7jv5 R 3.0 BS01 SK0 R 1 D103 S107 S188 L190 S198 F288 N292 D83 S87 S152 L154 S162 F230 N234 ? 0001588,0001659,0001661,0001662,0001764,0001963,0001965,0001975,0004930,0004952,0005515,0005634,0005783,0005789,0005886,0005929,0006606,0006936,0007186,0007187,0007189,0007190,0007191,0007212,0007416,0007612,0007613,0007617,0007625,0007626,0007628,0007631,0008306,0008542,0009410,0012505,0014002,0015872,0016020,0016477,0019226,0019228,0021542,0021756,0021766,0021853,0030335,0030425,0030432,0032795,0035106,0035240,0035249,0042053,0042220,0042311,0042417,0042711,0042734,0042995,0043197,0043268,0043410,0045202,0045211,0046323,0046959,0046960,0048148,0051281,0051584,0051968,0060134,0060158,0060170,0060291,0060292,0071870,0071880,0097648,0097730,0098978,0098982,0099010,0099171,1990763,2001224 EC50=4.7nM, Ki=7nM P21728 33571431 501 SVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCY 7jv5 R 3.0 BS02 CLR R 1 R192 T193 I201 R156 T157 I165 ? 0001588,0001659,0001661,0001662,0001764,0001963,0001965,0001975,0004930,0004952,0005515,0005634,0005783,0005789,0005886,0005929,0006606,0006936,0007186,0007187,0007189,0007190,0007191,0007212,0007416,0007612,0007613,0007617,0007625,0007626,0007628,0007631,0008306,0008542,0009410,0012505,0014002,0015872,0016020,0016477,0019226,0019228,0021542,0021756,0021766,0021853,0030335,0030425,0030432,0032795,0035106,0035240,0035249,0042053,0042220,0042311,0042417,0042711,0042734,0042995,0043197,0043268,0043410,0045202,0045211,0046323,0046959,0046960,0048148,0051281,0051584,0051968,0060134,0060158,0060170,0060291,0060292,0071870,0071880,0097648,0097730,0098978,0098982,0099010,0099171,1990763,2001224 P21728 33571431 502 SVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCY 7jv5 R 3.0 BS03 CLR R 2 T268 L271 G279 T210 L213 G221 ? 0001588,0001659,0001661,0001662,0001764,0001963,0001965,0001975,0004930,0004952,0005515,0005634,0005783,0005789,0005886,0005929,0006606,0006936,0007186,0007187,0007189,0007190,0007191,0007212,0007416,0007612,0007613,0007617,0007625,0007626,0007628,0007631,0008306,0008542,0009410,0012505,0014002,0015872,0016020,0016477,0019226,0019228,0021542,0021756,0021766,0021853,0030335,0030425,0030432,0032795,0035106,0035240,0035249,0042053,0042220,0042311,0042417,0042711,0042734,0042995,0043197,0043268,0043410,0045202,0045211,0046323,0046959,0046960,0048148,0051281,0051584,0051968,0060134,0060158,0060170,0060291,0060292,0071870,0071880,0097648,0097730,0098978,0098982,0099010,0099171,1990763,2001224 P21728 33571431 504 SVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCY 7jv5 R 3.0 BS04 CLR R 3 F156 Q160 F136 Q140 ? 0001588,0001659,0001661,0001662,0001764,0001963,0001965,0001975,0004930,0004952,0005515,0005634,0005783,0005789,0005886,0005929,0006606,0006936,0007186,0007187,0007189,0007190,0007191,0007212,0007416,0007612,0007613,0007617,0007625,0007626,0007628,0007631,0008306,0008542,0009410,0012505,0014002,0015872,0016020,0016477,0019226,0019228,0021542,0021756,0021766,0021853,0030335,0030425,0030432,0032795,0035106,0035240,0035249,0042053,0042220,0042311,0042417,0042711,0042734,0042995,0043197,0043268,0043410,0045202,0045211,0046323,0046959,0046960,0048148,0051281,0051584,0051968,0060134,0060158,0060170,0060291,0060292,0071870,0071880,0097648,0097730,0098978,0098982,0099010,0099171,1990763,2001224 P21728 33571431 505 SVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCY 7jv5 R 3.0 BS05 CLR R 4 I142 V146 I122 V126 ? 0001588,0001659,0001661,0001662,0001764,0001963,0001965,0001975,0004930,0004952,0005515,0005634,0005783,0005789,0005886,0005929,0006606,0006936,0007186,0007187,0007189,0007190,0007191,0007212,0007416,0007612,0007613,0007617,0007625,0007626,0007628,0007631,0008306,0008542,0009410,0012505,0014002,0015872,0016020,0016477,0019226,0019228,0021542,0021756,0021766,0021853,0030335,0030425,0030432,0032795,0035106,0035240,0035249,0042053,0042220,0042311,0042417,0042711,0042734,0042995,0043197,0043268,0043410,0045202,0045211,0046323,0046959,0046960,0048148,0051281,0051584,0051968,0060134,0060158,0060170,0060291,0060292,0071870,0071880,0097648,0097730,0098978,0098982,0099010,0099171,1990763,2001224 P21728 33571431 507 SVRILTACFLSLLILSTLLGNTLVCAAVIRFRHLRSKVTNFFVISLAVSDLLVAVLVMPWKAVAEIAGFWPFGSFCNIWVAFDIMCSTASILNLCVISVDRYWAISSPFRYERKMTPKAAFILISVAWTLSVLISFIPVQLSWHKAKPNCDSSLSRTYAISSSVISFYIPVAIMIVTYTRIYRIAQKQIRRIAALERAAVHAKNSFKRETKVLKTLSVIMGVFVCCWLPFFILNCILPFCCIDSNTFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCY