7bwd A 4.32 BS01 dna I 0 R40 Y41 P43 G44 V46 R49 R63 R4 Y5 P7 G8 V10 R13 R27 ? 0000786,0003677,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0010467,0016020,0030527,0032200,0032991,0040029,0045296,0046982,0070062 P68431 2 ~ 147 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEACEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 7bwd A 4.32 BS02 dna J 0 H39 Y41 R42 R72 R83 Q85 S86 V117 T118 H3 Y5 R6 R36 R47 Q49 S50 V81 T82 ? 0000786,0003677,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0010467,0016020,0030527,0032200,0032991,0040029,0045296,0046982,0070062 P68431 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEACEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGERA 7bwd B 4.32 BS01 dna I 0 R35 I46 G48 R78 K79 R17 I28 G30 R60 K61 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 P62805 2 ~ 147 RKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 7bwd B 4.32 BS02 dna J 0 T30 R36 T12 R18 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 P62805 1 ~ 146 RKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 7bwd C 4.32 BS01 dna I 0 K13 R29 R42 V43 K75 T76 R77 K3 R19 R32 V33 K65 T66 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031492,0031507,0043505,0046982,0061644,0070062 P04908 2 ~ 147 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLPKKTES 7bwd C 4.32 BS02 dna J 0 R11 K15 T16 R17 R20 R32 R77 R1 K5 T6 R7 R10 R22 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031492,0031507,0043505,0046982,0061644,0070062 P04908 1 ~ 146 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLPKKTES 7bwd D 4.32 BS01 dna I 0 R31 Y40 R1 Y10 ? 0000786,0002227,0003674,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0019731,0030527,0031640,0042742,0046982,0050829,0050830,0061844 O60814 2 ~ 147 RSRKESYSVYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 7bwd D 4.32 BS02 dna J 0 R33 S55 S56 R86 S87 T88 R3 S25 S26 R56 S57 T58 ? 0000786,0002227,0003674,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0019731,0030527,0031640,0042742,0046982,0050829,0050830,0061844 O60814 1 ~ 146 RSRKESYSVYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 7bwd E 4.32 BS01 dna I 0 R42 R63 R72 R83 Q85 T118 R6 R27 R36 R47 Q49 T82 ? 0000786,0003677,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0010467,0016020,0030527,0032200,0032991,0040029,0045296,0046982,0070062 P68431 2 ~ 147 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEACEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGE 7bwd E 4.32 BS02 dna J 0 R40 Y41 V46 R49 R63 L65 R69 R83 R4 Y5 V10 R13 R27 L29 R33 R47 ? 0000786,0003677,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0010467,0016020,0030527,0032200,0032991,0040029,0045296,0046982,0070062 P68431 1 ~ 146 KPHRYRPGTVALREIRRYQKSTELLIRKLPFQRLVREIAQDFKTDLRFQSSAVMALQEACEAYLVGLFEDTNLCAIHAKRVTIMPKDIQLARRIRGE 7bwd F 4.32 BS01 dna J 0 R45 I46 S47 G48 R78 R30 I31 S32 G33 R63 ? 0000781,0000786,0003677,0003723,0005515,0005576,0005634,0005654,0005694,0006325,0006334,0016020,0030527,0032200,0032991,0043505,0045653,0046982,0061644,0070062 P62805 1 ~ 146 KRHRKVLRDNIQGITKPAIRRLARRGGVKRISGLIYEETRGVLKVFLENVIRDAVTYTEHAKRKTVTAMDVVYALKRQGRTLYGFGG 7bwd G 4.32 BS01 dna I 0 R11 K15 R77 R1 K5 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031492,0031507,0043505,0046982,0061644,0070062 P04908 2 ~ 147 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLPKK 7bwd G 4.32 BS02 dna J 0 R11 R42 V43 A45 K75 T76 R77 R1 R32 V33 A35 K65 T66 R67 ? 0000786,0003677,0005515,0005634,0005694,0006325,0008285,0030527,0031492,0031507,0043505,0046982,0061644,0070062 P04908 1 ~ 146 RAKAKTRSSRAGLQFPVGRVHRLLRKGNYSERVGAGAPVYLAAVLEYLTAEILELAGNAARDNKKTRIIPRHLQLAIRNDEELNKLLGRVTIAQGGVLPNIQAVLLPKK 7bwd H 4.32 BS01 dna I 0 R33 S56 R86 S87 T88 R3 S26 R56 S57 T58 ? 0000786,0002227,0003674,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0019731,0030527,0031640,0042742,0046982,0050829,0050830,0061844 O60814 2 ~ 147 RSRKESYSVYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 7bwd H 4.32 BS02 dna J 0 E35 Y40 E5 Y10 ? 0000786,0002227,0003674,0003677,0005515,0005615,0005634,0005654,0005694,0005829,0019731,0030527,0031640,0042742,0046982,0050829,0050830,0061844 O60814 1 ~ 146 RSRKESYSVYVYKVLKQVHPDTGISSKAMGIMNSFVNDIFERIAGEASRLAHYNKRSTITSREIQTAVRLLLPGELAKHAVSEGTKAVTKYTSA 7bwd K 4.32 BS01 SAH K 1 P133 E134 V135 Y136 T139 G163 S164 Q168 V169 E186 F223 F239 N241 F245 P129 E130 V131 Y132 T135 G159 S160 Q164 V165 E182 F219 F235 N237 F241 2.1.1.360 0031151,0051726 Ki=160nM, IC50=600nM, Kd=150nM Q8TEK3 501 LELRLKSPVGAEPAVYPWPLPVYDKHHDAAHEIIETIRWVCEEIPDLKLAMENYVLIDYDTKSFESMQRLCDKYNRAIDSIHQLWKGTTQPMKLNTRPSTGLLRHILQQVYNHSVTDPEKLNNYEPFSPEVYGETSFDLVAQMIDEIKMTDDDLFVDLGSGVGQVVLQVAAATNCKHHYGVEKADIPAKYAETMDREFRKWMKWYGKKHAEYTLERGDFLSEEWRERIANTSVIFVNNFAFGPEVDHQLKERFANMKEGGRIVSSKPFAPLNFRINSRNLSDIGTIMRVVELSPLKGSVSWTGKPVSYYLHTIDRTILENYFSSLKNP 7bwd L 4.32 BS01 dna J 0 R42 L71 R72 R74 R42 L71 R72 R74 ? P62979 1 ~ 146 MQIFVKTLTGKTITLEVEPSDTIENVKAKIQDKEGIPPDQQRLIFAGKQLEDGRTLSDYNIQKESTLHLVLRLRGC