6vkk A 2.1 BS01 RPB A 1 E763 H862 G863 G888 Y889 Y896 F897 A898 S904 Y907 E102 H196 G197 G222 Y223 Y230 F231 A232 S238 Y241 S904 Y907 E988 S238 Y241 E322 2.4.2.-,2.4.2.30 0003950 Ki=1.4nM, IC50=3.2nM, EC50=4.7nM P09874 32241924 1101 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 6vkk B 2.1 BS01 RPB B 1 Q759 E763 H862 G863 Y889 Y896 F897 A898 K903 S904 Y907 E988 Q98 E102 H196 G197 Y223 Y230 F231 A232 K237 S238 Y241 E322 S904 Y907 E988 S238 Y241 E322 2.4.2.-,2.4.2.30 0003950 Ki=1.4nM, IC50=3.2nM, EC50=4.7nM P09874 32241924 1202 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDFGMKKPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 6vkk C 2.1 BS01 RPB C 1 Q759 E763 H862 G863 G888 Y889 Y896 F897 A898 S904 Y907 E988 Q93 E97 H191 G192 G217 Y218 Y225 F226 A227 S233 Y236 E317 S904 Y907 E988 S233 Y236 E317 2.4.2.-,2.4.2.30 0003950 Ki=1.4nM, IC50=3.2nM, EC50=4.7nM P09874 32241924 1101 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHDPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT 6vkk D 2.1 BS01 RPB D 1 E763 H862 G863 G888 Y889 Y896 F897 A898 S904 Y907 E988 E96 H190 G191 G216 Y217 Y224 F225 A226 S232 Y235 E316 S904 Y907 E988 S232 Y235 E316 2.4.2.-,2.4.2.30 0003950 Ki=1.4nM, IC50=3.2nM, EC50=4.7nM P09874 32241924 1101 KSKLPKPVQDLIKMIFDVESMKKAMVEYEIDLQKMPLGKLSKRQIQAAYSILSEVQQAVSQGSSDSQILDLSNRFYTLIPHPPLLNNADSVQAKAEMLDNLLDIEVAYSLLRGSKDPIDVNYEKLKTDIKVVDRDSEEAEIIRKYVKNTHATTHNAYDLEVIDIFKIEREGECQRYKPFKQLHNRRLLWHGSRTTNFAGILSQGLRIAPPEAPVTGYMFGKGIYFADMVSKSANYCHTSQGDPIGLILLGEVALGNMYELKHASHISKLPKGKHSVKGLGKTTPDPSANISLDGVDVPLGTGISSGVNDTSLLYNEYIVYDIAQVNLKYLLKLKFNFKT