6ur8 A 3.71 BS01 QMR A 1 W156 T157 Y197 C199 Y204 W152 T153 Y193 C195 Y200 ? 0004888,0005216,0005230,0005506,0006811,0009055,0016020,0020037,0022848,0022900,0034220,0042597,0045211,0046872 P0ABE7,P43681 32221310 702 ETRAHAEERLLKKLFSGYNKWSRPVANISDVVLVRFGLSIAQLIDVDEKNQMMTTNVWVKQEWHDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAVTHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVNMHSRVDQLDFWESGEWVIVDAVGTYNTRKYECCAEIYPDITYAFVIRRLPLFYTINLIIPCLLISCLTVLVFYLPSECGEKITLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMIFVTLSIVITVFVLNVHHRSPRTHTMPTWVRRVFLDIVPRLLLMEDWKYVAMVIDRIFLWMFIIVCLLGTVGLFLPPW 6ur8 B 3.71 BS01 QMR A 1 F119 L121 F118 L120 ? 0004888,0005216,0005230,0006811,0016020,0022848,0034220,0045211 Ki=0.480nM P17787 32221310 702 DTEERLVEHLLDPSRYNKLIRPATNGSELVTVQLMVSLAQLISVHEREQIMTTNVWLTQEWEDYRLTWKPEEFDNMKKVRLPSKHIWLPDVVLYNNADGMYEVSFYSNAVVSYDGSIFWLPPAIYKSACKIEVKHFPFDQQNCTMKFRSWTYDRTEIDLVLKSEVASLDDFTPSGEWDIVALPGRRNENPDDSTYVDITYDFIIRRKPLFYTINLIIPCVLITSLAILVFYLPSDCGEKMTLCISVLLALTVFLLLISKIVPPTSLDVPLVGKYLMFTMVLVTFSIVTSVCVLNVHHRSPTTHTMAPWVKVVFLEKLPALLFMQQSVSEDWKYVAMVIDRLFLWIFVFVCVFGTIGMF 6ur8 D 3.71 BS01 QMR D 1 W156 T157 C199 Y204 W152 T153 C195 Y200 ? 0004888,0005216,0005230,0005506,0006811,0009055,0016020,0020037,0022848,0022900,0034220,0042597,0045211,0046872 P0ABE7,P43681 32221310 702 ETRAHAEERLLKKLFSGYNKWSRPVANISDVVLVRFGLSIAQLIDVDEKNQMMTTNVWVKQEWHDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAVTHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVNMHSRVDQLDFWESGEWVIVDAVGTYNTRKYECCAEIYPDITYAFVIRRLPLFYTINLIIPCLLISCLTVLVFYLPSECGEKITLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMIFVTLSIVITVFVLNVHHRSPRTHTMPTWVRRVFLDIVPRLLLMEDWKYVAMVIDRIFLWMFIIVCLLGTVGLFLPPW