6vzl A 2.07 BS01 EDK A 1 F282 C285 Q286 R288 S289 H323 Y327 L330 I341 S342 F363 M364 H449 Y473 F61 C64 Q65 R67 S68 H102 Y106 L109 I120 S121 F142 M143 H228 Y252 ? 0003677,0004879,0005634,0006355 EC50=130nM, Ki=0.049700nM P37231 33713599 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGTDKSPFVIYDMNSLMMGEDKIEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYK 6vzl B 2.07 BS01 EDK B 1 R280 G284 C285 F287 R288 S289 L330 I341 S342 E343 R56 G60 C61 F63 R64 S65 L106 I117 S118 E119 ? 0003677,0004879,0005634,0006355 EC50=130nM, Ki=0.049700nM P37231 33713599 501 ESADLRALAKHLYDSYIKSFPLTKAKARAILTKSPFVIYDMNSLMMGEDKIEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETHPLLQEIYKDL