6vnk A 2.0 BS01 RXT A 1 L855 G856 G858 A880 M929 E930 L932 R980 N981 L983 L21 G22 G24 A46 M94 E95 L97 R145 N146 L148 D976 R980 N981 D994 D141 R145 N146 D159 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.8nM, EC50=12nM, Kd=0.036000nM, Ki=0.100000nM O60674 33570945 1201 LYFQGDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 6vnk B 2.0 BS01 RXT B 1 L855 A880 M929 E930 L932 R980 N981 L983 G993 L21 A46 M94 E95 L97 R145 N146 L148 G158 D976 R980 N981 D994 D141 R145 N146 D159 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.8nM, EC50=12nM, Kd=0.036000nM, Ki=0.100000nM O60674 33570945 1201 LYFQGDPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMAG 6vnk C 2.0 BS01 RXT C 1 L855 G856 A880 M929 E930 L932 R980 N981 L983 G993 D994 L13 G14 A38 M87 E88 L90 R138 N139 L141 G151 D152 D976 R980 N981 D994 D134 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.8nM, EC50=12nM, Kd=0.036000nM, Ki=0.100000nM O60674 33570945 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA 6vnk D 2.0 BS01 RXT D 1 L855 G856 G858 V863 A880 M929 E930 L932 R980 N981 L983 G993 D994 L13 G14 G16 V21 A38 M87 E88 L90 R138 N139 L141 G151 D152 D976 R980 N981 D994 D134 R138 N139 D152 2.7.10.2 0004672,0004713,0005524,0006468 IC50=2.8nM, EC50=12nM, Kd=0.036000nM, Ki=0.100000nM O60674 33570945 1201 QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSAGRRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNMA