 I226 T229 I248 1.5.1.7 0003729,0004753,0004754,0005515,0005737,0005777,0006553,0009085,0016491,0016558,0019878 Ki=55uM -logKd/Ki=4.26, Ki=55uM P38998 17939687 500 AVTLHLRAETKPLEARAALTPTTVKKLIAKGFKIYVEDSPQSTFNINEYRQAGAIIVPAGSWKTAPRDRIIIGLKEMPETDTFPLVHEHIQFAHCYKDQAGWQNVLMRFIKGHGTLYDLEFLENDQGRRVAAFGFYAGFAGAALGVRDWAFKQTHSDDEDLPAVSPYPNEKALVKDVTKDYKEALATGARKPTVLIIGALGRCGSGAIDLLHKVGIPDANILKWDIKETSRGGPFDEIPQADIFINCIYLSKPIAPFTNMEKLNNPNRRLRTVVDVSADTTNPHNPIPIYTVATVFNKPTVLVPTTAGPKLSVISIDHLPSLLPREASEFFSHDLLPSLELLPQRKTAPVWVRAKKLFDRHCARV