6uip A 3.7 BS01 Q8J A 1 I165 F170 A186 K188 L241 N292 L294 V306 I35 F40 A56 K58 L111 N162 L164 V176 D287 K289 N292 D307 S324 D157 K159 N162 D177 S194 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 IC50=6.2nM Q13627 32077280 501 KERKVYNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPKRSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSFF 6uip B 3.7 BS01 Q8J B 1 I165 K188 L241 Y243 N292 L294 V306 I30 K53 L106 Y108 N157 L159 V169 D287 K289 N292 D307 S324 D152 K154 N157 D170 S187 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 IC50=6.2nM Q13627 32077280 501 YNDGYDDDNYDYIVKNGEKWMDRYEIDSLIGKGSFGQVVKAYDRVEQEWVAIKIIKNKKAFLNQAQIEVRLLELMNKHDTEMKYYIVHLKRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPELSIIHCDLKPENILLCNPSAIKIVDFGSSCQLGQRIYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTKREYKPPGTRKLHNILGVETGGPGGRRAGESGHTVADYLKFKDLILRMLDYDPKTRIQPYYALQHSF 6uip C 3.7 BS01 Q8J C 1 I165 A186 K188 F238 E239 L241 N292 L294 V306 D307 I31 A47 K49 F90 E91 L93 N141 L143 V155 D156 D287 K289 N292 D307 S324 D136 K138 N141 D156 S164 2.7.11.23,2.7.12.1 0004672,0004712,0005524,0006468,0046777 IC50=6.2nM Q13627 32077280 501 KERKVYNDGYDDDNYDYIVKNGEKYEIDSLIGKGSFGQVVKAYDWVAIKIIKNKKAFLNQAQIEVRLLELMNKHIVHRHFMFRNHLCLVFEMLSYNLYDLLRNTNFRGVSLNLTRKFAQQMCTALLFLATPIIHCDLKPENILLCNPKRSAIKIVDFGYQYIQSRFYRSPEVLLGMPYDLAIDMWSLGCILVEMHTGEPLFSGANEVDQMNKIVEVLGIPPAHILDQAPKARKFFEKLPDGTWNLKKTREYKPPGTRKLHNILGVETGGPGGRRVADYLKFKDLILRMLDYDPKTRIQPYYALQHS